JP2019526628A - セニクリビロクメシレートの固体形態及びセニクリビロクメシレートの固体形態を製造するプロセス - Google Patents

セニクリビロクメシレートの固体形態及びセニクリビロクメシレートの固体形態を製造するプロセス Download PDF

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JP2019526628A
JP2019526628A JP2019531594A JP2019531594A JP2019526628A JP 2019526628 A JP2019526628 A JP 2019526628A JP 2019531594 A JP2019531594 A JP 2019531594A JP 2019531594 A JP2019531594 A JP 2019531594A JP 2019526628 A JP2019526628 A JP 2019526628A
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crystalline form
compound
msoh
acetonitrile
ethyl acetate
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JP2019526628A5 (https=
Inventor
パシット・フィアシヴォンサ
マーティン・イアン・クーパー
エマ・ケイ・シャープ
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トビラ セラピューティクス， インコーポレイテッド
トビラ セラピューティクス， インコーポレイテッド
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Publication of JP2019526628A publication Critical patent/JP2019526628A/ja
Publication of JP2019526628A5 publication Critical patent/JP2019526628A5/ja
Priority to JP2022113230A priority Critical patent/JP2022137223A/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01—Sulfonic acids
    • C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/03—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C309/04—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing only one sulfo group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2019531594A 2016-08-31 2017-08-30 セニクリビロクメシレートの固体形態及びセニクリビロクメシレートの固体形態を製造するプロセス Pending JP2019526628A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2022113230A JP2022137223A (ja) 2016-08-31 2022-07-14 セニクリビロクメシレートの固体形態及びセニクリビロクメシレートの固体形態を製造するプロセス

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662382153P 2016-08-31 2016-08-31
US62/382,153 2016-08-31
PCT/US2017/049400 WO2018045043A1 (en) 2016-08-31 2017-08-30 Solid forms of cenicriviroc mesylate and processes of making solid forms of cenicriviroc mesylate

Related Child Applications (1)

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JP2022113230A Division JP2022137223A (ja) 2016-08-31 2022-07-14 セニクリビロクメシレートの固体形態及びセニクリビロクメシレートの固体形態を製造するプロセス

Publications (2)

Publication Number Publication Date
JP2019526628A true JP2019526628A (ja) 2019-09-19
JP2019526628A5 JP2019526628A5 (https=) 2020-10-08

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JP2019531594A Pending JP2019526628A (ja) 2016-08-31 2017-08-30 セニクリビロクメシレートの固体形態及びセニクリビロクメシレートの固体形態を製造するプロセス
JP2022113230A Pending JP2022137223A (ja) 2016-08-31 2022-07-14 セニクリビロクメシレートの固体形態及びセニクリビロクメシレートの固体形態を製造するプロセス

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Country Status (13)

Country Link
US (1) US10301287B2 (https=)
EP (1) EP3506896A4 (https=)
JP (2) JP2019526628A (https=)
KR (1) KR20190057066A (https=)
CN (1) CN110167550A (https=)
AU (1) AU2017321594A1 (https=)
BR (1) BR112019003987A2 (https=)
CA (1) CA3034606A1 (https=)
MX (1) MX2019002057A (https=)
RU (1) RU2019109019A (https=)
SG (1) SG11201901438VA (https=)
TW (1) TW201823235A (https=)
WO (1) WO2018045043A1 (https=)

Cited By (1)

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JPWO2022177014A1 (https=) * 2021-02-22 2022-08-25

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WO2019238041A1 (zh) * 2018-06-12 2019-12-19 南京明德新药研发有限公司 一种丙烯酰胺类化合物的晶型及其制备方法
WO2019245517A1 (en) * 2018-06-18 2019-12-26 Hewlett-Packard Development Company, L.P. Three-dimensional printing
US11613670B2 (en) 2018-06-18 2023-03-28 Hewlett-Packard Development Company, L.P. Three-dimensional printing
US11298876B2 (en) 2018-06-19 2022-04-12 Hewlett-Packard Development Company, L.P. Three-dimensional printing
US11591486B2 (en) 2018-06-19 2023-02-28 Hewlett-Packard Development Company, L.P. Three-dimensional printing
US11426931B2 (en) 2018-06-19 2022-08-30 Hewlett-Packard Development Company, L.P. Three-dimensional printing
KR20210053921A (ko) * 2018-08-31 2021-05-12 에보니크 오퍼레이션즈 게엠베하 중합체 분말을 제조하는 방법
WO2021133811A1 (en) 2019-12-26 2021-07-01 Teva Pharmaceuticals International Gmbh Solid state forms of cenicriviroc and process for preparation thereof
US12466817B2 (en) 2020-05-22 2025-11-11 Nicoya Therapeutics (Shanghai) Co., Ltd Pyridine derivative and application thereof

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JP2004123694A (ja) * 2002-03-12 2004-04-22 Takeda Chem Ind Ltd 光学活性スルホキシド誘導体の製造法
JP2007269628A (ja) * 2004-05-28 2007-10-18 Takeda Chem Ind Ltd 医薬化合物の結晶
JP2013136629A (ja) * 2001-08-08 2013-07-11 Tobira Therapeutics Inc 二環性化合物、その製造法および用途
WO2016105527A1 (en) * 2014-12-23 2016-06-30 Tobira Therapeutics, Inc. Process of making cenicriviroc and related analogs

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JPS62265270A (ja) 1986-05-13 1987-11-18 Zeria Shinyaku Kogyo Kk 新規イミダゾ−ル誘導体およびそれらを有効成分とする抗潰瘍剤
CA2191980A1 (en) 1994-07-04 1996-01-18 Takashi Sohda Phosphonic acid compounds, their production and use
US6172061B1 (en) 1997-12-19 2001-01-09 Takeda Chemical Industries, Ltd. Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative
AU5301599A (en) 1998-08-20 2000-03-14 Takeda Chemical Industries Ltd. Quaternary ammonium salts and their use
AU6870600A (en) 1999-09-06 2001-04-10 Takeda Chemical Industries Ltd. Process for the preparation of 2,3-dihydroazepine compounds
WO2005089714A1 (ja) 2004-03-24 2005-09-29 Takeda Pharmaceutical Company Limited エマルション安定化製剤
GT200600148A (es) 2005-04-14 2006-11-22 Metodos para el tratamiento y la prevencion de fibrosis
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JP2015520144A (ja) 2012-05-11 2015-07-16 アクロン・モレキュールズ・アクチェンゲゼルシャフトＡｋｒｏｎ Ｍｏｌｅｃｕｌｅｓ Ａｇ 疼痛の治療のための化合物の使用
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JP2013136629A (ja) * 2001-08-08 2013-07-11 Tobira Therapeutics Inc 二環性化合物、その製造法および用途
JP2004123694A (ja) * 2002-03-12 2004-04-22 Takeda Chem Ind Ltd 光学活性スルホキシド誘導体の製造法
JP2007269628A (ja) * 2004-05-28 2007-10-18 Takeda Chem Ind Ltd 医薬化合物の結晶
WO2016105527A1 (en) * 2014-12-23 2016-06-30 Tobira Therapeutics, Inc. Process of making cenicriviroc and related analogs

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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPWO2022177014A1 (https=) * 2021-02-22 2022-08-25
JP7374372B2 (ja) 2021-02-22 2023-11-06 旭化成株式会社 セルロースナノファイバーを含む組成物

Also Published As

Publication number Publication date
EP3506896A4 (en) 2020-08-26
EP3506896A1 (en) 2019-07-10
CA3034606A1 (en) 2018-03-08
WO2018045043A1 (en) 2018-03-08
TW201823235A (zh) 2018-07-01
CN110167550A (zh) 2019-08-23
RU2019109019A3 (https=) 2021-08-23
BR112019003987A2 (pt) 2019-05-28
KR20190057066A (ko) 2019-05-27
JP2022137223A (ja) 2022-09-21
SG11201901438VA (en) 2019-03-28
MX2019002057A (es) 2019-11-18
US20180057481A1 (en) 2018-03-01
US10301287B2 (en) 2019-05-28
RU2019109019A (ru) 2020-10-01
AU2017321594A1 (en) 2019-04-18

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