JP2018521956A5 - - Google Patents
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- JP2018521956A5 JP2018521956A5 JP2017548194A JP2017548194A JP2018521956A5 JP 2018521956 A5 JP2018521956 A5 JP 2018521956A5 JP 2017548194 A JP2017548194 A JP 2017548194A JP 2017548194 A JP2017548194 A JP 2017548194A JP 2018521956 A5 JP2018521956 A5 JP 2018521956A5
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562166240P | 2015-05-26 | 2015-05-26 | |
| US62/166,240 | 2015-05-26 | ||
| PCT/US2016/033923 WO2016191424A2 (en) | 2015-05-26 | 2016-05-24 | Novel heteroaromatic silicon-fluoride-acceptors useful for 18f labeling of molecules and biomolecules, and methods of preparing same |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021017722A Division JP2021073293A (ja) | 2015-05-26 | 2021-02-05 | 分子および生体分子の１８ｆ標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018521956A JP2018521956A (ja) | 2018-08-09 |
| JP2018521956A5 true JP2018521956A5 (https=) | 2019-06-27 |
| JP7266365B2 JP7266365B2 (ja) | 2023-04-28 |
Family
ID=57394170
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017548194A Active JP7266365B2 (ja) | 2015-05-26 | 2016-05-24 | 分子および生体分子の１８ｆ標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 |
| JP2021017722A Withdrawn JP2021073293A (ja) | 2015-05-26 | 2021-02-05 | 分子および生体分子の１８ｆ標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021017722A Withdrawn JP2021073293A (ja) | 2015-05-26 | 2021-02-05 | 分子および生体分子の１８ｆ標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 |
Country Status (6)
| Country | Link |
|---|---|
| US (4) | US10800797B2 (https=) |
| EP (1) | EP3303349B1 (https=) |
| JP (2) | JP7266365B2 (https=) |
| CN (1) | CN107667109B (https=) |
| CA (1) | CA2982269C (https=) |
| WO (1) | WO2016191424A2 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN107667109B (zh) | 2015-05-26 | 2021-08-03 | 加利福尼亚大学董事会 | 可用于分子和生物分子的18f标记的新的杂芳族硅-氟化物-受体及其制备方法 |
| EA202090370A1 (ru) * | 2017-07-28 | 2020-05-25 | Технише Универзитет Мюнхен | Двухрежимная радиоактивная метка и радиотерапевтическое средство |
| US11464784B2 (en) | 2017-09-15 | 2022-10-11 | The Regents Of The University Of California | Inhibition of aminocylase 3 (AA3) in the treatment of cancer |
| CN113677375B (zh) * | 2019-01-30 | 2024-07-23 | 慕尼黑工业大学 | 氟化硅受体取代的放射性药物及其前体 |
| WO2020220020A1 (en) * | 2019-04-26 | 2020-10-29 | The Regents Of The University Of California | Silicon-fluoride heteroaromatic systems for applications in positron emission tomography (pet) molecular imaging |
| CN114206937B (zh) * | 2019-05-24 | 2025-06-03 | 杜克大学 | 18f放射性标记的生物分子 |
| WO2021243337A1 (en) * | 2020-05-29 | 2021-12-02 | Fuzionaire. Inc. | Methods for rapid formation of chemicals including positron emission tomography biomarkers |
| CA3249624A1 (en) * | 2022-04-20 | 2023-10-26 | Fuzionaire Theranostics, Inc. | HETEROAROMATIC SYSTEMS OF THERANOSTIC SILICON FLUORIDE AND ASSOCIATED METHODS |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6972336B2 (en) * | 2002-07-18 | 2005-12-06 | Novartis Ag | N-alkylation of indole derivatives |
| US20090035215A1 (en) | 2006-10-02 | 2009-02-05 | Ananth Srinivasan | Radiofluorination |
| US20120046242A1 (en) * | 2008-12-24 | 2012-02-23 | Massachusetts Institute Of Technology | Molecular activators of the wnt/beta-catenin pathway |
| CA3159948A1 (en) * | 2010-12-22 | 2012-07-19 | General Electric Company | Radiolabled her2 binding peptides |
| CN107667109B (zh) * | 2015-05-26 | 2021-08-03 | 加利福尼亚大学董事会 | 可用于分子和生物分子的18f标记的新的杂芳族硅-氟化物-受体及其制备方法 |
-
2016
- 2016-05-24 CN CN201680030562.8A patent/CN107667109B/zh active Active
- 2016-05-24 CA CA2982269A patent/CA2982269C/en active Active
- 2016-05-24 EP EP16800638.5A patent/EP3303349B1/en active Active
- 2016-05-24 WO PCT/US2016/033923 patent/WO2016191424A2/en not_active Ceased
- 2016-05-24 US US15/575,979 patent/US10800797B2/en active Active
- 2016-05-24 JP JP2017548194A patent/JP7266365B2/ja active Active
-
2020
- 2020-08-19 US US16/997,240 patent/US11447508B2/en active Active
-
2021
- 2021-02-05 JP JP2021017722A patent/JP2021073293A/ja not_active Withdrawn
-
2022
- 2022-09-19 US US17/933,234 patent/US12371445B2/en active Active
-
2025
- 2025-06-25 US US19/248,601 patent/US20250333425A1/en active Pending
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| JP2018521956A5 (https=) | ||
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