JP2017512762A5 - - Google Patents
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- Publication number
- JP2017512762A5 JP2017512762A5 JP2016555478A JP2016555478A JP2017512762A5 JP 2017512762 A5 JP2017512762 A5 JP 2017512762A5 JP 2016555478 A JP2016555478 A JP 2016555478A JP 2016555478 A JP2016555478 A JP 2016555478A JP 2017512762 A5 JP2017512762 A5 JP 2017512762A5
- Authority
- JP
- Japan
- Prior art keywords
- hexafluorophosphate
- acid
- compound
- hydrogen
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201461947286P | 2014-03-03 | 2014-03-03 | |
| US61/947,286 | 2014-03-03 | ||
| PCT/US2014/072267 WO2015134096A1 (en) | 2014-03-03 | 2014-12-23 | Pharmaceutically relevant aromatic-cationic peptides |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2017512762A JP2017512762A (ja) | 2017-05-25 |
| JP2017512762A5 true JP2017512762A5 (https=) | 2018-02-08 |
Family
ID=54055710
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016555478A Pending JP2017512762A (ja) | 2014-03-03 | 2014-12-23 | 薬学的に妥当な芳香族カチオン性ペプチド及びその生成方法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20170081363A1 (https=) |
| EP (1) | EP3114136A4 (https=) |
| JP (1) | JP2017512762A (https=) |
| CN (1) | CN106459169A (https=) |
| CA (1) | CA2942143A1 (https=) |
| HK (1) | HK1231493A1 (https=) |
| WO (1) | WO2015134096A1 (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10221213B2 (en) | 2013-12-27 | 2019-03-05 | Stealth Biotherapeutics Corp | Pharmaceutically relevant aromatic-cationic peptides |
| EP3265109B1 (en) | 2015-03-06 | 2020-10-21 | Stealth BioTherapeutics Corp | Processes for preparing pharmaceutically relevant peptides |
| WO2017043626A1 (ja) * | 2015-09-11 | 2017-03-16 | 株式会社カネカ | 光学活性４－カルバモイル－２，６－ジメチルフェニルアラニン誘導体の製造法 |
| WO2017180535A1 (en) | 2016-04-11 | 2017-10-19 | Carnot, Llc | Chiral peptides |
| US11034724B2 (en) | 2017-04-05 | 2021-06-15 | Stealth Biotherapeutics Corp. | Crystalline salt forms of Boc-D-Arg-DMT-Lys-(Boc)-Phe-NH2 |
| US20200361987A1 (en) * | 2017-11-15 | 2020-11-19 | Stealth Biotherapeutics Corp. | Deuterated tetrapeptides that target mitochondria |
| US10676506B2 (en) | 2018-01-26 | 2020-06-09 | Stealth Biotherapeutics Corp. | Crystalline bis- and tris-hydrochloride salt of elamipretide |
| US12252554B2 (en) | 2018-12-18 | 2025-03-18 | Stealth Biotherapeutics Inc. | Analogs that target mitochondrial diseases |
| TW202346255A (zh) * | 2022-01-06 | 2023-12-01 | 日商中外製藥股份有限公司 | 醯胺化合物的製造方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004501875A (ja) * | 2000-06-14 | 2004-01-22 | メダレックス，インコーポレイティド | トリペプチドプロドラッグ化合物 |
| PL2604286T3 (pl) * | 2003-05-01 | 2015-03-31 | Cornell Res Foundation Inc | Sposoby i kompleksy nośnikowe do transportu cząsteczek do komórek |
| US20070213505A1 (en) * | 2006-03-08 | 2007-09-13 | David Epstein | Solution Synthesis of Peptide Cell Growth Stimulators |
| EP3375449A1 (en) * | 2010-03-15 | 2018-09-19 | Stealth Peptides International, Inc. | Combination therapies using cyclosporine and aromatic cationic peptides |
| CA2839408A1 (en) * | 2011-06-14 | 2012-12-20 | Stealth Peptides International, Inc. | Aromatic-cationic peptides and uses of same |
| CN104244964A (zh) * | 2012-02-22 | 2014-12-24 | 康肽德生物医药技术有限公司 | 用于预防或治疗眼科病状的方法和组合物 |
| JP2016506391A (ja) * | 2012-12-06 | 2016-03-03 | ステルス ペプチドズ インターナショナル インコーポレイテッド | ペプチド治療薬およびその使用方法 |
-
2014
- 2014-12-23 JP JP2016555478A patent/JP2017512762A/ja active Pending
- 2014-12-23 CN CN201480078597.XA patent/CN106459169A/zh active Pending
- 2014-12-23 EP EP14884543.1A patent/EP3114136A4/en not_active Withdrawn
- 2014-12-23 US US15/123,437 patent/US20170081363A1/en not_active Abandoned
- 2014-12-23 HK HK17105171.1A patent/HK1231493A1/zh unknown
- 2014-12-23 CA CA2942143A patent/CA2942143A1/en not_active Abandoned
- 2014-12-23 WO PCT/US2014/072267 patent/WO2015134096A1/en not_active Ceased
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