JP2015500293A5 - - Google Patents
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- Publication number
- JP2015500293A5 JP2015500293A5 JP2014546080A JP2014546080A JP2015500293A5 JP 2015500293 A5 JP2015500293 A5 JP 2015500293A5 JP 2014546080 A JP2014546080 A JP 2014546080A JP 2014546080 A JP2014546080 A JP 2014546080A JP 2015500293 A5 JP2015500293 A5 JP 2015500293A5
- Authority
- JP
- Japan
- Prior art keywords
- neuropeptide
- receptor antagonist
- pharmaceutical composition
- aryl
- receptor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161568540P | 2011-12-08 | 2011-12-08 | |
| US61/568,540 | 2011-12-08 | ||
| PCT/US2012/068257 WO2013086200A1 (en) | 2011-12-08 | 2012-12-06 | Composition and method for neuropeptide s receptor (npsr) antagonists |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015500293A JP2015500293A (ja) | 2015-01-05 |
| JP2015500293A5 true JP2015500293A5 (https=) | 2015-12-24 |
| JP6381445B2 JP6381445B2 (ja) | 2018-08-29 |
Family
ID=48574884
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014546080A Active JP6381445B2 (ja) | 2011-12-08 | 2012-12-06 | ニューロペプチドｓレセプター（ｎｐｓｒ）アンタゴニストの組成物および方法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US9150582B2 (https=) |
| EP (1) | EP2788359B1 (https=) |
| JP (1) | JP6381445B2 (https=) |
| AU (1) | AU2012347758B2 (https=) |
| CA (1) | CA2858571C (https=) |
| ES (1) | ES2624853T3 (https=) |
| WO (1) | WO2013086200A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2017246706B2 (en) * | 2016-04-04 | 2020-09-17 | Research Triangle Institute | Neuropeptide s receptor (NPSR) agonists |
| JOP20190060A1 (ar) * | 2016-09-26 | 2019-03-26 | Chugai Pharmaceutical Co Ltd | مشتق بيرازولو بيريدين له تأثير مساعد لمستقبل glp-1 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4917489B1 (https=) * | 1970-01-22 | 1974-05-01 | ||
| DE3469531D1 (en) * | 1983-09-15 | 1988-04-07 | Ciba Geigy Ag | 5- and 6-azaphthalides, their mixture of isomers, process for their production and their use in recording materials which are sensitive to pressure and heat |
| WO1992009577A1 (en) * | 1990-11-22 | 1992-06-11 | Janssen Pharmaceutica N.V. | Isonicotinic acid derivatives and related spiro compounds with herbicidal action |
| AU2001294239A1 (en) | 2000-10-13 | 2002-04-22 | Takeda Chemical Industries Ltd. | Novel g protein-coupled receptor protein and dna thereof |
| US6642255B2 (en) | 2001-01-11 | 2003-11-04 | Bristol-Myers Squibb Pharma Company | 1,2,-Disubstituted cyclic inhibitors of matrix metalloproteases and TNF-alpha |
| US9012407B2 (en) * | 2004-04-23 | 2015-04-21 | The Regents Of The University Of California | Therapies which act on neuropeptide S receptors |
| US8541595B2 (en) * | 2008-11-13 | 2013-09-24 | Merch Sharp & Dohme Corp. | Imidazoisoindole neuropeptide S receptor antagonists |
| WO2010056564A1 (en) * | 2008-11-13 | 2010-05-20 | Merck Sharp & Dohme Corp. | Quinolone neuropeptide s receptor antagonists |
-
2012
- 2012-12-06 WO PCT/US2012/068257 patent/WO2013086200A1/en not_active Ceased
- 2012-12-06 EP EP12854821.1A patent/EP2788359B1/en active Active
- 2012-12-06 CA CA2858571A patent/CA2858571C/en active Active
- 2012-12-06 US US14/363,079 patent/US9150582B2/en active Active
- 2012-12-06 AU AU2012347758A patent/AU2012347758B2/en active Active
- 2012-12-06 JP JP2014546080A patent/JP6381445B2/ja active Active
- 2012-12-06 ES ES12854821.1T patent/ES2624853T3/es active Active
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