JP2018528985A - カンナビノイドを含む経口医薬組成物、その調製及び使用のための方法 - Google Patents

カンナビノイドを含む経口医薬組成物、その調製及び使用のための方法 Download PDF

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Publication number
JP2018528985A
JP2018528985A JP2018533979A JP2018533979A JP2018528985A JP 2018528985 A JP2018528985 A JP 2018528985A JP 2018533979 A JP2018533979 A JP 2018533979A JP 2018533979 A JP2018533979 A JP 2018533979A JP 2018528985 A JP2018528985 A JP 2018528985A
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oil
composition according
acid
combinations
cannabinoid
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JP2018533979A
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Japanese (ja)
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JP2018528985A5 (enExample
Inventor
ドナドゥッチ、ルイス
マリア ドナドゥッチ、カルメン
マリア ドナドゥッチ、カルメン
メネゼス、クリスチャン グレゴリー ブルゴス デ
メネゼス、クリスチャン グレゴリー ブルゴス デ
ブラム ジュニオール、リベラート
ブラム ジュニオール、リベラート
ホセ トンド フィルホ、ヴォルネイ
ホセ トンド フィルホ、ヴォルネイ
モウラ ローザ、パトリシア
モウラ ローザ、パトリシア
アレクサンドル クリッパ、ホセ
アレクサンドル クリッパ、ホセ
エデュアルド セシリオ ハラック、ハイメ
エデュアルド セシリオ ハラック、ハイメ
ワルド ズアルディ、アントニオ
ワルド ズアルディ、アントニオ
シルヴェイラ ギマラエス、フランシスコ
シルヴェイラ ギマラエス、フランシスコ
Original Assignee
プラティ、ドナドゥッチ エー シア リミターダ
プラティ、ドナドゥッチ エー シア リミターダ
ウニヴェルシダーデ デ サンパウロ
ウニヴェルシダーデ デ サンパウロ
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Application filed by プラティ、ドナドゥッチ エー シア リミターダ, プラティ、ドナドゥッチ エー シア リミターダ, ウニヴェルシダーデ デ サンパウロ, ウニヴェルシダーデ デ サンパウロ filed Critical プラティ、ドナドゥッチ エー シア リミターダ
Publication of JP2018528985A publication Critical patent/JP2018528985A/ja
Publication of JP2018528985A5 publication Critical patent/JP2018528985A5/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44—Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/05—Phenols
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/658—Medicinal preparations containing organic active ingredients o-phenolic cannabinoids, e.g. cannabidiol, cannabigerolic acid, cannabichromene or tetrahydrocannabinol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Pain & Pain Management (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
JP2018533979A 2015-09-18 2016-09-16 カンナビノイドを含む経口医薬組成物、その調製及び使用のための方法 Pending JP2018528985A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
BR102015024165A BR102015024165A2 (pt) 2015-09-18 2015-09-18 composição farmacêutica oral compreendendo canabinóide, processo para sua preparação e seu uso
BRBR102015024165-8 2015-09-18
PCT/BR2016/050231 WO2017045053A1 (pt) 2015-09-18 2016-09-16 Composição farmacêutica oral compreendendo canabinóide, processo para sua preparação e seu uso

Publications (2)

Publication Number Publication Date
JP2018528985A true JP2018528985A (ja) 2018-10-04
JP2018528985A5 JP2018528985A5 (enExample) 2021-02-04

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ID=58288018

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JP2018533979A Pending JP2018528985A (ja) 2015-09-18 2016-09-16 カンナビノイドを含む経口医薬組成物、その調製及び使用のための方法

Country Status (8)

Country Link
US (1) US20180264121A1 (enExample)
EP (1) EP3351242A4 (enExample)
JP (1) JP2018528985A (enExample)
CN (1) CN108366988A (enExample)
AU (1) AU2016322148A1 (enExample)
BR (2) BR102015024165A2 (enExample)
CA (1) CA2998739A1 (enExample)
WO (1) WO2017045053A1 (enExample)

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JP2022552056A (ja) * 2019-09-09 2022-12-15 カーディオル セラピューティクス インコーポレイテッド 安定な薬用カンナビジオール組成物
JP2023039414A (ja) * 2021-09-08 2023-03-20 株式会社東洋新薬 経口組成物

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EP3658137A4 (en) * 2017-07-27 2020-06-03 Shaaban, Basil Adil CANNABINOID COMPOSITION WITH OPTIMIZED FATTY ACID PROFILE
US20190083622A1 (en) * 2017-10-16 2019-03-21 Joshua Raderman Cannabinoid formulations and methods including the antioxidant c60
AU2019217673A1 (en) 2018-02-07 2020-09-24 Scf Pharma Inc. Polyunsaturated fatty acid monoglycerides, compositions, methods and uses thereof
BR102018002843A2 (pt) * 2018-02-09 2019-08-27 Prati Donaduzzi & Cia Ltda composição farmacêutica e uso da mesma
ES2992095T3 (es) 2018-05-03 2024-12-09 Scf Pharma Inc Monoglicéridos de ácidos grasos poliinsaturados, composiciones y uso de los mismos para modular la composición de la microbiota de un sujeto
US20220304963A1 (en) * 2018-07-27 2022-09-29 Basil Shaaban Composition having an optimized fatty acid excipient profile
IL261132A (en) * 2018-08-13 2018-11-04 Yissum Res Dev Co Of Hebrew Univ Jerusalem Ltd Formulated cannabis oil powder by nanoemulsifycation, methods of producing and uses thereof
WO2020044118A1 (en) * 2018-08-27 2020-03-05 Emerald Health Therapeutics Canada Inc. Improved cannabinoid bioavailability
CN108968071A (zh) * 2018-09-26 2018-12-11 江西中医药大学 代代花和火麻仁组合物在制备改善记忆力减退或治疗抑郁症药物或保健功能饮料中的应用
US12484606B2 (en) 2018-12-14 2025-12-02 Natural Extraction Systems, LLC Compositions and methods related to anionic cannabinoid molecules
US11026888B1 (en) 2019-01-04 2021-06-08 Nutrition Therapeutics, Inc. Functional beverage compositions and methods of using and making same
CA3040547C (en) * 2019-04-17 2021-12-07 Medcan Pharma A/S Cannabinoid lozenge formulation
US12226390B2 (en) 2019-07-21 2025-02-18 Scf Pharma Inc. Cannabinoids compositions with polyunsaturated fatty acid monoglycerides, methods and uses thereof
AU2020318671B2 (en) * 2019-07-21 2021-12-23 Scf Pharma Inc. Cannabinoids compositions with polyunsaturated fatty acid monoglycerides, methods and uses thereof
MX2022001634A (es) * 2019-08-08 2022-05-11 Neptune Wellness Solutions Inc Formulaciones orales de extractos de cannabis y metodos para elaborar las mismas.
US12419855B2 (en) 2019-08-28 2025-09-23 Natural Extraction Systems, LLC Compositions comprising cannabinoid ions that are dissolved in glycerol
CN113694049B (zh) * 2020-05-21 2022-11-22 汉义生物科技（北京）有限公司 大麻素类化合物及其在治疗帕金森症中的应用
CN111603443B (zh) * 2020-06-12 2022-06-28 苏州旺山旺水生物医药有限公司 一种稳定的cbd组合物及其应用
WO2022026960A1 (en) 2020-07-31 2022-02-03 Natural Extraction Systems, LLC Compositions and methods related to excipients and cannabinoid formulations
CA3217137A1 (en) 2021-04-29 2022-11-03 Christopher Adair Cannabidiol-dominant formulations, methods of manufacturing, and uses thereof
AU2023361756A1 (en) * 2022-10-12 2025-05-22 Leiutis Pharmaceuticals Llp Novel liquid oral formulations of cannabidiol
WO2024168426A1 (en) 2023-02-13 2024-08-22 Apogee Pharmaceuticals, Inc. Small molecules as monoacylglycerol lipase (magl) inhibitors, compositions and use thereof
EP4522133A4 (en) * 2023-07-24 2025-03-19 Poviva Corp. COMPOSITIONS AND METHODS FOR THE TREATMENT OF EPILEPSY

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JP2022552056A (ja) * 2019-09-09 2022-12-15 カーディオル セラピューティクス インコーポレイテッド 安定な薬用カンナビジオール組成物
JP7487292B2 (ja) 2019-09-09 2024-05-20 カーディオル セラピューティクス インコーポレイテッド 安定な薬用カンナビジオール組成物
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JP2023039414A (ja) * 2021-09-08 2023-03-20 株式会社東洋新薬 経口組成物

Also Published As

Publication number Publication date
CN108366988A (zh) 2018-08-03
EP3351242A4 (en) 2019-05-15
BR112018005423B1 (pt) 2020-06-23
US20180264121A1 (en) 2018-09-20
WO2017045053A1 (pt) 2017-03-23
EP3351242A1 (en) 2018-07-25
AU2016322148A1 (en) 2018-04-12
CA2998739A1 (en) 2017-03-23
BR102015024165A2 (pt) 2017-03-28

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