JP2017531678A5 - - Google Patents
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- JP2017531678A5 JP2017531678A5 JP2017522086A JP2017522086A JP2017531678A5 JP 2017531678 A5 JP2017531678 A5 JP 2017531678A5 JP 2017522086 A JP2017522086 A JP 2017522086A JP 2017522086 A JP2017522086 A JP 2017522086A JP 2017531678 A5 JP2017531678 A5 JP 2017531678A5
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14190073.8 | 2014-10-23 | ||
| EP14190073 | 2014-10-23 | ||
| PCT/EP2015/074431 WO2016062790A1 (en) | 2014-10-23 | 2015-10-22 | New pyrazolopyrimidine derivatives as nik inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017531678A JP2017531678A (ja) | 2017-10-26 |
| JP2017531678A5 true JP2017531678A5 (enrdf_load_stackoverflow) | 2019-11-21 |
| JP6616412B2 JP6616412B2 (ja) | 2019-12-04 |
Family
ID=51846471
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017522086A Expired - Fee Related JP6616412B2 (ja) | 2014-10-23 | 2015-10-22 | Ｎｉｋ阻害剤としての新規のピラゾロピリミジン誘導体 |
Country Status (13)
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI663166B (zh) | 2013-04-24 | 2019-06-21 | 健生藥品公司 | 新化合物 |
| TWI704146B (zh) | 2013-09-26 | 2020-09-11 | 比利時商健生藥品公司 | 用作ＮＩＫ抑制劑之新的1-(４-嘧啶基)-１Ｈ-吡唑並[３,２-ｃ]吡啶衍生物 |
| TWI627173B (zh) | 2013-09-26 | 2018-06-21 | 比利時商健生藥品公司 | 作為ＮＩＫ抑制劑的新穎３－（１Ｈ－吡唑－４－基）－１Ｈ－吡咯并［２，３－ｃ］吡啶衍生物 |
| WO2016062790A1 (en) | 2014-10-23 | 2016-04-28 | Janssen Pharmaceutica Nv | New pyrazolopyrimidine derivatives as nik inhibitors |
| AU2015334917B2 (en) | 2014-10-23 | 2019-08-29 | Janssen Pharmaceutica Nv | New compounds as NIK inhibitors |
| WO2016062791A1 (en) | 2014-10-23 | 2016-04-28 | Janssen Pharmaceutica Nv | New pyrazole derivatives as nik inhibitors |
| CA2960567C (en) | 2014-10-23 | 2023-03-07 | Janssen Pharmaceutica Nv | Thienopyrimidine derivatives as nik inhibitors |
| ES2988933T3 (es) | 2018-06-07 | 2024-11-22 | Disarm Therapeutics Inc | Inhibidores de SARM1 |
| EP3810609B1 (en) * | 2018-06-18 | 2024-06-12 | Janssen Pharmaceutica NV | Pyrazole derivatives as malt1 inhibitors |
| JP7212781B2 (ja) | 2018-12-19 | 2023-01-25 | ディスアーム セラピューティクス， インコーポレイテッド | 神経保護剤と組み合わせたｓａｒｍ１の阻害剤 |
| KR20210146320A (ko) * | 2019-03-29 | 2021-12-03 | 교와 가부시키가이샤 | 신규 아자인돌 유도체 |
| HUE068694T2 (hu) | 2019-05-31 | 2025-01-28 | Janssen Pharmaceutica Nv | NF-KB indukáló kináz kismolekulás inhibitorai |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1990007926A1 (en) * | 1989-01-20 | 1990-07-26 | Pfizer Inc. | 3-(1,2,5,6-tetrahydropyridyl)-pyrrolopyridines |
| MXPA06012449A (es) | 2004-04-26 | 2007-01-17 | Pfizer | Inhibidores de la enzima integrasa de vih. |
| AR056786A1 (es) | 2005-11-10 | 2007-10-24 | Smithkline Beecham Corp | Compuesto de 1h- imidazo ( 4,5-c) piridin-2-ilo, composicion farmaceutica que lo comprende, procedimiento para preparar dicha composicion, su uso para preparar unmedicamento, uso de una combinacion que omprende al compuesto y al menos un agente antineoplasico para preparar un medicamento y dicha com |
| DE102008005493A1 (de) | 2008-01-22 | 2009-07-23 | Merck Patent Gmbh | 4-(Pyrrolo[2,3-c] pyridine-3-yl)-pyrimidin-2-yl-amin-derivate |
| JP2011525915A (ja) | 2008-06-26 | 2011-09-29 | アムジエン・インコーポレーテツド | キナーゼ阻害薬としてのアルキニルアルコール類 |
| AU2009266806A1 (en) | 2008-07-03 | 2010-01-07 | Exelixis Inc. | CDK modulators |
| US20110183975A1 (en) | 2008-10-07 | 2011-07-28 | Yasuhiro Goto | Novel 6-azaindole aminopyrimidine derivatives having nik inhibitory activity |
| CN101723936B (zh) | 2008-10-27 | 2014-01-15 | 上海睿星基因技术有限公司 | 激酶抑制剂及其在药学中的用途 |
| WO2011050245A1 (en) | 2009-10-23 | 2011-04-28 | Yangbo Feng | Bicyclic heteroaryls as kinase inhibitors |
| KR20130133051A (ko) | 2011-03-16 | 2013-12-05 | 에프. 호프만-라 로슈 아게 | 6,5-헤테로사이클릭 프로파길릭 알콜 화합물 및 이의 용도 |
| TWI663166B (zh) * | 2013-04-24 | 2019-06-21 | 健生藥品公司 | 新化合物 |
| TWI704146B (zh) | 2013-09-26 | 2020-09-11 | 比利時商健生藥品公司 | 用作ＮＩＫ抑制劑之新的1-(４-嘧啶基)-１Ｈ-吡唑並[３,２-ｃ]吡啶衍生物 |
| TWI627173B (zh) | 2013-09-26 | 2018-06-21 | 比利時商健生藥品公司 | 作為ＮＩＫ抑制劑的新穎３－（１Ｈ－吡唑－４－基）－１Ｈ－吡咯并［２，３－ｃ］吡啶衍生物 |
| WO2016062791A1 (en) | 2014-10-23 | 2016-04-28 | Janssen Pharmaceutica Nv | New pyrazole derivatives as nik inhibitors |
| AU2015334917B2 (en) | 2014-10-23 | 2019-08-29 | Janssen Pharmaceutica Nv | New compounds as NIK inhibitors |
| CA2960567C (en) * | 2014-10-23 | 2023-03-07 | Janssen Pharmaceutica Nv | Thienopyrimidine derivatives as nik inhibitors |
| WO2016062790A1 (en) | 2014-10-23 | 2016-04-28 | Janssen Pharmaceutica Nv | New pyrazolopyrimidine derivatives as nik inhibitors |
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2015
- 2015-10-22 WO PCT/EP2015/074431 patent/WO2016062790A1/en not_active Ceased
- 2015-10-22 CN CN201580057545.9A patent/CN107074882B/zh not_active Expired - Fee Related
- 2015-10-22 BR BR112017007704-3A patent/BR112017007704B1/pt not_active IP Right Cessation
- 2015-10-22 EA EA201790907A patent/EA033237B1/ru not_active IP Right Cessation
- 2015-10-22 ES ES15784050T patent/ES2715104T3/es active Active
- 2015-10-22 CA CA2960574A patent/CA2960574C/en active Active
- 2015-10-22 JP JP2017522086A patent/JP6616412B2/ja not_active Expired - Fee Related
- 2015-10-22 MX MX2017005284A patent/MX371152B/es active IP Right Grant
- 2015-10-22 KR KR1020177010805A patent/KR102523405B1/ko active Active
- 2015-10-22 US US15/520,346 patent/US10221180B2/en active Active
- 2015-10-22 AU AU2015334915A patent/AU2015334915B2/en not_active Ceased
- 2015-10-22 EP EP15784050.5A patent/EP3209663B1/en active Active
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2017
- 2017-04-19 IL IL251778A patent/IL251778B/en active IP Right Grant
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2019
- 2019-02-01 US US16/265,679 patent/US10822342B2/en active Active