JP2021515775A5 - - Google Patents

Info

Publication number
JP2021515775A5
JP2021515775A5 JP2020547008A JP2020547008A JP2021515775A5 JP 2021515775 A5 JP2021515775 A5 JP 2021515775A5 JP 2020547008 A JP2020547008 A JP 2020547008A JP 2020547008 A JP2020547008 A JP 2020547008A JP 2021515775 A5 JP2021515775 A5 JP 2021515775A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
composition according
optionally substituted
group
cancer
Prior art date
Application number
JP2020547008A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021515775A (ja
JP7417530B2 (ja
JPWO2019173682A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/021300 external-priority patent/WO2019173682A1/en
Publication of JP2021515775A publication Critical patent/JP2021515775A/ja
Publication of JP2021515775A5 publication Critical patent/JP2021515775A5/ja
Publication of JPWO2019173682A5 publication Critical patent/JPWO2019173682A5/ja
Priority to JP2023170366A priority Critical patent/JP2023165998A/ja
Application granted granted Critical
Publication of JP7417530B2 publication Critical patent/JP7417530B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020547008A 2018-03-09 2019-03-08 優先投与される免疫増強薬 Active JP7417530B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023170366A JP2023165998A (ja) 2018-03-09 2023-09-29 優先投与される免疫増強薬

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862641003P 2018-03-09 2018-03-09
US62/641,003 2018-03-09
US201862700548P 2018-07-19 2018-07-19
US62/700,548 2018-07-19
PCT/US2019/021300 WO2019173682A1 (en) 2018-03-09 2019-03-08 Parenterally administered immune enhancing drugs

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023170366A Division JP2023165998A (ja) 2018-03-09 2023-09-29 優先投与される免疫増強薬

Publications (4)

Publication Number Publication Date
JP2021515775A JP2021515775A (ja) 2021-06-24
JP2021515775A5 true JP2021515775A5 (https=) 2022-03-16
JPWO2019173682A5 JPWO2019173682A5 (https=) 2022-03-16
JP7417530B2 JP7417530B2 (ja) 2024-01-18

Family

ID=67846288

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020547008A Active JP7417530B2 (ja) 2018-03-09 2019-03-08 優先投与される免疫増強薬
JP2023170366A Withdrawn JP2023165998A (ja) 2018-03-09 2023-09-29 優先投与される免疫増強薬

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023170366A Withdrawn JP2023165998A (ja) 2018-03-09 2023-09-29 優先投与される免疫増強薬

Country Status (8)

Country Link
US (1) US12433836B2 (https=)
EP (1) EP3761993A4 (https=)
JP (2) JP7417530B2 (https=)
KR (1) KR102822181B1 (https=)
CN (1) CN112004541A (https=)
AU (1) AU2019231781B2 (https=)
CA (1) CA3092585A1 (https=)
WO (1) WO2019173682A1 (https=)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE063388T2 (hu) 2016-01-08 2024-01-28 Arcus Biosciences Inc Ekto-5'-nukleotidáz modulátorok és ezek alkalmazása
US10881681B2 (en) * 2018-09-11 2021-01-05 Risen (Suzhou) Pharma Tech Co., Ltd. CD73 inhibitors and pharmaceutical uses thereof
US11530234B2 (en) 2018-09-11 2022-12-20 Risen (Suzhou) Pharma Tech Co., Ltd. CD73 inhibitors and pharmaceutical uses thereof
WO2020123772A1 (en) 2018-12-13 2020-06-18 Arcus Biosciences, Inc. Solid forms of a cd73 inhibitor and the use thereof
WO2020185859A1 (en) 2019-03-12 2020-09-17 Arcus Biosciences, Inc. Treatment of oncogene-driven cancers
US12310965B2 (en) 2019-03-29 2025-05-27 Arcus Biosciences, Inc. Treatment of cancer utilizing an identified adenosine fingerprint
TWI821559B (zh) * 2019-04-28 2023-11-11 大陸商上海和譽生物醫藥科技有限公司 一種cd73抑制劑,其製備方法和應用
TW202131932A (zh) * 2019-11-05 2021-09-01 美商博奥阿迪斯有限公司 作為cd73抑制劑的化合物
WO2021152548A1 (en) * 2020-01-30 2021-08-05 Benitah Salvador Aznar Combination therapy for treatment of cancer and cancer metastasis
TWI775313B (zh) 2020-02-18 2022-08-21 美商基利科學股份有限公司 抗病毒化合物
TWI794742B (zh) 2020-02-18 2023-03-01 美商基利科學股份有限公司 抗病毒化合物
AU2021224588B2 (en) 2020-02-18 2024-07-18 Gilead Sciences, Inc. Antiviral compounds
US11633416B1 (en) 2020-03-06 2023-04-25 Arcus Biosciences, Inc. Oral formulations of CD73 compounds
AU2021292195A1 (en) 2020-06-17 2023-01-05 Arcus Biosciences, Inc. Crystalline forms of a CD73 inhibitor and uses thereof
EP4323362B1 (en) 2021-04-16 2025-05-07 Gilead Sciences, Inc. Methods of preparing carbanucleosides using amides
WO2022237747A1 (zh) * 2021-05-11 2022-11-17 四川海思科制药有限公司 小分子cd73拮抗剂及其用途
AU2022328698B2 (en) 2021-08-18 2025-02-20 Gilead Sciences, Inc. Phospholipid compounds and methods of making and using the same
US12103943B2 (en) 2021-10-26 2024-10-01 Southern Research Institute Development of novel clofarabine analogs for cancer therapy
JP2025520300A (ja) * 2022-06-17 2025-07-03 上海森輝医薬有限公司 シクロペンチルアデノシン誘導体及びその医薬的使用
EP4604920A1 (en) * 2022-10-20 2025-08-27 Arcus Biosciences, Inc. Lyophilized formulations of cd73 compounds
CN117924394A (zh) * 2023-09-05 2024-04-26 厦门大学 核苷酸类化合物及其制备方法和应用、核素靶向探针及其制备方法和应用、药物组合物
CN117562915A (zh) * 2023-12-05 2024-02-20 中国药科大学 一种腺苷衍生物在制备预防、缓解或治疗纤维化疾病的药物中的应用
CN120285176A (zh) * 2025-04-25 2025-07-11 谈高 抗CD73单抗联合Adora1抑制剂在治疗肠纤维化中的应用

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5569650A (en) * 1993-06-11 1996-10-29 Sloan-Kettering Institute For Cancer Research C-nucleoside isosters of analogs thereof and pharmaceutical compositions
WO2001049287A1 (en) 1999-12-30 2001-07-12 Sugen, Inc. 3-heteroarylidenyl-2-indolinone compounds for modulating protein kinase activity and for use in cancer chemotherapy
US9090697B2 (en) 2013-03-15 2015-07-28 Bayer Healthcare Llc Methods for treating bleeding disorders
WO2015164573A1 (en) 2014-04-25 2015-10-29 Vitae Pharmaceuticals, Inc. Purine derivatives as cd73 inhibitors for the treatment of cancer
HUE063388T2 (hu) 2016-01-08 2024-01-28 Arcus Biosciences Inc Ekto-5'-nukleotidáz modulátorok és ezek alkalmazása
KR20230038311A (ko) * 2016-03-04 2023-03-17 브리스톨-마이어스 스큅 컴퍼니 항-cd73 항체와의 조합 요법
WO2018047139A1 (en) * 2016-09-12 2018-03-15 Aurigene Discovery Technologies Limited Compounds as modulators of tigit signalling pathway
CN110049767B (zh) 2016-10-03 2023-04-04 艾库斯生物科学有限公司 腺苷5′-核苷酸酶的抑制剂
EP3541396A4 (en) 2016-11-18 2020-07-22 Arcus Biosciences, Inc. CD73-MEDIATED IMMUNOSUPPRESSION INHIBITORS
TW202012637A (zh) * 2018-04-24 2020-04-01 瑞典商阿斯特捷利康公司 治療癌症之方法
WO2020123772A1 (en) * 2018-12-13 2020-06-18 Arcus Biosciences, Inc. Solid forms of a cd73 inhibitor and the use thereof

Similar Documents

Publication Publication Date Title
JP2021515775A5 (https=)
JPWO2019173682A5 (https=)
ES2981830T3 (es) Uso de riluzol, profármacos de riluzol o análogos de riluzol con inmunoterapias para tratar cánceres
JP2019518741A5 (https=)
JP2020508310A5 (https=)
JPWO2021085653A5 (https=)
US20230165859A1 (en) N-substituted indole derivatives
ES2946472T3 (es) Agente antitumoral y potenciador del efecto antitumoral
JP2021502423A5 (https=)
US20250281514A1 (en) Treatment of cancer patients having kras mutations
JP2008506710A5 (https=)
CN114728994A (zh) 芳基磷氧类化合物及其用途
US10829495B2 (en) Thieno-pyrimidine derivatives and uses thereof
TW202028182A (zh) 用於癌症治療之免疫調節之組合
TW201811323A (zh) 抗腫瘤劑、抗腫瘤效果增強劑及抗腫瘤用套組
US10744134B2 (en) Pharmaceutical composition for cancer immunotherapy and/or immunological activation containing diamino heterocyclic carboxamide compound as active ingredient
ES2440799T3 (es) Métodos para tratar cáncer resistente a los fármacos
US20230330081A1 (en) Pharmaceutical composition for treating tumors
CN114040765A (zh) 癌症免疫治疗佐剂
JPWO2018117196A1 (ja) がん幹細胞を標的とする医薬
RU2004135307A (ru) Производное эпотилона для лечения гепатомы и других раковых заболеваний
BR112020023866A2 (pt) Agonistas de tlr7
US20100098691A1 (en) Combination of benzimidazole anti-cancer agent and a second anti-cancer agent
JPWO2022076859A5 (https=)
JPWO2020142742A5 (https=)