JP2019535788A5 - - Google Patents

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Publication number
JP2019535788A5
JP2019535788A5 JP2019528512A JP2019528512A JP2019535788A5 JP 2019535788 A5 JP2019535788 A5 JP 2019535788A5 JP 2019528512 A JP2019528512 A JP 2019528512A JP 2019528512 A JP2019528512 A JP 2019528512A JP 2019535788 A5 JP2019535788 A5 JP 2019535788A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2019528512A
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Japanese (ja)
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JPWO2018098412A5 (https=
JP2019535788A (ja
JP7114591B2 (ja
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Priority claimed from PCT/US2017/063231 external-priority patent/WO2018098412A1/en
Publication of JP2019535788A publication Critical patent/JP2019535788A/ja
Publication of JP2019535788A5 publication Critical patent/JP2019535788A5/ja
Publication of JPWO2018098412A5 publication Critical patent/JPWO2018098412A5/ja
Application granted granted Critical
Publication of JP7114591B2 publication Critical patent/JP7114591B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2019528512A 2016-11-28 2017-11-27 Gsk-3阻害剤 Active JP7114591B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662426631P 2016-11-28 2016-11-28
US62/426,631 2016-11-28
PCT/US2017/063231 WO2018098412A1 (en) 2016-11-28 2017-11-27 Gsk-3 inhibitors

Publications (4)

Publication Number Publication Date
JP2019535788A JP2019535788A (ja) 2019-12-12
JP2019535788A5 true JP2019535788A5 (https=) 2022-03-01
JPWO2018098412A5 JPWO2018098412A5 (https=) 2022-03-01
JP7114591B2 JP7114591B2 (ja) 2022-08-08

Family

ID=60655130

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019528512A Active JP7114591B2 (ja) 2016-11-28 2017-11-27 Gsk-3阻害剤

Country Status (8)

Country Link
US (1) US10752609B2 (https=)
EP (1) EP3544613B1 (https=)
JP (1) JP7114591B2 (https=)
KR (1) KR102575990B1 (https=)
CN (1) CN110545817B (https=)
ES (1) ES2878078T3 (https=)
MA (1) MA46889A (https=)
WO (1) WO2018098412A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2850773T3 (es) * 2016-11-28 2021-08-31 Bristol Myers Squibb Co Piridincarboxamidas como inhibidores de GSK-3
WO2020132651A1 (en) 2018-12-20 2020-06-25 Amgen Inc. Kif18a inhibitors
EP3898616B1 (en) * 2018-12-20 2024-10-02 Amgen Inc. Heteroaryl amides useful as kif18a inhibitors
JP7676308B2 (ja) 2018-12-20 2025-05-14 アムジエン・インコーポレーテツド Kif18a阻害剤として有用なヘテロアリールアミド
US12540129B2 (en) 2019-08-02 2026-02-03 Amgen Inc. KIF18A inhibitors
WO2021026099A1 (en) 2019-08-02 2021-02-11 Amgen Inc. Kif18a inhibitors
CN116178281B (zh) * 2023-04-27 2023-07-21 中国药科大学 一种双功能免疫抑制剂及其制备方法和应用
EP4709712A1 (en) * 2023-05-10 2026-03-18 Blueprint Medicines Corporation Gsk3a inhibitors and methods of use thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0102438D0 (sv) 2001-07-05 2001-07-05 Astrazeneca Ab New compounds
JP5241834B2 (ja) * 2007-07-19 2013-07-17 メルク・シャープ・アンド・ドーム・コーポレーション プロテインキナーゼ阻害剤としての複素環アミド化合物
WO2012024179A1 (en) * 2010-08-18 2012-02-23 Merck Sharp & Dohme Corp. Substituted amide derivatives as dgat-1 inhibitors
CN105849098A (zh) * 2013-11-06 2016-08-10 百时美施贵宝公司 Gsk-3抑制剂
CN105849097A (zh) 2013-11-06 2016-08-10 百时美施贵宝公司 取代的吡啶衍生物用作gsk-3抑制剂
WO2016144792A1 (en) * 2015-03-06 2016-09-15 Alpharmagen, Llc Alpha 7 nicotinic acetylcholine receptor allosteric modulators, their derivatives and uses thereof
ES2850773T3 (es) 2016-11-28 2021-08-31 Bristol Myers Squibb Co Piridincarboxamidas como inhibidores de GSK-3

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