JP2015533163A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2015533163A5 JP2015533163A5 JP2015536853A JP2015536853A JP2015533163A5 JP 2015533163 A5 JP2015533163 A5 JP 2015533163A5 JP 2015536853 A JP2015536853 A JP 2015536853A JP 2015536853 A JP2015536853 A JP 2015536853A JP 2015533163 A5 JP2015533163 A5 JP 2015533163A5
- Authority
- JP
- Japan
- Prior art keywords
- multiple sclerosis
- laquinimod
- relapsing
- presenting
- preventing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 201000006417 multiple sclerosis Diseases 0.000 claims 3
- 206010071068 Clinically isolated syndrome Diseases 0.000 claims 1
- GKWPCEFFIHSJOE-UHFFFAOYSA-N Laquinimod Chemical compound OC=1C2=C(Cl)C=CC=C2N(C)C(=O)C=1C(=O)N(CC)C1=CC=CC=C1 GKWPCEFFIHSJOE-UHFFFAOYSA-N 0.000 claims 1
- 208000007400 Relapsing-Remitting Multiple Sclerosis Diseases 0.000 claims 1
- 229960004577 laquinimod Drugs 0.000 claims 1
- 239000008203 oral pharmaceutical composition Substances 0.000 claims 1
- 230000000750 progressive Effects 0.000 claims 1
- 230000000542 thalamic Effects 0.000 claims 1
Claims (1)
- ある形態の多発性硬化症に罹患し、または臨床的に摘出された症候群を呈するヒト被験者における視床損傷を阻止または低減するための、有効量のラキニモドを含有する経口医薬組成物であって、好ましくは、前記形態の多発性硬化症は、再発−寛解型の多発性硬化症または進行性形態の多発性硬化症である経口医薬組成物。
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261713256P | 2012-10-12 | 2012-10-12 | |
US61/713,256 | 2012-10-12 | ||
PCT/US2013/064061 WO2014058979A2 (en) | 2012-10-12 | 2013-10-09 | Laquinimod for reducing thalamic damage in multiple sclerosis |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2015533163A JP2015533163A (ja) | 2015-11-19 |
JP2015533163A5 true JP2015533163A5 (ja) | 2016-11-24 |
Family
ID=50475887
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2015536853A Pending JP2015533163A (ja) | 2012-10-12 | 2013-10-09 | 多発性硬化症における視床損傷を低減するためのラキニモド |
Country Status (18)
Country | Link |
---|---|
US (2) | US20140107154A1 (ja) |
EP (1) | EP2961406A4 (ja) |
JP (1) | JP2015533163A (ja) |
KR (1) | KR20150080509A (ja) |
CN (1) | CN105263325A (ja) |
AR (1) | AR092993A1 (ja) |
AU (2) | AU2013329348A1 (ja) |
BR (1) | BR112015007782A2 (ja) |
CA (1) | CA2884272A1 (ja) |
CL (2) | CL2015000732A1 (ja) |
EA (1) | EA201590726A1 (ja) |
HK (1) | HK1218865A1 (ja) |
IL (1) | IL237745A0 (ja) |
MX (1) | MX2015004564A (ja) |
PE (1) | PE20151435A1 (ja) |
SG (1) | SG11201501874TA (ja) |
TW (1) | TW201420101A (ja) |
WO (1) | WO2014058979A2 (ja) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN106063787A (zh) | 2012-02-03 | 2016-11-02 | 泰华制药工业有限公司 | 拉喹莫德用于治疗一线抗TNFα疗法失败的克罗恩氏病患者的用途 |
EP3225617A1 (en) | 2012-02-16 | 2017-10-04 | Teva Pharmaceutical Industries Ltd | N-ethyl-n-phenyl-1,2-dihydro-4,5-di-hydroxy-1-methyl-2-oxo-3-quinoline carboxamide, preparation and uses thereof |
TW201400117A (zh) | 2012-06-05 | 2014-01-01 | Teva Pharma | 使用拉喹莫德治療眼發炎疾病 |
TW201410244A (zh) | 2012-08-13 | 2014-03-16 | Teva Pharma | 用於治療gaba媒介之疾病之拉喹莫德(laquinimod) |
JP2016510343A (ja) * | 2013-02-15 | 2016-04-07 | テバ ファーマシューティカル インダストリーズ リミティド | ラキニモドを用いる多発性硬化症の治療 |
TW201609098A (zh) * | 2013-12-20 | 2016-03-16 | 泰瓦藥品工業有限公司 | 拉喹莫德(laquinimod)於延緩亨丁頓舞蹈症進展的用途 |
CA2945978A1 (en) | 2014-04-29 | 2015-11-05 | Teva Pharmaceutical Industries Ltd. | Laquinimod for the treatment of relapsing-remitting multiple sclerosis (rrms) patients with a high disability status |
EA201791982A1 (ru) | 2015-03-09 | 2020-02-17 | Интекрин Терапьютикс, Инк. | Способы лечения неалкогольной жировой болезни печени и/или липодистрофии |
WO2017048457A1 (en) * | 2015-09-18 | 2017-03-23 | Teva Pharmaceuticals Industries Ltd. | Combination of laquinimod and pridopidine to treat multiple sclerosis |
US20190224186A1 (en) * | 2016-09-13 | 2019-07-25 | Intekrin Therapeutics, Inc. | Treatment of multiple sclerosis with chs-131 |
EP3606527A1 (en) | 2017-04-03 | 2020-02-12 | Coherus Biosciences, Inc. | Ppar-gamma agonist for treatment of progressive supranuclear palsy |
CN113397757A (zh) * | 2021-06-07 | 2021-09-17 | 温州医科大学 | 用于测试拉喹莫德在治疗缺血性脑卒中的作用的方法 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2595159A1 (en) * | 2005-01-13 | 2006-07-20 | Sirtris Pharmaceuticals, Inc. | Novel compositions for preventing and treating neurodegenerative and blood coagulation disorders |
JP2009543823A (ja) * | 2006-07-17 | 2009-12-10 | ノバルティス アクチエンゲゼルシャフト | 免疫調節剤として使用するための胆汁酸アミドのスルホニルアミノカルボニル誘導体 |
AR073295A1 (es) * | 2008-09-16 | 2010-10-28 | Genentech Inc | Metodos para tratar la esclerosis multiple progresiva. articulo de fabricacion. |
ES2548999T3 (es) * | 2009-06-19 | 2015-10-22 | Teva Pharmaceutical Industries Ltd. | Tratamiento de la esclerosis múltiple con laquinimod |
JP5859438B2 (ja) * | 2009-08-10 | 2016-02-10 | テバ ファーマシューティカル インダストリーズ リミティド | ラキニモドを用いたbdnf関連疾患の治療 |
US20130035390A1 (en) * | 2010-01-13 | 2013-02-07 | Ramot At Tel-Aviv University Ltd. | Treatment of multiple sclerosis |
SG10201509831XA (en) * | 2010-12-07 | 2015-12-30 | Teva Pharma | Use of laquinimod for reducing fatigue, improving functional status, and improving quality of life in multiple sclerosis patients |
WO2012131539A1 (en) * | 2011-03-31 | 2012-10-04 | Pfizer Inc. | Novel bicyclic pyridinones |
SG11201401330YA (en) * | 2011-10-12 | 2014-05-29 | Teva Pharma | Treatment of multiple sclerosis with combination of laquinimod and fingolimod |
TW201347762A (zh) * | 2012-05-02 | 2013-12-01 | Teva Pharma | 高劑量拉喹莫德(laquinimod)於治療多發性硬化症之用途 |
-
2013
- 2013-10-09 CA CA2884272A patent/CA2884272A1/en not_active Abandoned
- 2013-10-09 PE PE2015000472A patent/PE20151435A1/es not_active Application Discontinuation
- 2013-10-09 EA EA201590726A patent/EA201590726A1/ru unknown
- 2013-10-09 EP EP13895446.6A patent/EP2961406A4/en not_active Withdrawn
- 2013-10-09 US US14/049,411 patent/US20140107154A1/en not_active Abandoned
- 2013-10-09 AU AU2013329348A patent/AU2013329348A1/en not_active Abandoned
- 2013-10-09 KR KR1020157012465A patent/KR20150080509A/ko not_active Application Discontinuation
- 2013-10-09 WO PCT/US2013/064061 patent/WO2014058979A2/en active Application Filing
- 2013-10-09 CN CN201380053184.1A patent/CN105263325A/zh active Pending
- 2013-10-09 SG SG11201501874TA patent/SG11201501874TA/en unknown
- 2013-10-09 BR BR112015007782A patent/BR112015007782A2/pt active Search and Examination
- 2013-10-09 JP JP2015536853A patent/JP2015533163A/ja active Pending
- 2013-10-09 MX MX2015004564A patent/MX2015004564A/es unknown
- 2013-10-11 TW TW102136847A patent/TW201420101A/zh unknown
- 2013-10-11 AR ARP130103705A patent/AR092993A1/es unknown
-
2015
- 2015-03-15 IL IL237745A patent/IL237745A0/en unknown
- 2015-03-23 CL CL2015000732A patent/CL2015000732A1/es unknown
-
2016
- 2016-06-15 HK HK16106893.7A patent/HK1218865A1/zh unknown
- 2016-06-17 US US15/186,163 patent/US20160296511A1/en not_active Abandoned
- 2016-11-11 CL CL2016002873A patent/CL2016002873A1/es unknown
-
2017
- 2017-06-08 AU AU2017203896A patent/AU2017203896A1/en not_active Abandoned
Similar Documents
Publication | Publication Date | Title |
---|---|---|
JP2015533163A5 (ja) | ||
HRP20210819T1 (hr) | Fenfluramin za uporabu u liječenju dravet sindroma | |
CL2016002132A1 (es) | Uso de una cantidad de laquinimod, que sirve para preparar un medicamento para tratar un paciente humano afectado con esclerosis múltiple o que presenta un síndrome clínicamente aislado; un paquete, una cantidad de laquinimod y una composición farmacéutica del mismo. | |
JP2016518337A5 (ja) | ||
JP2013520167A5 (ja) | ||
MX355065B (es) | Método y dispositivo para conmutación de cámaras. | |
JP2014507446A5 (ja) | ||
JP2014515597A5 (ja) | ||
CL2013001602A1 (es) | Metodo para reducir o inhibir la progresion del nivel de fatiga en pacientes con esclerosis multiple y para proporcionarles neuroproteccion que comprende administrar oralmente laquinimod o una sal del mismo; laquinimod para reducir el nivel de fatiga, mejorar el estado funcional y entregar neuroproteccion en esclerosis multiple. | |
JP2015525757A5 (ja) | ||
JP2012126725A5 (ja) | ||
WO2015077503A8 (en) | Autotaxin inhibitor compounds | |
BR112014010177A2 (pt) | composto, composição farmacêutica, uso do composto, e, método para a profilaxia ou tratamento de um estado ou uma condição de doença | |
EP3682875A3 (en) | Methods of treating pediatric metabolic syndrome | |
JP2014530840A5 (ja) | ||
CL2014000844A1 (es) | Formulacion farmaceutica oral de liberacion prolongada en forma de multiparticulas, que comprende a) 40-o-(2-hidroxi)etil-rapamicina y b) al menos un recubrimiento de liberacion prolongada. | |
JP2015534562A5 (ja) | ||
AR090491A1 (es) | Tratamiento de la esclerosis multiple con una combinacion de laquinimod y fumarato de dimetilo | |
WO2014058979A8 (en) | Laquinimod for reducing thalamic damage in multiple sclerosis | |
JP2015528502A5 (ja) | ||
JP2017514871A5 (ja) | ||
JP2012193216A5 (ja) | ||
WO2013003669A3 (en) | Compositions, methods of use, and methods of treatment | |
JP2014526468A5 (ja) | ||
BR112012003280A2 (pt) | composição farmacêutica para administração oral, método para tratar uma doença, uso do composto, e, composto. |