JP2021519294A5 - - Google Patents

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Publication number
JP2021519294A5
JP2021519294A5 JP2020551599A JP2020551599A JP2021519294A5 JP 2021519294 A5 JP2021519294 A5 JP 2021519294A5 JP 2020551599 A JP2020551599 A JP 2020551599A JP 2020551599 A JP2020551599 A JP 2020551599A JP 2021519294 A5 JP2021519294 A5 JP 2021519294A5
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JP
Japan
Prior art keywords
methyl
difluoromethoxy
fluoro
benzamide
group
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JP2020551599A
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English (en)
Japanese (ja)
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JP7279067B2 (ja
JP2021519294A (ja
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Priority claimed from PCT/JP2019/014901 external-priority patent/WO2019189945A1/en
Publication of JP2021519294A publication Critical patent/JP2021519294A/ja
Publication of JP2021519294A5 publication Critical patent/JP2021519294A5/ja
Application granted granted Critical
Publication of JP7279067B2 publication Critical patent/JP7279067B2/ja
Active legal-status Critical Current
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JP2020551599A 2018-03-28 2019-03-27 複素環化合物及びその用途 Active JP7279067B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2018062939 2018-03-28
JP2018062939 2018-03-28
PCT/JP2019/014901 WO2019189945A1 (en) 2018-03-28 2019-03-27 Heterocyclic compound and use thereof

Publications (3)

Publication Number Publication Date
JP2021519294A JP2021519294A (ja) 2021-08-10
JP2021519294A5 true JP2021519294A5 (enExample) 2022-04-01
JP7279067B2 JP7279067B2 (ja) 2023-05-22

Family

ID=66397395

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020551599A Active JP7279067B2 (ja) 2018-03-28 2019-03-27 複素環化合物及びその用途

Country Status (17)

Country Link
US (2) US10807987B2 (enExample)
EP (1) EP3774800B1 (enExample)
JP (1) JP7279067B2 (enExample)
KR (1) KR20200136957A (enExample)
CN (1) CN111936495A (enExample)
AR (1) AR115020A1 (enExample)
AU (1) AU2019241765B2 (enExample)
BR (1) BR112020018238A2 (enExample)
CA (1) CA3100133A1 (enExample)
EA (1) EA202092294A1 (enExample)
ES (1) ES3006012T3 (enExample)
IL (1) IL276912A (enExample)
MA (1) MA52214A (enExample)
MX (1) MX2020010148A (enExample)
SG (1) SG11202008519RA (enExample)
TW (1) TW202003519A (enExample)
WO (1) WO2019189945A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11230541B2 (en) 2017-07-28 2022-01-25 Takeda Pharmaceutical Company Limited Heterocyclic compound
EP3774800B1 (en) * 2018-03-28 2024-11-13 Takeda Pharmaceutical Company Limited Heterocyclic compound and use thereof
US12637418B2 (en) 2019-01-24 2026-05-26 Takeda Pharmaceutical Company Limited Heterocyclic compounds as antagonist of NMDA
JP2021050161A (ja) 2019-09-25 2021-04-01 武田薬品工業株式会社 複素環化合物及びその用途
JP2021080177A (ja) 2019-11-14 2021-05-27 武田薬品工業株式会社 複素環化合物及びその用途

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492382A1 (fr) * 1980-10-22 1982-04-23 Synthelabo Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique
US5252563A (en) * 1991-12-19 1993-10-12 G. D. Searle & Company 5,6,7,8-tetrahydro-imidazo[1,2-a]pyrimidine compounds for treatment of neurotoxic injury
JP3439551B2 (ja) * 1994-11-08 2003-08-25 富士写真フイルム株式会社 ハロゲン化銀写真感光材料
CA2214247C (en) 1995-03-14 2004-02-10 Praecis Pharmaceuticals Incorporated Modulators of amyloid aggregation
EP1586584A1 (en) 1996-08-27 2005-10-19 Praecis Pharmaceuticals Incorporated Modulators of beta-amyloid peptide aggregation comprising D-amino acids
US6331640B1 (en) 1998-10-13 2001-12-18 Hoffmann-La Roche Inc. Diaminopropionic acid derivatives
EP1194449B1 (en) 1999-06-28 2010-09-22 Oklahoma Medical Research Foundation Inhibitors of memapsin 2 and use thereof
EP1390034A4 (en) * 2001-04-03 2005-07-13 Merck & Co Inc N-SUBSTITUTED NONARYL HETEROCYCLO AMIDYL-NMDA / NR2B ANTAGONISTS
JP2004161716A (ja) * 2002-11-15 2004-06-10 Takeda Chem Ind Ltd Jnk阻害剤
CA2521907A1 (en) * 2003-04-10 2004-10-21 Pfizer Inc. Bicyclic compounds as nr2b receptor antagonists
US20080234318A1 (en) 2005-08-31 2008-09-25 Kristjan Gudmundsson Chemical Compounds
AU2010210426B2 (en) * 2009-02-06 2015-06-11 Imago Pharmaceuticals, Inc. Inhibitors of Jun N-terminal kinase
US8404859B2 (en) 2011-03-16 2013-03-26 Hoffmann-La Roche Inc. Thiazole and thiophene compounds
EP2694509B1 (en) * 2011-04-05 2016-05-18 Pfizer Limited Pyrrolo[2,3-d]pyrimidine derivatives as inhibitors of tropomyosin-related kinases
FR2998892B1 (fr) 2012-12-04 2015-01-02 Pf Medicament Derives d'aminocyclobutane, leur procede de preparation et leur utilisation a titre de medicaments
US9243001B2 (en) 2013-03-15 2016-01-26 Epizyme, Inc. Substituted benzene compounds
US20160031907A1 (en) 2013-03-15 2016-02-04 Epizyme, Inc. Substituted Benzene Compounds
US10202376B2 (en) 2014-12-24 2019-02-12 Takeda Pharmaceutical Company Limited Heterocyclic compound
JP6827757B2 (ja) 2016-10-11 2021-02-10 鬼怒川ゴム工業株式会社 ウエザーストリップ取付用クリップ
US11230541B2 (en) 2017-07-28 2022-01-25 Takeda Pharmaceutical Company Limited Heterocyclic compound
EP3774800B1 (en) * 2018-03-28 2024-11-13 Takeda Pharmaceutical Company Limited Heterocyclic compound and use thereof
US12637418B2 (en) 2019-01-24 2026-05-26 Takeda Pharmaceutical Company Limited Heterocyclic compounds as antagonist of NMDA
WO2020196828A1 (ja) 2019-03-28 2020-10-01 武田薬品工業株式会社 含窒素複素環化合物

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