JP2018521956A5 - - Google Patents
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- JP2018521956A5 JP2018521956A5 JP2017548194A JP2017548194A JP2018521956A5 JP 2018521956 A5 JP2018521956 A5 JP 2018521956A5 JP 2017548194 A JP2017548194 A JP 2017548194A JP 2017548194 A JP2017548194 A JP 2017548194A JP 2018521956 A5 JP2018521956 A5 JP 2018521956A5
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562166240P | 2015-05-26 | 2015-05-26 | |
| US62/166,240 | 2015-05-26 | ||
| PCT/US2016/033923 WO2016191424A2 (en) | 2015-05-26 | 2016-05-24 | Novel heteroaromatic silicon-fluoride-acceptors useful for 18f labeling of molecules and biomolecules, and methods of preparing same |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021017722A Division JP2021073293A (ja) | 2015-05-26 | 2021-02-05 | 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018521956A JP2018521956A (ja) | 2018-08-09 |
| JP2018521956A5 true JP2018521956A5 (https=) | 2019-06-27 |
| JP7266365B2 JP7266365B2 (ja) | 2023-04-28 |
Family
ID=57394170
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017548194A Active JP7266365B2 (ja) | 2015-05-26 | 2016-05-24 | 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 |
| JP2021017722A Withdrawn JP2021073293A (ja) | 2015-05-26 | 2021-02-05 | 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021017722A Withdrawn JP2021073293A (ja) | 2015-05-26 | 2021-02-05 | 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 |
Country Status (6)
| Country | Link |
|---|---|
| US (4) | US10800797B2 (https=) |
| EP (1) | EP3303349B1 (https=) |
| JP (2) | JP7266365B2 (https=) |
| CN (1) | CN107667109B (https=) |
| CA (1) | CA2982269C (https=) |
| WO (1) | WO2016191424A2 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10800797B2 (en) | 2015-05-26 | 2020-10-13 | California Institute Of Technology | Heteroaromatic silicon-fluoride-acceptors useful for 18F labeling of molecules and biomolecules, and methods of preparing same |
| HUE070098T2 (hu) * | 2017-07-28 | 2025-05-28 | Univ Muenchen Tech | Kettõs módusú radioaktív jelzõ és terapeutikumok |
| DE112018005145T5 (de) | 2017-09-15 | 2020-07-23 | The Regents Of The University Of California | Hemmung von aminoacylase 3 (aa3) bei der behandlung von krebs |
| BR112021012110A2 (pt) * | 2019-01-30 | 2021-09-08 | Technische Universität München | Radiofarmacêuticos substituídos por aceptor de fluoreto de silício |
| WO2020220020A1 (en) * | 2019-04-26 | 2020-10-29 | The Regents Of The University Of California | Silicon-fluoride heteroaromatic systems for applications in positron emission tomography (pet) molecular imaging |
| KR102899941B1 (ko) * | 2019-05-24 | 2025-12-16 | 듀크 유니버시티 | 18f-방사선 표지된 생체 분자 |
| WO2021243337A1 (en) * | 2020-05-29 | 2021-12-02 | Fuzionaire. Inc. | Methods for rapid formation of chemicals including positron emission tomography biomarkers |
| KR20250006177A (ko) * | 2022-04-20 | 2025-01-10 | 퓨지오네어 테라노스틱스, 인크. | 테라노스틱 플루오르화규소 헤테로방향족 시스템 및 이의 방법 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6972336B2 (en) * | 2002-07-18 | 2005-12-06 | Novartis Ag | N-alkylation of indole derivatives |
| US20090035215A1 (en) * | 2006-10-02 | 2009-02-05 | Ananth Srinivasan | Radiofluorination |
| US20120046242A1 (en) * | 2008-12-24 | 2012-02-23 | Massachusetts Institute Of Technology | Molecular activators of the wnt/beta-catenin pathway |
| NZ612161A (en) * | 2010-12-22 | 2015-04-24 | Gen Electric | Radiolabled her2 binding peptides |
| US10800797B2 (en) | 2015-05-26 | 2020-10-13 | California Institute Of Technology | Heteroaromatic silicon-fluoride-acceptors useful for 18F labeling of molecules and biomolecules, and methods of preparing same |
-
2016
- 2016-05-24 US US15/575,979 patent/US10800797B2/en active Active
- 2016-05-24 JP JP2017548194A patent/JP7266365B2/ja active Active
- 2016-05-24 CN CN201680030562.8A patent/CN107667109B/zh active Active
- 2016-05-24 WO PCT/US2016/033923 patent/WO2016191424A2/en not_active Ceased
- 2016-05-24 CA CA2982269A patent/CA2982269C/en active Active
- 2016-05-24 EP EP16800638.5A patent/EP3303349B1/en active Active
-
2020
- 2020-08-19 US US16/997,240 patent/US11447508B2/en active Active
-
2021
- 2021-02-05 JP JP2021017722A patent/JP2021073293A/ja not_active Withdrawn
-
2022
- 2022-09-19 US US17/933,234 patent/US12371445B2/en active Active
-
2025
- 2025-06-25 US US19/248,601 patent/US20250333425A1/en active Pending
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