JP2016506417A - キナーゼ阻害剤の治療指標 - Google Patents

キナーゼ阻害剤の治療指標 Download PDF

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JP2016506417A
JP2016506417A JP2015552755A JP2015552755A JP2016506417A JP 2016506417 A JP2016506417 A JP 2016506417A JP 2015552755 A JP2015552755 A JP 2015552755A JP 2015552755 A JP2015552755 A JP 2015552755A JP 2016506417 A JP2016506417 A JP 2016506417A
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ジスマン、ローレンス、エス.
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プルモキネ、インコーポレイテッド
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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JP2015552755A 2013-01-10 2014-01-09 キナーゼ阻害剤の治療指標 Pending JP2016506417A (ja)

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US201361751217P 2013-01-10 2013-01-10
US61/751,217 2013-01-10
PCT/US2014/010773 WO2014110198A2 (en) 2013-01-10 2014-01-09 Therapeutic indications of kinase inhibitors

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AU (1) AU2014205481A1 (enExample)
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WO (1) WO2014110198A2 (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2016506418A (ja) * 2013-01-10 2016-03-03 プルモキネ、インコーポレイテッド 非選択的キナーゼ阻害剤
JP2016534153A (ja) * 2013-10-11 2016-11-04 ローレンス エス. ジスマン, 噴霧乾燥製剤
US10231966B2 (en) 2016-10-27 2019-03-19 Pulmokine, Inc. Combination therapy for treating pulmonary hypertension

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113244399A (zh) 2015-01-26 2021-08-13 耶鲁大学 利用酪氨酸激酶抑制剂的组合物和方法
JP2022532431A (ja) * 2019-05-16 2022-07-14 エアロベイト セラピューティクス, インコーポレイテッド イマチニブ製剤、その製造および使用
US20240325390A1 (en) * 2020-11-23 2024-10-03 Aerovate Therapeutics, Inc. Imatinib formulations, manufacture, and uses thereof

Citations (3)

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JP2005535596A (ja) * 2002-05-23 2005-11-24 サイトピア・リサーチ・ピーティーワイ・リミテッド プロテインキナーゼ阻害剤
JP2010509375A (ja) * 2006-11-15 2010-03-25 サイトピア・リサーチ・ピーティーワイ・リミテッド キナーゼ活性の阻害剤
JP2016506418A (ja) * 2013-01-10 2016-03-03 プルモキネ、インコーポレイテッド 非選択的キナーゼ阻害剤

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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