JP2020529472A - ペプチド化合物の環化放出関連する出願の相互参照 - Google Patents

ペプチド化合物の環化放出関連する出願の相互参照 Download PDF

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JP2020529472A
JP2020529472A JP2020527859A JP2020527859A JP2020529472A JP 2020529472 A JP2020529472 A JP 2020529472A JP 2020527859 A JP2020527859 A JP 2020527859A JP 2020527859 A JP2020527859 A JP 2020527859A JP 2020529472 A JP2020529472 A JP 2020529472A
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compound
alkyl
acid
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JP2020529472A5 (enExample
Inventor
ラマセシャン マヘシュ
ラマセシャン マヘシュ
ボックス アンドリュー
ボックス アンドリュー
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サークル ファーマ，インコーポレイティド
サークル ファーマ，インコーポレイティド
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Publication of JP2020529472A publication Critical patent/JP2020529472A/ja
Publication of JP2020529472A5 publication Critical patent/JP2020529472A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/042—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers characterised by the nature of the carrier
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64—Cyclic peptides containing only normal peptide links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2020527859A 2017-07-28 2018-07-27 ペプチド化合物の環化放出関連する出願の相互参照 Pending JP2020529472A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762538477P 2017-07-28 2017-07-28
US62/538,477 2017-07-28
PCT/US2018/044182 WO2019023634A1 (en) 2017-07-28 2018-07-27 CYCLATIVE RELEASE OF PEPTIDE COMPOUNDS

Publications (2)

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JP2020529472A true JP2020529472A (ja) 2020-10-08
JP2020529472A5 JP2020529472A5 (enExample) 2021-09-09

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Family Applications (1)

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JP2020527859A Pending JP2020529472A (ja) 2017-07-28 2018-07-27 ペプチド化合物の環化放出関連する出願の相互参照

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Country Link
US (1) US11299513B2 (enExample)
EP (1) EP3658567A1 (enExample)
JP (1) JP2020529472A (enExample)
WO (1) WO2019023634A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112592382A (zh) * 2020-11-27 2021-04-02 安徽大学 一种树脂及其制备方法以及其在制备头尾环肽中的应用

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN120309693B (zh) * 2025-06-12 2025-09-16 杭州湃肽生化科技有限公司 一类环肽化合物及其制备方法和应用

Citations (1)

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JP2002525376A (ja) * 1998-09-25 2002-08-13 ザ ユニバーシティ オブ クイーンズランド アミド結合形成のための補助基

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GB2369823B (en) 1999-11-30 2003-06-04 Cyclacel Ltd Assays for cyclin-interacting compounds
GB9928323D0 (en) 1999-11-30 2000-01-26 Cyclacel Ltd Peptides
US20050153894A1 (en) 1999-11-30 2005-07-14 Cyclacel Limited p21 peptides
CN1592752A (zh) 2000-12-20 2005-03-09 诺瓦提斯公司 用于治疗癌症的e2f－1/细胞周期蛋白相互作用的抑制剂
US20040053849A1 (en) 2000-12-20 2004-03-18 Bair Kenneth Walter Inhibitors of the E2F-1/cyclin interaction for cancer therapy
US20040077549A1 (en) 2000-12-20 2004-04-22 Bair Kenneth Walter Inhibitors of the E2F-1/cyclin interaction for cancer therapy
JP2004269357A (ja) 2002-01-25 2004-09-30 Marine Biotechnol Inst Co Ltd 鉄と高い結合能を有する化合物およびその製造方法
WO2006105386A1 (en) 2005-03-30 2006-10-05 Genentech, Inc. Cdk2 inhibitors
WO2008000870A1 (es) 2006-06-19 2008-01-03 Fundación De La Comunidad Valenciana, Centro De Investigación Principe Felipe Compuestos orgánicos que inhiben la actividad catalítica del complejo ciclina a/kinasa 2 dependiente de ciclina mediante su unión a un nuevo sitio farmacofórico en la molécula de ciclina
US20100184684A1 (en) 2009-01-06 2010-07-22 C3 Jian, Inc. Antibacterial and antifungal peptides
US9376465B2 (en) 2012-03-27 2016-06-28 University Of South Carolina Cyclin based inhibitors of CDK2 and CDK4
US20140296484A1 (en) 2013-03-27 2014-10-02 University Of South Carolina Cyclin Based Inhibitors of CDK2 and CDK4
US10011635B2 (en) 2013-09-27 2018-07-03 H. Lee Moffitt Cancer Center And Research Institute, Inc. Cyclic peptide conjugates and methods of use
WO2017046229A1 (en) 2015-09-17 2017-03-23 Histide Ag Pharmaceutical association of growth factor receptor agonist and adhesion protein inhibitor for converting a neoplastic cell into a non-neoplastic cell and uses thereof
EP3349777B1 (en) 2015-09-17 2025-05-07 Histide AG Pharmaceutical association comprising a growth factor receptor agonist conjugated to a bioactive carrierfor converting a neoplastic cell into a non-neoplastic cell and uses thereof
EP3349782A2 (en) 2015-09-17 2018-07-25 Histide AG Pharmaceutical association comprising a growth factor receptor agonist conjugated to a bioactive carrier for converting a neoplastic cell into a non-neoplastic cell and uses thereof
KR20180052726A (ko) 2015-09-17 2018-05-18 히스티드 아게 신생물성 세포를 비-신생물성 세포로 전환시키기 위한 약제학적 회합물 및 이것의 용도
IL299622A (en) 2015-09-17 2023-03-01 Histide Ag A pharmaceutical composition containing a growth receptor agonist and an adhesion protein inhibitor for converting a neoplastic cell into a non-neoplastic cell and its uses
WO2017046226A2 (en) 2015-09-17 2017-03-23 Histide Ag Pharmaceutical association for converting a neoplastic cell into a non-neoplastic cell and uses thereof.

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002525376A (ja) * 1998-09-25 2002-08-13 ザ ユニバーシティ オブ クイーンズランド アミド結合形成のための補助基

Non-Patent Citations (6)

* Cited by examiner, † Cited by third party
Title
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS (2008) VOL.18, PP.4731-4735, JPN6022021031, ISSN: 0004959467 *
J. AM. CHEM. SOC. (1999) VOL.121, PP.3311-3320, JPN6022021028, ISSN: 0004959466 *
ORGANIC LETTERS (2005) VOL.7, NO.13, PP.2647-2650, JPN6022021026, ISSN: 0004959465 *
TETRAHEDRON (2006) VOL.62, PP.9533-9540, JPN6022021024, ISSN: 0004959463 *
TETRAHEDRON LETTERS (1999) VOL.40, PP.8197-8200, JPN6022021025, ISSN: 0004959464 *
有機合成化学 (1981) VOL.39, NO.4, PP.312-321, JPN6022021029, ISSN: 0004787206 *

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112592382A (zh) * 2020-11-27 2021-04-02 安徽大学 一种树脂及其制备方法以及其在制备头尾环肽中的应用

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US20200207803A1 (en) 2020-07-02
WO2019023634A1 (en) 2019-01-31
US11299513B2 (en) 2022-04-12
EP3658567A1 (en) 2020-06-03

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