JP2021523179A5 - - Google Patents
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- Publication number
- JP2021523179A5 JP2021523179A5 JP2020563698A JP2020563698A JP2021523179A5 JP 2021523179 A5 JP2021523179 A5 JP 2021523179A5 JP 2020563698 A JP2020563698 A JP 2020563698A JP 2020563698 A JP2020563698 A JP 2020563698A JP 2021523179 A5 JP2021523179 A5 JP 2021523179A5
- Authority
- JP
- Japan
- Prior art keywords
- cycloalkyl
- alkyl
- hydrogen
- linear
- group
- Prior art date
Links
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024011236A JP7629123B2 (ja) | 2018-05-11 | 2024-01-29 | ５－ヒドロキシトリプタミン受容体７の調節物質としての新規官能化ラクタムおよびその使用方法 |
| JP2025013946A JP2025061975A (ja) | 2018-05-11 | 2025-01-30 | ５－ヒドロキシトリプタミン受容体７の調節物質としての新規官能化ラクタムおよびその使用方法 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862670116P | 2018-05-11 | 2018-05-11 | |
| US62/670,116 | 2018-05-11 | ||
| PCT/US2019/031824 WO2019217890A1 (en) | 2018-05-11 | 2019-05-10 | Novel functionalized lactams as modulators of the 5-hydroxytryptamine receptor 7 and their method of use |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024011236A Division JP7629123B2 (ja) | 2018-05-11 | 2024-01-29 | ５－ヒドロキシトリプタミン受容体７の調節物質としての新規官能化ラクタムおよびその使用方法 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2021523179A JP2021523179A (ja) | 2021-09-02 |
| JPWO2019217890A5 JPWO2019217890A5 (https=) | 2022-05-17 |
| JP2021523179A5 true JP2021523179A5 (https=) | 2022-05-17 |
| JP7429652B2 JP7429652B2 (ja) | 2024-02-08 |
Family
ID=66655471
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020563698A Active JP7429652B2 (ja) | 2018-05-11 | 2019-05-10 | ５－ヒドロキシトリプタミン受容体７の調節物質としての新規官能化ラクタムおよびその使用方法 |
| JP2024011236A Active JP7629123B2 (ja) | 2018-05-11 | 2024-01-29 | ５－ヒドロキシトリプタミン受容体７の調節物質としての新規官能化ラクタムおよびその使用方法 |
| JP2025013946A Pending JP2025061975A (ja) | 2018-05-11 | 2025-01-30 | ５－ヒドロキシトリプタミン受容体７の調節物質としての新規官能化ラクタムおよびその使用方法 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024011236A Active JP7629123B2 (ja) | 2018-05-11 | 2024-01-29 | ５－ヒドロキシトリプタミン受容体７の調節物質としての新規官能化ラクタムおよびその使用方法 |
| JP2025013946A Pending JP2025061975A (ja) | 2018-05-11 | 2025-01-30 | ５－ヒドロキシトリプタミン受容体７の調節物質としての新規官能化ラクタムおよびその使用方法 |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US12559494B2 (https=) |
| EP (1) | EP3790859A1 (https=) |
| JP (3) | JP7429652B2 (https=) |
| KR (1) | KR20210020182A (https=) |
| CN (2) | CN112437768B (https=) |
| AU (2) | AU2019267846B2 (https=) |
| BR (1) | BR112020023072A2 (https=) |
| CA (1) | CA3110799A1 (https=) |
| EA (1) | EA202092328A1 (https=) |
| IL (3) | IL317778A (https=) |
| MA (1) | MA52567A (https=) |
| MX (2) | MX2020012030A (https=) |
| TW (2) | TW202523659A (https=) |
| WO (1) | WO2019217890A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2970223B1 (en) | 2013-03-11 | 2020-04-15 | Temple University Of The Commonwealth System Of Higher Education | Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
| US10544117B2 (en) | 2014-09-10 | 2020-01-28 | Temple University—Of the Commonwealth System of Higher Education | 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
| AU2017361078B2 (en) | 2016-11-15 | 2022-01-06 | Praeventix, Llc | Novel modulators of the 5-hydroxytryptamine receptor 7 and their method of use |
| MA49019A (fr) | 2017-03-21 | 2020-02-05 | Univ Temple | Nouveaux modulateurs du récepteur sigma 2 et leur procédé d'utilisation |
| MA49017A (fr) | 2017-03-21 | 2020-02-05 | Univ Temple | Modulateurs du récepteur 7 de la 5-hydroxytryptamine et utilisation de ces derniers en tant qu'agents thérapeutiques |
| EA202092328A1 (ru) | 2018-05-11 | 2021-04-08 | Темпл Юниверсити-Оф Зэ Коммонвелс Систем Оф Хаер Эдьюкейшн | Новые функционализированные лактамы в качестве модуляторов 5-гидрокситриптаминового рецептора 7 и способ их применения |
| GB201809295D0 (en) * | 2018-06-06 | 2018-07-25 | Institute Of Cancer Res Royal Cancer Hospital | Lox inhibitors |
| JP7730811B2 (ja) * | 2019-11-13 | 2025-08-28 | テンプル・ユニバーシティ－オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション | ５－ヒドロキシトリプタミン受容体７の調節因子としての新規官能化ラクタムおよびその使用方法 |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2647785B1 (fr) * | 1989-05-31 | 1991-09-06 | Adir | Nouveaux derives de la pyrrolidone, leur procede de preparation et les compositions pharmaceutiques les renfermant |
| DE4127404A1 (de) * | 1991-08-19 | 1993-02-25 | Thomae Gmbh Dr K | Cyclische iminoderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung |
| GB9912701D0 (en) * | 1999-06-01 | 1999-08-04 | Smithkline Beecham Plc | Novel compounds |
| CA2440803A1 (en) * | 2001-03-07 | 2002-09-12 | Pfizer Products Inc. | Modulators of chemokine receptor activity |
| JP4203235B2 (ja) | 2001-07-05 | 2008-12-24 | 日本板硝子株式会社 | ガラスパネル |
| TWI319387B (en) | 2002-04-05 | 2010-01-11 | Astrazeneca Ab | Benzamide derivatives |
| MXPA05008137A (es) | 2003-01-31 | 2005-09-30 | Pfizer Prod Inc | Antagonistas y agonistas de 5ht7. |
| JP2006025227A (ja) | 2004-07-08 | 2006-01-26 | Sony Corp | 情報処理装置、情報処理方法、およびプログラム、並びに記録媒体 |
| EP1875899A1 (en) | 2006-06-29 | 2008-01-09 | Laboratorios Del Dr. Esteve, S.A. | Use of 5HT7 receptor agonists for the treatment of pain |
| CA2699674C (en) | 2007-10-12 | 2013-07-16 | Eli Lilly And Company | 5-ht7 receptor antagonists |
| EP2341912B1 (en) | 2008-09-05 | 2014-01-22 | Supernus Pharmaceuticals, Inc. | Method of treatment of attention deficit/hyperactivity disorder (adhd) |
| WO2010069390A1 (en) | 2008-12-19 | 2010-06-24 | Nokia Siemens Networks Oy | Method and device for data processing in an udwdm network and communication system comprising such device |
| GB201002563D0 (en) | 2010-02-15 | 2010-03-31 | Cambridge Entpr Ltd | Compounds |
| US20130287705A1 (en) | 2010-11-03 | 2013-10-31 | Mcmaster University | Method of treating mucosal inflammation |
| CN103570722A (zh) | 2012-07-19 | 2014-02-12 | 中国科学院上海药物研究所 | 稠环哒嗪酮类化合物及其制备方法和用途 |
| WO2014085413A1 (en) | 2012-11-28 | 2014-06-05 | Temple University - Of The Commonwealth System Of Higher Education | Disubstituted oxazolidin-2-ones 5-hydroxytryptamine receptor 2b activity modulators |
| EP2970223B1 (en) * | 2013-03-11 | 2020-04-15 | Temple University Of The Commonwealth System Of Higher Education | Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
| US10544117B2 (en) | 2014-09-10 | 2020-01-28 | Temple University—Of the Commonwealth System of Higher Education | 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
| US20180221365A1 (en) | 2015-05-12 | 2018-08-09 | Temple University-Of The Commonwealth System Of Higher Education | Novel sigma-2 receptor binders and their method of use |
| AU2017361078B2 (en) | 2016-11-15 | 2022-01-06 | Praeventix, Llc | Novel modulators of the 5-hydroxytryptamine receptor 7 and their method of use |
| MA49019A (fr) * | 2017-03-21 | 2020-02-05 | Univ Temple | Nouveaux modulateurs du récepteur sigma 2 et leur procédé d'utilisation |
| MA49017A (fr) * | 2017-03-21 | 2020-02-05 | Univ Temple | Modulateurs du récepteur 7 de la 5-hydroxytryptamine et utilisation de ces derniers en tant qu'agents thérapeutiques |
| EA202092328A1 (ru) | 2018-05-11 | 2021-04-08 | Темпл Юниверсити-Оф Зэ Коммонвелс Систем Оф Хаер Эдьюкейшн | Новые функционализированные лактамы в качестве модуляторов 5-гидрокситриптаминового рецептора 7 и способ их применения |
| CN110272425B (zh) | 2018-07-02 | 2022-11-04 | 广东东阳光药业有限公司 | 吡啶酰基八氢吡咯并[3,4-c]吡咯衍生物及其用途 |
| WO2021097117A2 (en) | 2019-11-13 | 2021-05-20 | Temple University-Of The Commonwealth System Of Higher Education | Novel functionalized lactones as modulators of the 5-hydroxytryptamine receptor 7 and their method of use |
| JP7730811B2 (ja) | 2019-11-13 | 2025-08-28 | テンプル・ユニバーシティ－オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション | ５－ヒドロキシトリプタミン受容体７の調節因子としての新規官能化ラクタムおよびその使用方法 |
-
2019
- 2019-05-10 EA EA202092328A patent/EA202092328A1/ru unknown
- 2019-05-10 AU AU2019267846A patent/AU2019267846B2/en active Active
- 2019-05-10 MA MA052567A patent/MA52567A/fr unknown
- 2019-05-10 KR KR1020207035307A patent/KR20210020182A/ko not_active Ceased
- 2019-05-10 US US17/054,468 patent/US12559494B2/en active Active
- 2019-05-10 WO PCT/US2019/031824 patent/WO2019217890A1/en not_active Ceased
- 2019-05-10 EP EP19726837.8A patent/EP3790859A1/en active Pending
- 2019-05-10 MX MX2020012030A patent/MX2020012030A/es unknown
- 2019-05-10 CA CA3110799A patent/CA3110799A1/en active Pending
- 2019-05-10 TW TW113132100A patent/TW202523659A/zh unknown
- 2019-05-10 IL IL317778A patent/IL317778A/en unknown
- 2019-05-10 TW TW108116303A patent/TWI856012B/zh active
- 2019-05-10 CN CN201980046137.1A patent/CN112437768B/zh active Active
- 2019-05-10 CN CN202510743117.7A patent/CN120365202A/zh active Pending
- 2019-05-10 BR BR112020023072-3A patent/BR112020023072A2/pt unknown
- 2019-05-10 IL IL324877A patent/IL324877A/en unknown
- 2019-05-10 JP JP2020563698A patent/JP7429652B2/ja active Active
-
2020
- 2020-11-05 IL IL278523A patent/IL278523B1/en unknown
- 2020-11-10 MX MX2024008100A patent/MX2024008100A/es unknown
-
2024
- 2024-01-29 JP JP2024011236A patent/JP7629123B2/ja active Active
- 2024-12-10 AU AU2024278241A patent/AU2024278241A1/en active Pending
-
2025
- 2025-01-30 JP JP2025013946A patent/JP2025061975A/ja active Pending
- 2025-11-14 US US19/390,312 patent/US20260070908A1/en active Pending
- 2025-11-14 US US19/390,298 patent/US20260070907A1/en active Pending
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