JP2017530193A5 - - Google Patents
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- Publication number
- JP2017530193A5 JP2017530193A5 JP2017535616A JP2017535616A JP2017530193A5 JP 2017530193 A5 JP2017530193 A5 JP 2017530193A5 JP 2017535616 A JP2017535616 A JP 2017535616A JP 2017535616 A JP2017535616 A JP 2017535616A JP 2017530193 A5 JP2017530193 A5 JP 2017530193A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- heteroaryl
- heterocycloalkyl
- aryl
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- RXYPXQSKLGGKOL-UHFFFAOYSA-N CN1CCN(C)CC1 Chemical compound CN1CCN(C)CC1 RXYPXQSKLGGKOL-UHFFFAOYSA-N 0.000 description 2
- TZYFCEGYHDNOFE-UHFFFAOYSA-N CC(CC1N(C)CCCC1)[n]1nncc1 Chemical compound CC(CC1N(C)CCCC1)[n]1nncc1 TZYFCEGYHDNOFE-UHFFFAOYSA-N 0.000 description 1
- PAMIQIKDUOTOBW-UHFFFAOYSA-N CN1CCCCC1 Chemical compound CN1CCCCC1 PAMIQIKDUOTOBW-UHFFFAOYSA-N 0.000 description 1
- JWAWEQBUZOGIBZ-UHFFFAOYSA-N C[n]1nncc1 Chemical compound C[n]1nncc1 JWAWEQBUZOGIBZ-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462053389P | 2014-09-22 | 2014-09-22 | |
| US62/053,389 | 2014-09-22 | ||
| PCT/US2015/051143 WO2016048861A2 (en) | 2014-09-22 | 2015-09-21 | Heterocyclic compounds and use thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017530193A JP2017530193A (ja) | 2017-10-12 |
| JP2017530193A5 true JP2017530193A5 (https=) | 2018-11-01 |
| JP6615207B2 JP6615207B2 (ja) | 2019-12-04 |
Family
ID=55525127
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017535616A Active JP6615207B2 (ja) | 2014-09-22 | 2015-09-21 | 複素環式化合物及びその使用 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US9862703B2 (https=) |
| EP (1) | EP3197885B1 (https=) |
| JP (1) | JP6615207B2 (https=) |
| KR (1) | KR102509431B1 (https=) |
| CN (1) | CN107207465B (https=) |
| AU (1) | AU2015321654B2 (https=) |
| BR (1) | BR112017005713B1 (https=) |
| CA (1) | CA2962329C (https=) |
| ES (1) | ES2849998T3 (https=) |
| RU (1) | RU2704008C2 (https=) |
| TW (1) | TWI598348B (https=) |
| WO (1) | WO2016048861A2 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6982716B2 (ja) * | 2017-01-10 | 2021-12-17 | ナショナル ヘルス リサーチ インスティチューツ | 複素環式化合物及びその使用 |
| IL302338B2 (en) * | 2017-09-08 | 2024-10-01 | Univ Leland Stanford Junior | Enpp1 inhibitors and their use for the treatment of cancer |
| WO2020060268A1 (ko) | 2018-09-20 | 2020-03-26 | 한미약품 주식회사 | 상피세포 성장인자 수용체 돌연변이 저해 효과를 갖는 신규 융합 피리미딘 골격 설폰아마이드 유도체 |
| MX2021009269A (es) * | 2019-02-01 | 2021-08-24 | Univ Leland Stanford Junior | Inhibidores de enpp1 y metodos para modular una respuesta inmunitaria. |
| CN111138417B (zh) * | 2019-12-18 | 2021-03-23 | 浙江工业大学 | 一种三氮唑修饰的5-氟-2,4-嘧啶二胺类化合物及其应用 |
| WO2023014611A1 (en) * | 2021-08-02 | 2023-02-09 | Yeh, Teng-Kuang | Pyrimidine compounds and use thereof |
| WO2024101337A1 (ja) * | 2022-11-07 | 2024-05-16 | 国立大学法人京都大学 | キナゾリン誘導体 |
| TW202435887A (zh) | 2023-03-01 | 2024-09-16 | 瑞士商諾華公司 | 用於治療疾病或障礙的氫喹唑啉衍生物 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4936700A (https=) * | 1972-08-16 | 1974-04-05 | ||
| FI944602A0 (fi) * | 1992-04-03 | 1994-10-03 | Upjohn Co | Farmaseuttisesti aktiiviset bisyklis-heterosykliset amiinit |
| US6156758A (en) * | 1999-09-08 | 2000-12-05 | Isis Pharmaceuticals, Inc. | Antibacterial quinazoline compounds |
| EP2043651A2 (en) | 2006-07-05 | 2009-04-08 | Exelixis, Inc. | Methods of using igf1r and abl kinase modulators |
| AU2009228034A1 (en) * | 2008-03-28 | 2009-10-01 | Altiris Therapeutics | Chemokine receptor modulators |
| CN102046609B (zh) | 2008-03-31 | 2014-05-14 | 全药工业株式会社 | 具有细胞保护效果的嘧啶衍生物及其应用 |
| AU2008355098B2 (en) | 2008-04-21 | 2012-11-15 | Gpcr Therapeutics, Inc | Heterocyclic compounds |
| WO2010046780A2 (en) | 2008-10-22 | 2010-04-29 | Institut Pasteur Korea | Anti viral compounds |
| GB201015411D0 (en) | 2010-09-15 | 2010-10-27 | Univ Leuven Kath | Anti-cancer activity of novel bicyclic heterocycles |
| KR20140069235A (ko) | 2011-09-27 | 2014-06-09 | 노파르티스 아게 | 돌연변이체 idh의 억제제로서의 3-피리미딘-4-일-옥사졸리딘-2-온 |
| CN104379180A (zh) | 2012-04-10 | 2015-02-25 | 佐治亚州立大学研究基金会公司 | 用cyld抑制剂治疗中耳炎及其它病状的组合物和方法 |
| LT2906563T (lt) | 2012-10-10 | 2018-06-11 | Janssen Sciences Ireland Uc | Pirolo[3,2-d]pirimidino dariniai virusinių infekcijų ir kitų ligų gydymui |
| US20150259649A1 (en) | 2012-11-08 | 2015-09-17 | Emory University | Cellular compositions used to restore stem cell or progenitor cell function and methods related thereto |
-
2015
- 2015-09-21 WO PCT/US2015/051143 patent/WO2016048861A2/en not_active Ceased
- 2015-09-21 KR KR1020177010762A patent/KR102509431B1/ko active Active
- 2015-09-21 RU RU2017109355A patent/RU2704008C2/ru active
- 2015-09-21 US US14/860,033 patent/US9862703B2/en active Active
- 2015-09-21 AU AU2015321654A patent/AU2015321654B2/en active Active
- 2015-09-21 ES ES15844487T patent/ES2849998T3/es active Active
- 2015-09-21 JP JP2017535616A patent/JP6615207B2/ja active Active
- 2015-09-21 BR BR112017005713-1A patent/BR112017005713B1/pt active IP Right Grant
- 2015-09-21 CN CN201580050829.5A patent/CN107207465B/zh active Active
- 2015-09-21 EP EP15844487.7A patent/EP3197885B1/en active Active
- 2015-09-21 CA CA2962329A patent/CA2962329C/en active Active
- 2015-09-22 TW TW104131241A patent/TWI598348B/zh active
-
2017
- 2017-09-22 US US15/712,978 patent/US9926298B2/en active Active
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