JP2021527071A5 - - Google Patents

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Publication number
JP2021527071A5
JP2021527071A5 JP2020568471A JP2020568471A JP2021527071A5 JP 2021527071 A5 JP2021527071 A5 JP 2021527071A5 JP 2020568471 A JP2020568471 A JP 2020568471A JP 2020568471 A JP2020568471 A JP 2020568471A JP 2021527071 A5 JP2021527071 A5 JP 2021527071A5
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JP
Japan
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group
pharmaceutical composition
composition according
formula
alkyl
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JP2020568471A
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English (en)
Japanese (ja)
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JP2021527071A (ja
JP7445609B2 (ja
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Priority claimed from PCT/EP2019/064886 external-priority patent/WO2019234197A1/en
Publication of JP2021527071A publication Critical patent/JP2021527071A/ja
Publication of JP2021527071A5 publication Critical patent/JP2021527071A5/ja
Application granted granted Critical
Publication of JP7445609B2 publication Critical patent/JP7445609B2/ja
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JP2020568471A 2018-06-06 2019-06-06 Epac阻害剤としてのチエノ[2,3-b]ピリジン誘導体及びその医薬用途 Active JP7445609B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18305685 2018-06-06
EP18305685.2 2018-06-06
PCT/EP2019/064886 WO2019234197A1 (en) 2018-06-06 2019-06-06 Thieno[2,3-b]pyridine derivatives as epac inhibitors and their pharmaceutical uses

Publications (3)

Publication Number Publication Date
JP2021527071A JP2021527071A (ja) 2021-10-11
JP2021527071A5 true JP2021527071A5 (https=) 2023-11-16
JP7445609B2 JP7445609B2 (ja) 2024-03-07

Family

ID=62715982

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020568471A Active JP7445609B2 (ja) 2018-06-06 2019-06-06 Epac阻害剤としてのチエノ[2,3-b]ピリジン誘導体及びその医薬用途

Country Status (6)

Country Link
US (1) US20210230179A1 (https=)
EP (1) EP3801511A1 (https=)
JP (1) JP7445609B2 (https=)
KR (1) KR20210057704A (https=)
CN (1) CN112638382B (https=)
WO (1) WO2019234197A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4072547A1 (en) * 2019-12-13 2022-10-19 Institut National De La Sante Et De La Recherche Medicale - Inserm Epac1 inhibitors for the treatment of idiopathic pulmonary fibrosis
WO2021250231A1 (en) * 2020-06-12 2021-12-16 INSERM (Institut National de la Santé et de la Recherche Médicale) Thienopyridine derivatives for use in the treatment of coronavirus infection

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60325051D1 (de) * 2002-06-06 2009-01-15 Boehringer Ingelheim Pharma SUBSTITUIERTE 3-AMINO-THIENO(2,3-b)PYRIDINE-2-AMIDE UND HERSTELLUNGSVERFAHREN SOWIE DEREN VERWENDUNG
AU2007275221A1 (en) * 2006-07-20 2008-01-24 Allen J. Borchardt Benzothiophene inhibitors of RHO kinase
US20110077250A1 (en) * 2009-06-26 2011-03-31 Ryder Sean Compounds for modulating rna binding proteins and uses therefor
US9751838B2 (en) 2012-10-02 2017-09-05 Institut National De La Sante Et De La Recherche Medicale (Inserm) Tetrahydroquinoline derivatives and their use as Epac inhibitors
EP2928470A4 (en) * 2012-12-07 2015-12-16 Siga Technologies Inc THIENOPYRIDINE DERIVATIVES FOR THE TREATMENT AND PREVENTION OF DENGUE VIRUS INFECTIONS
AU2014342811B2 (en) 2013-10-15 2019-01-03 Board Of Regents Of The University Of Texas System Compositions and methods of modulating short-chain dehydrogenase activity

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