JP2018521956A5 - - Google Patents

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JP2018521956A5
JP2018521956A5 JP2017548194A JP2017548194A JP2018521956A5 JP 2018521956 A5 JP2018521956 A5 JP 2018521956A5 JP 2017548194 A JP2017548194 A JP 2017548194A JP 2017548194 A JP2017548194 A JP 2017548194A JP 2018521956 A5 JP2018521956 A5 JP 2018521956A5
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JP7266365B2 (ja
JP2018521956A (ja
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Priority claimed from PCT/US2016/033923 external-priority patent/WO2016191424A2/en
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JP2017548194A 2015-05-26 2016-05-24 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法 Active JP7266365B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562166240P 2015-05-26 2015-05-26
US62/166,240 2015-05-26
PCT/US2016/033923 WO2016191424A2 (en) 2015-05-26 2016-05-24 Novel heteroaromatic silicon-fluoride-acceptors useful for 18f labeling of molecules and biomolecules, and methods of preparing same

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JP2021017722A Division JP2021073293A (ja) 2015-05-26 2021-02-05 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法

Publications (3)

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JP2018521956A JP2018521956A (ja) 2018-08-09
JP2018521956A5 true JP2018521956A5 (https=) 2019-06-27
JP7266365B2 JP7266365B2 (ja) 2023-04-28

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JP2017548194A Active JP7266365B2 (ja) 2015-05-26 2016-05-24 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法
JP2021017722A Withdrawn JP2021073293A (ja) 2015-05-26 2021-02-05 分子および生体分子の18f標識化に有用な新規な複素芳香環フッ化ケイ素アクセプタおよびその調製方法

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US (4) US10800797B2 (https=)
EP (1) EP3303349B1 (https=)
JP (2) JP7266365B2 (https=)
CN (1) CN107667109B (https=)
CA (1) CA2982269C (https=)
WO (1) WO2016191424A2 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10800797B2 (en) 2015-05-26 2020-10-13 California Institute Of Technology Heteroaromatic silicon-fluoride-acceptors useful for 18F labeling of molecules and biomolecules, and methods of preparing same
HUE070098T2 (hu) * 2017-07-28 2025-05-28 Univ Muenchen Tech Kettõs módusú radioaktív jelzõ és terapeutikumok
DE112018005145T5 (de) 2017-09-15 2020-07-23 The Regents Of The University Of California Hemmung von aminoacylase 3 (aa3) bei der behandlung von krebs
BR112021012110A2 (pt) * 2019-01-30 2021-09-08 Technische Universität München Radiofarmacêuticos substituídos por aceptor de fluoreto de silício
WO2020220020A1 (en) * 2019-04-26 2020-10-29 The Regents Of The University Of California Silicon-fluoride heteroaromatic systems for applications in positron emission tomography (pet) molecular imaging
KR102899941B1 (ko) * 2019-05-24 2025-12-16 듀크 유니버시티 18f-방사선 표지된 생체 분자
WO2021243337A1 (en) * 2020-05-29 2021-12-02 Fuzionaire. Inc. Methods for rapid formation of chemicals including positron emission tomography biomarkers
KR20250006177A (ko) * 2022-04-20 2025-01-10 퓨지오네어 테라노스틱스, 인크. 테라노스틱 플루오르화규소 헤테로방향족 시스템 및 이의 방법

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* Cited by examiner, † Cited by third party
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US6972336B2 (en) * 2002-07-18 2005-12-06 Novartis Ag N-alkylation of indole derivatives
US20090035215A1 (en) * 2006-10-02 2009-02-05 Ananth Srinivasan Radiofluorination
US20120046242A1 (en) * 2008-12-24 2012-02-23 Massachusetts Institute Of Technology Molecular activators of the wnt/beta-catenin pathway
NZ612161A (en) * 2010-12-22 2015-04-24 Gen Electric Radiolabled her2 binding peptides
US10800797B2 (en) 2015-05-26 2020-10-13 California Institute Of Technology Heteroaromatic silicon-fluoride-acceptors useful for 18F labeling of molecules and biomolecules, and methods of preparing same

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