JP2016505534A5 - - Google Patents

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Publication number
JP2016505534A5
JP2016505534A5 JP2015543399A JP2015543399A JP2016505534A5 JP 2016505534 A5 JP2016505534 A5 JP 2016505534A5 JP 2015543399 A JP2015543399 A JP 2015543399A JP 2015543399 A JP2015543399 A JP 2015543399A JP 2016505534 A5 JP2016505534 A5 JP 2016505534A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2015543399A
Other languages
English (en)
Japanese (ja)
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JP2016505534A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2013/074012 external-priority patent/WO2014079787A1/en
Publication of JP2016505534A publication Critical patent/JP2016505534A/ja
Publication of JP2016505534A5 publication Critical patent/JP2016505534A5/ja
Pending legal-status Critical Current

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JP2015543399A 2012-11-20 2013-11-18 置換1,6−ナフチリジン Pending JP2016505534A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12193311 2012-11-20
EP12193311.3 2012-11-20
PCT/EP2013/074012 WO2014079787A1 (en) 2012-11-20 2013-11-18 Substituted 1,6-naphthyridines

Publications (2)

Publication Number Publication Date
JP2016505534A JP2016505534A (ja) 2016-02-25
JP2016505534A5 true JP2016505534A5 (cg-RX-API-DMAC7.html) 2017-01-05

Family

ID=47189816

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015543399A Pending JP2016505534A (ja) 2012-11-20 2013-11-18 置換1,6−ナフチリジン

Country Status (13)

Country Link
US (1) US9657014B2 (cg-RX-API-DMAC7.html)
EP (1) EP2922540A1 (cg-RX-API-DMAC7.html)
JP (1) JP2016505534A (cg-RX-API-DMAC7.html)
KR (1) KR20150085538A (cg-RX-API-DMAC7.html)
CN (1) CN104812387A (cg-RX-API-DMAC7.html)
AR (1) AR093519A1 (cg-RX-API-DMAC7.html)
BR (1) BR112015011094A2 (cg-RX-API-DMAC7.html)
CA (1) CA2890685A1 (cg-RX-API-DMAC7.html)
HK (1) HK1207317A1 (cg-RX-API-DMAC7.html)
MX (1) MX2015006364A (cg-RX-API-DMAC7.html)
RU (1) RU2015120217A (cg-RX-API-DMAC7.html)
TW (1) TW201425312A (cg-RX-API-DMAC7.html)
WO (1) WO2014079787A1 (cg-RX-API-DMAC7.html)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI529171B (zh) * 2013-07-29 2016-04-11 赫孚孟拉羅股份公司 1,7-萘啶衍生物
AU2015289044A1 (en) * 2014-07-17 2016-12-08 Cancer Research Technology Limited Novel naphthryidines and isoquinolines and their use as CDK8/19 inhibitors
BR112017017032A2 (pt) * 2015-02-11 2018-04-10 Basilea Pharmaceutica International AG derivados de mono e poliazanaftaleno substituídos e uso dos mesmos
CN108516958B (zh) 2015-03-24 2020-07-17 上海璎黎药业有限公司 稠环衍生物、其制备方法、中间体、药物组合物及应用
SG11201803757UA (en) 2015-11-06 2018-06-28 Neurocrine Biosciences Inc N-[2-(1 -benzylpiperidin-4-yl)ethyl]-4-(pyrazin-2-yl)-piperazine-1 -carboxamide derivatives and related compounds as muscarinic receptor 4 (m4) antagonists for treating neurological diseases
EA039638B1 (ru) * 2016-01-06 2022-02-21 Нейрокрин Байосайенсиз, Инк. Антагонисты мускаринового рецептора 4 и способы их применения
JPWO2018159805A1 (ja) 2017-03-03 2020-01-09 国立大学法人京都大学 膵前駆細胞の製造方法
BR112021012950A2 (pt) 2019-01-03 2021-09-14 University Of Pittsburgh - Of The Commonwealth System Of Higher Education Métodos e materiais para aumentar os níveis de polipeptídeo do fator de transcrição eb
ES2983860T3 (es) 2019-12-06 2024-10-25 Neurocrine Biosciences Inc Antagonistas del receptor muscarínico 4 y métodos de uso
CA3202961A1 (en) * 2020-12-18 2022-06-23 The Scripps Research Institute Compounds and use thereof for treatment of neurodegenerative, degenerative and metabolic disorders
WO2025252732A1 (en) * 2024-06-04 2025-12-11 Syngenta Crop Protection Ag Nitrogen-containing 6-membered bicyclic derivatives with microbiocidal activity

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9605437D0 (en) 1996-03-15 1996-05-15 Iaf Biochem Int Cytomegalovirus inhibiting compounds
DE69818094T2 (de) * 1997-12-11 2004-07-08 Biochem Pharma Inc., Laval Antivirale verbindungen
AU2002218902A1 (en) 2000-12-27 2002-07-08 Shire Biochem Inc. Macrocyclic anti-viral compounds
JP2008509151A (ja) 2004-08-03 2008-03-27 セレネックス, インコーポレイテッド 2,8−二置換ナフチリジン誘導体
FR2904317A1 (fr) 2006-07-27 2008-02-01 Inst Nat Sante Rech Med Analogues d'halogenobenzamides marques a titre de radiopharmaceutiques
US20080242694A1 (en) 2006-09-18 2008-10-02 D Sidocky Neil R Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith
WO2008046072A2 (en) 2006-10-13 2008-04-17 The Board Of Regents Of The University Of Texas System Chemical inducers of neurogenesis
NZ593996A (en) * 2009-01-19 2012-10-26 Daiichi Sankyo Co Ltd Naphthyridine-carboxamide and isoquinoline-carboxamide derivatives for treating osteoporosis
MX2011009213A (es) 2009-03-02 2011-12-14 Sirtris Pharmaceuticals Inc Quinolinas 8-sustituidas y analogos relacionados como moduladores de sirtuina.
WO2010116915A1 (ja) * 2009-04-06 2010-10-14 第一三共株式会社 置換フェニル基を有する環状化合物
EP2590647B1 (en) 2010-07-07 2017-11-08 Board of Regents of the University of Texas System Pro-neurogenic compounds
JP2012036168A (ja) 2010-07-15 2012-02-23 Daiichi Sankyo Co Ltd ヘテロ原子を有する環状化合物を含有する医薬組成物

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