JP2016513704A - チロシンキナーゼ阻害薬の結晶形態物及びその塩 - Google Patents

チロシンキナーゼ阻害薬の結晶形態物及びその塩 Download PDF

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JP2016513704A
JP2016513704A JP2016502487A JP2016502487A JP2016513704A JP 2016513704 A JP2016513704 A JP 2016513704A JP 2016502487 A JP2016502487 A JP 2016502487A JP 2016502487 A JP2016502487 A JP 2016502487A JP 2016513704 A JP2016513704 A JP 2016513704A
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powder
ray diffraction
diffraction pattern
crystalline
cancer
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JP2016513704A5 (enExample
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ジェイ ジィー‐チャン ウー
ジェイ ジィー‐チャン ウー
リン ワン
リン ワン
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ムンディファーマ インターナショナル コーポレイション リミテッド
ムンディファーマ インターナショナル コーポレイション リミテッド
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2016502487A 2013-03-15 2014-03-14 チロシンキナーゼ阻害薬の結晶形態物及びその塩 Pending JP2016513704A (ja)

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US201361801112P 2013-03-15 2013-03-15
US61/801,112 2013-03-15
PCT/US2014/027591 WO2014152663A1 (en) 2013-03-15 2014-03-14 Crystalline forms of tyrosine kinase inhibitors and their salts

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KR (1) KR20150142688A (enExample)
CN (1) CN105377821A (enExample)
AU (1) AU2014239254B2 (enExample)
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WO2016043975A1 (en) 2014-09-17 2016-03-24 Vm Pharma Llc Crystalline forms of tyrosine kinase inhibitors and their salts
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US20160002182A1 (en) 2016-01-07
EA201591684A1 (ru) 2016-02-29
US20170001969A9 (en) 2017-01-05
UA116466C2 (uk) 2018-03-26
NI201500139A (es) 2016-02-16
US9718794B2 (en) 2017-08-01
EP2970148A1 (en) 2016-01-20
EP2970148A4 (en) 2016-10-12
CN105377821A (zh) 2016-03-02
US9388146B2 (en) 2016-07-12
CR20150560A (es) 2016-08-31
PE20151884A1 (es) 2016-01-08
MX2015012403A (es) 2016-04-04
AU2014239254A1 (en) 2015-10-15
SG11201507516XA (en) 2015-10-29
TN2015000407A1 (en) 2017-01-03
BR112015022631A2 (pt) 2017-12-19
HK1220193A1 (zh) 2017-04-28
US20170105990A1 (en) 2017-04-20
US20150174124A1 (en) 2015-06-25
US10124002B2 (en) 2018-11-13
SG10201707484UA (en) 2017-10-30
US9993473B2 (en) 2018-06-12
KR20150142688A (ko) 2015-12-22
US20140275113A1 (en) 2014-09-18
US8999992B2 (en) 2015-04-07
PH12015502110A1 (en) 2016-01-11
AU2014239254B2 (en) 2018-06-28
CL2015002593A1 (es) 2016-08-19
ZA201507154B (en) 2017-09-27
US20180057469A1 (en) 2018-03-01
CA2904403A1 (en) 2014-09-25
GT201500292A (es) 2019-07-29
WO2014152663A1 (en) 2014-09-25
SV2015005074A (es) 2017-07-19

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