JP2016505534A5 - - Google Patents
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- Publication number
- JP2016505534A5 JP2016505534A5 JP2015543399A JP2015543399A JP2016505534A5 JP 2016505534 A5 JP2016505534 A5 JP 2016505534A5 JP 2015543399 A JP2015543399 A JP 2015543399A JP 2015543399 A JP2015543399 A JP 2015543399A JP 2016505534 A5 JP2016505534 A5 JP 2016505534A5
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12193311.3 | 2012-11-20 | ||
| EP12193311 | 2012-11-20 | ||
| PCT/EP2013/074012 WO2014079787A1 (en) | 2012-11-20 | 2013-11-18 | Substituted 1,6-naphthyridines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2016505534A JP2016505534A (ja) | 2016-02-25 |
| JP2016505534A5 true JP2016505534A5 (enExample) | 2017-01-05 |
Family
ID=47189816
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015543399A Pending JP2016505534A (ja) | 2012-11-20 | 2013-11-18 | 置換1,6−ナフチリジン |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US9657014B2 (enExample) |
| EP (1) | EP2922540A1 (enExample) |
| JP (1) | JP2016505534A (enExample) |
| KR (1) | KR20150085538A (enExample) |
| CN (1) | CN104812387A (enExample) |
| AR (1) | AR093519A1 (enExample) |
| BR (1) | BR112015011094A2 (enExample) |
| CA (1) | CA2890685A1 (enExample) |
| HK (1) | HK1207317A1 (enExample) |
| MX (1) | MX2015006364A (enExample) |
| RU (1) | RU2015120217A (enExample) |
| TW (1) | TW201425312A (enExample) |
| WO (1) | WO2014079787A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI529171B (zh) * | 2013-07-29 | 2016-04-11 | 赫孚孟拉羅股份公司 | 1,7-萘啶衍生物 |
| CN106817900A (zh) * | 2014-07-17 | 2017-06-09 | 默克专利有限公司 | 新颖的萘啶和异喹啉及其作为cdk8/19抑制剂的用途 |
| AU2016217874A1 (en) * | 2015-02-11 | 2017-08-10 | Basilea Pharmaceutica International AG | Substituted mono- and polyazanaphthalene derivatives and their use |
| CN108299425B (zh) * | 2015-03-24 | 2020-09-18 | 上海璎黎药业有限公司 | 稠环衍生物、其制备方法、中间体、药物组合物及应用 |
| CN108349936B (zh) | 2015-11-06 | 2021-10-01 | 纽罗克里生物科学有限公司 | 作为毒蕈碱性受体4拮抗剂的化合物 |
| EA039638B1 (ru) * | 2016-01-06 | 2022-02-21 | Нейрокрин Байосайенсиз, Инк. | Антагонисты мускаринового рецептора 4 и способы их применения |
| WO2018159805A1 (ja) | 2017-03-03 | 2018-09-07 | 国立大学法人京都大学 | 膵前駆細胞の製造方法 |
| JP7566753B2 (ja) | 2019-01-03 | 2024-10-15 | ユニバーシティ オブ ピッツバーグ -オブ ザ コモンウェルス システム オブ ハイヤー エデュケイション | 転写因子ebポリペプチドレベルを増加させるための方法および材料 |
| TW202134231A (zh) | 2019-12-06 | 2021-09-16 | 美商紐羅克里生物科學有限公司 | 蕈毒受體4拮抗劑及使用方法 |
| IL303924A (en) * | 2020-12-18 | 2023-08-01 | Scripps Research Inst | Compounds and use thereof for treatment of neurodegenerative, degenerative and metabolic disorders |
| WO2025252732A1 (en) * | 2024-06-04 | 2025-12-11 | Syngenta Crop Protection Ag | Nitrogen-containing 6-membered bicyclic derivatives with microbiocidal activity |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9605437D0 (en) | 1996-03-15 | 1996-05-15 | Iaf Biochem Int | Cytomegalovirus inhibiting compounds |
| BR9815166A (pt) * | 1997-12-11 | 2000-10-10 | Iaf Biochem Int | "método de inibição da replicação de vìrus, composto, método de inibição da replicação de citomegalovìrus, composto antiviral, utilização de um composto, composição farmacêutica, composição farmacêutica inibidora da replicação de vìrus e de citomegalovìrus e composição farmacêutica antiviral" |
| WO2002051413A2 (en) | 2000-12-27 | 2002-07-04 | Shire Biochem Inc. | Macrocyclic anti-viral compounds |
| EP1773834A2 (en) | 2004-08-03 | 2007-04-18 | Serenex, Inc. | 2, 8-disubstituted naphthyridine derivatives |
| FR2904317A1 (fr) | 2006-07-27 | 2008-02-01 | Inst Nat Sante Rech Med | Analogues d'halogenobenzamides marques a titre de radiopharmaceutiques |
| US20080242694A1 (en) | 2006-09-18 | 2008-10-02 | D Sidocky Neil R | Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith |
| WO2008046072A2 (en) | 2006-10-13 | 2008-04-17 | The Board Of Regents Of The University Of Texas System | Chemical inducers of neurogenesis |
| NZ593996A (en) * | 2009-01-19 | 2012-10-26 | Daiichi Sankyo Co Ltd | Naphthyridine-carboxamide and isoquinoline-carboxamide derivatives for treating osteoporosis |
| BRPI1011477A2 (pt) * | 2009-03-02 | 2016-03-22 | Sirtris Pharmaceuticals Inc | quinolinas 8-substituidas e analogos relacionados como moduladores de sirtuina |
| JP5698658B2 (ja) | 2009-04-06 | 2015-04-08 | 第一三共株式会社 | 置換フェニル基を有する環状化合物 |
| DK2590647T3 (en) | 2010-07-07 | 2018-02-12 | Univ Texas | Pro-neurogenic compounds |
| JP2012036168A (ja) | 2010-07-15 | 2012-02-23 | Daiichi Sankyo Co Ltd | ヘテロ原子を有する環状化合物を含有する医薬組成物 |
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2013
- 2013-11-18 CA CA2890685A patent/CA2890685A1/en not_active Abandoned
- 2013-11-18 RU RU2015120217A patent/RU2015120217A/ru not_active Application Discontinuation
- 2013-11-18 MX MX2015006364A patent/MX2015006364A/es unknown
- 2013-11-18 WO PCT/EP2013/074012 patent/WO2014079787A1/en not_active Ceased
- 2013-11-18 HK HK15108069.2A patent/HK1207317A1/xx unknown
- 2013-11-18 KR KR1020157016208A patent/KR20150085538A/ko not_active Ceased
- 2013-11-18 JP JP2015543399A patent/JP2016505534A/ja active Pending
- 2013-11-18 TW TW102141946A patent/TW201425312A/zh unknown
- 2013-11-18 BR BR112015011094A patent/BR112015011094A2/pt not_active IP Right Cessation
- 2013-11-18 EP EP13795705.6A patent/EP2922540A1/en not_active Withdrawn
- 2013-11-18 CN CN201380060294.0A patent/CN104812387A/zh active Pending
- 2013-11-18 AR ARP130104234A patent/AR093519A1/es unknown
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2015
- 2015-05-20 US US14/717,109 patent/US9657014B2/en not_active Expired - Fee Related