JP2019526561A5 - - Google Patents

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Publication number
JP2019526561A5
JP2019526561A5 JP2019510788A JP2019510788A JP2019526561A5 JP 2019526561 A5 JP2019526561 A5 JP 2019526561A5 JP 2019510788 A JP2019510788 A JP 2019510788A JP 2019510788 A JP2019510788 A JP 2019510788A JP 2019526561 A5 JP2019526561 A5 JP 2019526561A5
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JP
Japan
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formulation
alkylene
composition
alkyl
carbon atoms
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JP2019510788A
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English (en)
Japanese (ja)
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JP2019526561A (ja
JP6898429B2 (ja
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Priority claimed from PCT/CN2017/098575 external-priority patent/WO2018036498A1/en
Publication of JP2019526561A publication Critical patent/JP2019526561A/ja
Publication of JP2019526561A5 publication Critical patent/JP2019526561A5/ja
Application granted granted Critical
Publication of JP6898429B2 publication Critical patent/JP6898429B2/ja
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JP2019510788A 2016-08-24 2017-08-23 黄斑変性症を治療するためのエンタカポン関連化合物 Active JP6898429B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CNPCT/CN2016/096472 2016-08-24
CN2016096472 2016-08-24
PCT/CN2017/098575 WO2018036498A1 (en) 2016-08-24 2017-08-23 Entacapone-related compounds to treat macular degeneration

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021013670A Division JP7116202B2 (ja) 2016-08-24 2021-01-29 黄斑変性症を治療するための医薬の製造におけるエンタカポン関連化合物の使用

Publications (3)

Publication Number Publication Date
JP2019526561A JP2019526561A (ja) 2019-09-19
JP2019526561A5 true JP2019526561A5 (ja�@�@) 2020-07-16
JP6898429B2 JP6898429B2 (ja) 2021-07-07

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ID=61245496

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2019510788A Active JP6898429B2 (ja) 2016-08-24 2017-08-23 黄斑変性症を治療するためのエンタカポン関連化合物
JP2021013670A Active JP7116202B2 (ja) 2016-08-24 2021-01-29 黄斑変性症を治療するための医薬の製造におけるエンタカポン関連化合物の使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2021013670A Active JP7116202B2 (ja) 2016-08-24 2021-01-29 黄斑変性症を治療するための医薬の製造におけるエンタカポン関連化合物の使用

Country Status (7)

Country Link
US (1) US10980766B2 (ja�@�@)
EP (1) EP3503883B1 (ja�@�@)
JP (2) JP6898429B2 (ja�@�@)
CN (1) CN109689042B (ja�@�@)
AU (1) AU2017317129B2 (ja�@�@)
CA (1) CA3034547C (ja�@�@)
WO (1) WO2018036498A1 (ja�@�@)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10532976B2 (en) * 2015-06-23 2020-01-14 National Institute Of Biological Sciences, Beijing FTO inhibitors
WO2018036498A1 (en) * 2016-08-24 2018-03-01 National Institute Of Biological Sciences, Beijing Entacapone-related compounds to treat macular degeneration
DK4364724T3 (da) 2018-05-10 2025-12-22 Regeneron Pharma Formuleringer med høj koncentration af VEGF-receptorfusionsprotein
EP3886946A1 (en) 2019-06-05 2021-10-06 Regeneron Pharmaceuticals, Inc. Devices and methods for precision dose delivery
CN116963727A (zh) * 2020-11-13 2023-10-27 普莱克斯医药公司 用于治疗眼部病症的药剂
CA3216828A1 (en) * 2021-04-15 2022-10-20 Brown University Nitrophenyl-acrylamides and uses thereof
CA3263420A1 (en) * 2022-07-29 2024-02-01 Rpxds Co., Ltd FTO INHIBITORS
USD1120314S1 (en) 2022-11-30 2026-03-24 Regeneron Pharmaceuticals, Inc. Dose delivery device
WO2025162358A1 (en) * 2024-01-30 2025-08-07 Rpxds Co., Ltd Fto inhibitors of bicyclic structures
WO2025162373A1 (en) * 2024-01-30 2025-08-07 National Institute Of Biological Sciences, Beijing Electrophile-containing catechol-o-methyltransferase (comt) inhibitors for targeting the keap1/nrf2 pathway

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI864875A0 (fi) 1986-11-28 1986-11-28 Orion Yhtymae Oy Nya farmakologiskt aktiva foereningar, dessa innehaollande kompositioner samt foerfarande och mellanprodukter foer anvaendning vid framstaellning av dessa.
US20060034937A1 (en) * 1999-11-23 2006-02-16 Mahesh Patel Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
TW200817315A (en) 2006-06-16 2008-04-16 Sanol Arznei Schwarz Gmbh Entacapone-derivatives
EP1946756A1 (en) * 2007-01-17 2008-07-23 Revotar Biopharmaceuticals AG Use of entacapone in cosmetic, dermatological and pharmaceutical compositions
EP1978014A1 (en) 2007-04-02 2008-10-08 Esteve Quimica, S.A. Process for the preparation of entacapone and intermediates thereof
US9827210B2 (en) * 2007-06-29 2017-11-28 Phovitreal Pty Ltd Treatment or prophylaxis of a neurological or neuropsychiatric disorders via ocular administration
EP2273988B1 (en) * 2008-04-18 2015-09-09 Arizona Board Of Regents, A Body Corp. Of The State Of Arizona, Acting For And On Behalf Of The University Of Arizona L-dopa for treating age-related macular degeneration
US20110190356A1 (en) * 2008-08-19 2011-08-04 Knopp Neurosciences Inc. Compositions and Methods of Using (R)- Pramipexole
KR20130050939A (ko) * 2010-04-12 2013-05-16 가부시키가이샤 아루떼꾸 우에노 망막 질환의 치료 방법 및 이를 위한 안과용 조성물
WO2012142039A1 (en) * 2011-04-15 2012-10-18 University Of North Dakota Combination of liver x receptor modulator and estrogen receptor modulator for the treatment of age-related diseases
JP2016504270A (ja) * 2012-10-17 2016-02-12 ザ ユニバーシティ オブ ブリストル 眼血管形成(ocularneovasculan)を治療するのに有用な化合物
CN103845317B (zh) 2012-11-28 2018-05-08 北京生命科学研究所 恩他卡朋在预防或治疗肥胖等代谢综合征中的应用
US20160317474A1 (en) 2013-12-18 2016-11-03 Emory University Managing Visual Dysfunction or Loss of Vision for Diabetic Subjects
JP6858712B2 (ja) * 2015-01-30 2021-04-14 リーバー インスティテュート フォー ブレイン ディベロップメントLieber Institute For Brain Development Comt阻害方法及び組成物
WO2016123577A1 (en) * 2015-01-30 2016-08-04 Lieber Institute For Brain Development Comt inhibiting methods and compositions
EP3303283B1 (en) 2015-06-23 2021-04-21 National Institute Of Biological Sciences, Beijing Fto inhibitors
WO2018036498A1 (en) * 2016-08-24 2018-03-01 National Institute Of Biological Sciences, Beijing Entacapone-related compounds to treat macular degeneration

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