MXPA05008137A - Antagonistas y agonistas de 5ht7. - Google Patents
Antagonistas y agonistas de 5ht7.Info
- Publication number
- MXPA05008137A MXPA05008137A MXPA05008137A MXPA05008137A MXPA05008137A MX PA05008137 A MXPA05008137 A MX PA05008137A MX PA05008137 A MXPA05008137 A MX PA05008137A MX PA05008137 A MXPA05008137 A MX PA05008137A MX PA05008137 A MXPA05008137 A MX PA05008137A
- Authority
- MX
- Mexico
- Prior art keywords
- user
- questions
- fsd
- sexual function
- assessment
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/335—Radicals substituted by nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/14—Radicals substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
- Medical Treatment And Welfare Office Work (AREA)
- Management, Administration, Business Operations System, And Electronic Commerce (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyrrole Compounds (AREA)
Abstract
La presente invencion se refiere a compuestos de formula I, (ver formula (I)), y las sales farmaceuticamente aceptables de los mismos; estos compuestos son utiles como agentes psicoterapeuticos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US44436203P | 2003-01-31 | 2003-01-31 | |
PCT/IB2004/000172 WO2004067703A2 (en) | 2003-01-31 | 2004-01-20 | 5ht7 antagonists and inverse agonists |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA05008137A true MXPA05008137A (es) | 2005-09-30 |
Family
ID=32825411
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA05008137A MXPA05008137A (es) | 2003-01-31 | 2004-01-20 | Antagonistas y agonistas de 5ht7. |
Country Status (7)
Country | Link |
---|---|
US (1) | US20040229874A1 (es) |
EP (1) | EP1592772A2 (es) |
JP (1) | JP2006516604A (es) |
BR (1) | BRPI0406704A (es) |
CA (1) | CA2514656A1 (es) |
MX (1) | MXPA05008137A (es) |
WO (1) | WO2004067703A2 (es) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA200801812A1 (ru) * | 2003-09-17 | 2009-06-30 | Янссен Фармацевтика Н.В. | Сопряженные гетероциклические соединения |
US7598255B2 (en) * | 2005-08-04 | 2009-10-06 | Janssen Pharmaceutica Nv | Pyrimidine compounds as serotonin receptor modulators |
US8093279B2 (en) | 2005-12-13 | 2012-01-10 | Gillian Reed, legal representative | Compound |
GB0525323D0 (en) | 2005-12-13 | 2006-01-18 | Sterix Ltd | Compound |
EA016529B1 (ru) | 2007-05-11 | 2012-05-30 | Эли Лилли Энд Компани | 2-[4-(пиразол-4-илалкил)пиперазин-1-ил]-3-фенилпиразины и -пиридины и 3-[4-(пиразол-4-илалкил)пиперазин-1-ил]-2-фенилпиридины в качестве антагонистов рецепторов 5-ht |
TW200914020A (en) | 2007-08-28 | 2009-04-01 | Lilly Co Eli | Substituted piperazinyl pyrazines and pyridines as 5-HT7 receptor antagonists |
DK2201002T3 (da) * | 2007-10-12 | 2012-04-10 | Lilly Co Eli | 5-HT7-receptorantagonister |
US10154988B2 (en) | 2012-11-14 | 2018-12-18 | The Johns Hopkins University | Methods and compositions for treating schizophrenia |
EP3738955A1 (en) | 2013-03-11 | 2020-11-18 | Temple University Of The Commonwealth System Of Higher Education | Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
WO2016040554A1 (en) | 2014-09-10 | 2016-03-17 | Temple University-Of The Commonwealth System Of Higher Education | Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
CN105906614A (zh) * | 2016-05-12 | 2016-08-31 | 山东罗欣药业集团股份有限公司 | 一种奥美沙坦酯的制备方法 |
IL291029B2 (en) | 2016-11-15 | 2024-06-01 | Univ Temple | New modulators of 5-hydroxytryptamine receptor 7 and a method of using them |
JP7365238B2 (ja) | 2017-03-21 | 2023-10-19 | テンプル・ユニバーシティ-オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション | 5-ヒドロキシトリプタミン受容体7調節物質および治療剤としてのその使用 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US147200A (en) * | 1874-02-03 | Improvement in spinning-wheels | ||
MX18467A (es) * | 1988-11-23 | 1993-07-01 | Pfizer | Agentes terapeuticos de quinuclidinas |
US5232929A (en) * | 1990-11-28 | 1993-08-03 | Pfizer Inc. | 3-aminopiperidine derivatives and related nitrogen containing heterocycles and pharmaceutical compositions and use |
US6159979A (en) * | 1997-04-18 | 2000-12-12 | Smithkline Beecham P.L.C. | Bicyclic aryl or a bicyclic heterocyclic ring containing compounds having a combined 5HT1A, 5HT1B and 5HT1D receptor antagonistic activity |
DE60011269T2 (de) * | 1999-08-12 | 2005-06-23 | Nps Allelix Corp., Mississauga | Azaidole mit serotonin rezeptor affinität |
SE0004245D0 (sv) * | 2000-11-20 | 2000-11-20 | Pharmacia Ab | Novel compounds and their use |
-
2004
- 2004-01-20 BR BR0406704-5A patent/BRPI0406704A/pt not_active IP Right Cessation
- 2004-01-20 JP JP2006502361A patent/JP2006516604A/ja active Pending
- 2004-01-20 CA CA002514656A patent/CA2514656A1/en not_active Abandoned
- 2004-01-20 WO PCT/IB2004/000172 patent/WO2004067703A2/en not_active Application Discontinuation
- 2004-01-20 MX MXPA05008137A patent/MXPA05008137A/es not_active Application Discontinuation
- 2004-01-20 EP EP04703447A patent/EP1592772A2/en not_active Withdrawn
- 2004-01-27 US US10/766,741 patent/US20040229874A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
BRPI0406704A (pt) | 2005-12-20 |
WO2004067703A2 (en) | 2004-08-12 |
WO2004067703A3 (en) | 2004-11-04 |
US20040229874A1 (en) | 2004-11-18 |
EP1592772A2 (en) | 2005-11-09 |
CA2514656A1 (en) | 2004-08-12 |
JP2006516604A (ja) | 2006-07-06 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
WO2004063864A3 (en) | Method and system for computerized sexual function assessment of female users | |
Sanson-Fisher et al. | Adaptation and validation of the SF-36 Health Survey for use in Australia | |
Amorim et al. | Virtual reality therapy for rehabilitation of balance in the elderly: a systematic review and META-analysis | |
Sutton et al. | Eliciting salient beliefs in research on the theory of planned behaviour: The effect of question wording | |
Hanin et al. | Performance affect in junior ice hockey players: An application of the individual zones of optimal functioning model | |
Corbetta et al. | Rehabilitation that incorporates virtual reality is more effective than standard rehabilitation for improving walking speed, balance and mobility after stroke: a systematic review | |
Lenker et al. | A review of conceptual models for assistive technology outcomes research and practice | |
Mayer et al. | Changes in health behaviors of older adults: the San Diego Medicare Preventive Health Project | |
MXPA05008137A (es) | Antagonistas y agonistas de 5ht7. | |
Lin et al. | Assessing the stroke-specific quality of life for outcome measurement in stroke rehabilitation: minimal detectable change and clinically important difference | |
Lenert et al. | Public preferences for health states with schizophrenia and a mapping function to estimate utilities from positive and negative symptom scale scores | |
Choi et al. | The efficacy of female condom skills training in HIV risk reduction among women: a randomized controlled trial | |
Thomas et al. | Disordered eating and injuries among adolescent ballet dancers | |
Dennerstein et al. | Evaluation of a short scale to assess female sexual functioning | |
Palmcrantz et al. | An interactive distance solution for stroke rehabilitation in the home setting–A feasibility study | |
Abudarham et al. | Same critical features are used for identification of familiarized and unfamiliar faces | |
Learman et al. | No differences in outcomes in people with low back pain who met the clinical prediction rule for lumbar spine manipulation when a pragmatic non-thrust manipulation was used as the comparator | |
Versluys et al. | The influence of leg-to-body ratio, arm-to-body ratio and intra-limb ratio on male human attractiveness | |
Corcoran | Interpersonal stress and burnout: Unraveling the role of empathy | |
Wright et al. | Metronome‐Cued Stepping in Place after Hemiparetic Stroke: Comparison of a One‐and Two‐Tone Beat | |
Chan et al. | Judo‐based exercise programs to improve health outcomes in middle‐aged and older adults with no judo experience: A scoping review | |
Rosenblum et al. | Reliability and concurrent validity of the narrow path walking test in persons with multiple sclerosis | |
Veisani et al. | Health related quality of life in the female-headed households | |
Nyarko et al. | Prevalence and predictors of hypertension history among Ghanaian men | |
Montilla et al. | Effectiveness of virtual reality in balance training for fall prevention in older adults: systematic review |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |