JP2016508506A5 - - Google Patents
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- Publication number
- JP2016508506A5 JP2016508506A5 JP2015556454A JP2015556454A JP2016508506A5 JP 2016508506 A5 JP2016508506 A5 JP 2016508506A5 JP 2015556454 A JP2015556454 A JP 2015556454A JP 2015556454 A JP2015556454 A JP 2015556454A JP 2016508506 A5 JP2016508506 A5 JP 2016508506A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- alkyl
- ring
- groups
- ring member
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP13154261.5 | 2013-02-06 | ||
| EP13154261 | 2013-02-06 | ||
| PCT/EP2014/051878 WO2014122067A1 (en) | 2013-02-06 | 2014-01-31 | New indanyloxydihydrobenzofuranylacetic acids |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2016508506A JP2016508506A (ja) | 2016-03-22 |
| JP2016508506A5 true JP2016508506A5 (OSRAM) | 2017-03-09 |
| JP6314335B2 JP6314335B2 (ja) | 2018-04-25 |
Family
ID=47681765
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015556454A Expired - Fee Related JP6314335B2 (ja) | 2013-02-06 | 2014-01-31 | 新しいインダニルオキシジヒドロベンゾフラニル酢酸 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US8927531B2 (OSRAM) |
| EP (1) | EP2953681B1 (OSRAM) |
| JP (1) | JP6314335B2 (OSRAM) |
| AR (1) | AR095163A1 (OSRAM) |
| TW (1) | TW201518284A (OSRAM) |
| UY (1) | UY35312A (OSRAM) |
| WO (1) | WO2014122067A1 (OSRAM) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EA201690888A1 (ru) | 2013-11-14 | 2016-10-31 | Кадила Хелзкэр Лимитед | Новые гетероциклические соединения |
| CN105566263A (zh) * | 2016-01-27 | 2016-05-11 | 中国药科大学 | 一类新型含氮杂环衍生物、其制备方法及其作为药物的用途 |
| JOP20190060A1 (ar) | 2016-09-26 | 2019-03-26 | Chugai Pharmaceutical Co Ltd | مشتق بيرازولو بيريدين له تأثير مساعد لمستقبل glp-1 |
| JP7461104B2 (ja) * | 2017-11-29 | 2024-04-03 | 中外製薬株式会社 | Glp-1受容体アゴニスト作用を持つピラゾロピリジン誘導体を含有する医薬組成物 |
| MY196582A (en) | 2018-02-13 | 2023-04-19 | Gilead Sciences Inc | PD-1/PD-L1 Inhibitors |
| WO2019204609A1 (en) | 2018-04-19 | 2019-10-24 | Gilead Sciences, Inc. | Pd-1/pd-l1 inhibitors |
| PT3820572T (pt) | 2018-07-13 | 2023-11-10 | Gilead Sciences Inc | Inibidores pd-1/pd-l1 |
| EP3870566A1 (en) | 2018-10-24 | 2021-09-01 | Gilead Sciences, Inc. | Pd-1/pd-l1 inhibitors |
| KR20220150270A (ko) | 2019-10-07 | 2022-11-10 | 칼리오페, 인크. | Gpr119 효능제 |
| PL4097099T3 (pl) * | 2020-02-07 | 2024-11-04 | Gasherbrum Bio, Inc. | Heterocykliczne agonisty glp-1 |
| JP7745559B2 (ja) | 2020-02-28 | 2025-09-29 | キャリーオペ,インク. | Gpr40アゴニスト |
| BR112022023359A2 (pt) | 2020-05-19 | 2023-04-18 | Kallyope Inc | Ativadores de ampk |
| JP2023531726A (ja) | 2020-06-26 | 2023-07-25 | キャリーオペ,インク. | Ampkアクチベーター |
| IL322686A (en) | 2023-02-16 | 2025-10-01 | Gasherbrum Bio Inc | Heterocyclic glp-1 agonists |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4594611B2 (ja) * | 2002-11-08 | 2010-12-08 | 武田薬品工業株式会社 | 受容体機能調節剤 |
| CA2505322A1 (en) | 2002-11-08 | 2004-05-21 | Takeda Pharmaceutical Company Limited | Receptor function regulator |
| JP4805552B2 (ja) * | 2003-05-30 | 2011-11-02 | 武田薬品工業株式会社 | 縮合環化合物 |
| EP1924546A1 (en) | 2005-09-14 | 2008-05-28 | Amgen, Inc | Conformationally constrained 3- (4-hydroxy-phenyl) - substituted-propanoic acids useful for treating metabolic disorders |
| EP2001844A2 (en) * | 2006-03-14 | 2008-12-17 | Amgen, Inc | Bicyclic carboxylic acid derivatives useful for treating metabolic disorders |
| EP2431367A3 (en) | 2006-06-27 | 2012-07-04 | Takeda Pharmaceutical Company Limited | Fused cyclic compounds as GPR40 receptor modulators |
| WO2009157418A1 (ja) | 2008-06-25 | 2009-12-30 | 第一三共株式会社 | カルボン酸化合物 |
| WO2010143733A1 (en) * | 2009-06-09 | 2010-12-16 | Takeda Pharmaceutical Company Limited | Novel fused cyclic compound and use thereof |
| ES2546154T3 (es) | 2010-12-01 | 2015-09-21 | Boehringer Ingelheim International Gmbh | Ácidos indaniloxidihidrobenzofuranilacéticos, útiles para el tratamiento del síndrome metabólico |
| US8809376B2 (en) * | 2012-04-30 | 2014-08-19 | Boehringer Ingelheim International Gmbh | Indanyloxydihydrobenzofuranylacetic acids |
-
2014
- 2014-01-31 JP JP2015556454A patent/JP6314335B2/ja not_active Expired - Fee Related
- 2014-01-31 WO PCT/EP2014/051878 patent/WO2014122067A1/en not_active Ceased
- 2014-01-31 EP EP14702030.9A patent/EP2953681B1/en not_active Not-in-force
- 2014-02-03 US US14/170,660 patent/US8927531B2/en active Active
- 2014-02-05 AR ARP140100390A patent/AR095163A1/es unknown
- 2014-02-05 TW TW103103836A patent/TW201518284A/zh unknown
- 2014-02-06 UY UY0001035312A patent/UY35312A/es unknown
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