JP2017535546A5 - - Google Patents
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- JP2017535546A5 JP2017535546A5 JP2017525839A JP2017525839A JP2017535546A5 JP 2017535546 A5 JP2017535546 A5 JP 2017535546A5 JP 2017525839 A JP2017525839 A JP 2017525839A JP 2017525839 A JP2017525839 A JP 2017525839A JP 2017535546 A5 JP2017535546 A5 JP 2017535546A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutically acceptable
- acceptable salt
- prodrug
- formula
- trifluoromethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 125000001246 bromo group Chemical group Br* 0.000 claims description 46
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|---|---|---|---|---|
| KR20090090406A (ko) * | 2000-12-18 | 2009-08-25 | 가부시키가이샤 이야쿠 분지 셋케이 겐쿠쇼 | 염증성 사이토카인 생산 유리 억제제 |
| WO2003103658A1 (ja) * | 2002-06-05 | 2003-12-18 | 株式会社医薬分子設計研究所 | 免疫関連プロテインキナーゼ阻害剤 |
| JP4743382B2 (ja) * | 2002-06-06 | 2011-08-10 | 株式会社医薬分子設計研究所 | Ｏ−置換ヒドロキシアリール誘導体 |
| AU2008216612B2 (en) * | 2007-02-17 | 2014-12-04 | President And Fellows Of Harvard College | Compositions and method for tissue preservation |
| CN101842093B (zh) * | 2007-10-23 | 2012-08-22 | 株式会社医药分子设计研究所 | Pai-1产生抑制剂 |
| US20120238623A1 (en) * | 2011-03-14 | 2012-09-20 | Chandraratna Roshantha A | Inflammation and Autoimmune Disorder Treatment using RARa Selective Agonists |
| JP6238969B2 (ja) * | 2012-05-08 | 2017-11-29 | エアロミクス・インコーポレイテッドＡｅｒｏｍｉｃｓ，Ｉｎｃ． | 新規方法 |
-
2015
- 2015-11-13 JP JP2017525839A patent/JP2017535546A/ja not_active Withdrawn
- 2015-11-13 US US15/526,706 patent/US20180042873A1/en not_active Abandoned
- 2015-11-13 SG SG11201703801SA patent/SG11201703801SA/en unknown
- 2015-11-13 AU AU2015346076A patent/AU2015346076A1/en not_active Abandoned
- 2015-11-13 EP EP15859827.6A patent/EP3218354A4/en not_active Withdrawn
- 2015-11-13 WO PCT/US2015/060731 patent/WO2016077787A1/en not_active Ceased
- 2015-11-13 CA CA2966950A patent/CA2966950A1/en not_active Abandoned
- 2015-11-13 CN CN201580073130.0A patent/CN107207417A/zh active Pending
-
2016
- 2016-05-18 TW TW105115290A patent/TW201716059A/zh unknown
-
2017
- 2017-05-03 IL IL252086A patent/IL252086A0/en unknown
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