JP2021527640A5 - - Google Patents

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Publication number
JP2021527640A5
JP2021527640A5 JP2020568439A JP2020568439A JP2021527640A5 JP 2021527640 A5 JP2021527640 A5 JP 2021527640A5 JP 2020568439 A JP2020568439 A JP 2020568439A JP 2020568439 A JP2020568439 A JP 2020568439A JP 2021527640 A5 JP2021527640 A5 JP 2021527640A5
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JP
Japan
Prior art keywords
seq
solvate
salt
indicated
chain variable
Prior art date
Application number
JP2020568439A
Other languages
English (en)
Japanese (ja)
Other versions
JPWO2019243159A5 (https=
JP2021527640A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2019/065517 external-priority patent/WO2019243159A1/de
Publication of JP2021527640A publication Critical patent/JP2021527640A/ja
Publication of JPWO2019243159A5 publication Critical patent/JPWO2019243159A5/ja
Publication of JP2021527640A5 publication Critical patent/JP2021527640A5/ja
Pending legal-status Critical Current

Links

JP2020568439A 2018-06-18 2019-06-13 酵素的に切断可能なリンカーおよび改善された活性プロファイルを有する、cxcr5に対して向けられるバインダー/活性薬剤複合体 Pending JP2021527640A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18178299 2018-06-18
EP18178299.6 2018-06-18
PCT/EP2019/065517 WO2019243159A1 (de) 2018-06-18 2019-06-13 Gegen cxcr5 gerichtete binder-wirkstoff-konjugate mit enzymatisch spaltbaren linkern und verbessertem wirkungsprofil

Publications (3)

Publication Number Publication Date
JP2021527640A JP2021527640A (ja) 2021-10-14
JPWO2019243159A5 JPWO2019243159A5 (https=) 2022-06-21
JP2021527640A5 true JP2021527640A5 (https=) 2022-06-21

Family

ID=62705502

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020568439A Pending JP2021527640A (ja) 2018-06-18 2019-06-13 酵素的に切断可能なリンカーおよび改善された活性プロファイルを有する、cxcr5に対して向けられるバインダー/活性薬剤複合体

Country Status (14)

Country Link
US (1) US20210275686A1 (https=)
EP (1) EP3806908A1 (https=)
JP (1) JP2021527640A (https=)
KR (1) KR20210033470A (https=)
CN (1) CN112601553A (https=)
AU (1) AU2019289506A1 (https=)
BR (1) BR112020025718A2 (https=)
CA (1) CA3103327A1 (https=)
EA (1) EA202190059A1 (https=)
IL (1) IL279400A (https=)
MA (1) MA71421A (https=)
MX (1) MX2020013832A (https=)
SG (1) SG11202012608VA (https=)
WO (1) WO2019243159A1 (https=)

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RU2018102358A (ru) 2015-06-23 2019-07-25 Байер Фарма Акциенгезельшафт Нацеленные конъюгаты ksp ингибиторов
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JP7066714B2 (ja) 2016-12-21 2022-05-13 バイエル・ファルマ・アクティエンゲゼルシャフト 酵素的に切断可能な基を有する抗体薬物コンジュゲート(adc)
CA3047491A1 (en) 2016-12-21 2018-06-28 Bayer Aktiengesellschaft Prodrugs of cytotoxic active agents having enzymatically cleavable groups
JP7030811B2 (ja) 2016-12-21 2022-03-07 バイエル・ファルマ・アクティエンゲゼルシャフト Ksp阻害剤を有する特異的抗体-薬物コンジュゲート(adc)
TW202216771A (zh) 2020-06-26 2022-05-01 德商拜耳廠股份有限公司 用於治療應用之ccr8抗體
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