JP2014532744A - バニロイド受容体リガンドとしての、ｓｏ２含有基で置換されたフェニル部分を担持する置換ピラゾリルをベースとするカルボキサミドおよび尿素誘導体 - Google Patents
バニロイド受容体リガンドとしての、ｓｏ２含有基で置換されたフェニル部分を担持する置換ピラゾリルをベースとするカルボキサミドおよび尿素誘導体 Download PDFInfo
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- JP2014532744A JP2014532744A JP2014540456A JP2014540456A JP2014532744A JP 2014532744 A JP2014532744 A JP 2014532744A JP 2014540456 A JP2014540456 A JP 2014540456A JP 2014540456 A JP2014540456 A JP 2014540456A JP 2014532744 A JP2014532744 A JP 2014532744A
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- methyl
- phenyl
- fluoro
- pyrazol
- methylsulfonyl
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- 239000000203 mixture Substances 0.000 claims description 53
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- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- Health & Medical Sciences (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11008927 | 2011-11-09 | ||
| EP11008927.3 | 2011-11-09 | ||
| PCT/EP2012/072143 WO2013068464A1 (en) | 2011-11-09 | 2012-11-08 | Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2014532744A true JP2014532744A (ja) | 2014-12-08 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014540456A Withdrawn JP2014532744A (ja) | 2011-11-09 | 2012-11-08 | バニロイド受容体リガンドとしての、ｓｏ２含有基で置換されたフェニル部分を担持する置換ピラゾリルをベースとするカルボキサミドおよび尿素誘導体 |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP2776401A1 (OSRAM) |
| JP (1) | JP2014532744A (OSRAM) |
| KR (1) | KR20140091041A (OSRAM) |
| CN (1) | CN104066720A (OSRAM) |
| AR (1) | AR088799A1 (OSRAM) |
| AU (1) | AU2012334068A1 (OSRAM) |
| BR (1) | BR112014011108A2 (OSRAM) |
| CA (1) | CA2854424A1 (OSRAM) |
| HK (1) | HK1202117A1 (OSRAM) |
| IN (1) | IN2014KN00865A (OSRAM) |
| MX (1) | MX2014005233A (OSRAM) |
| TW (1) | TW201326135A (OSRAM) |
| WO (1) | WO2013068464A1 (OSRAM) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| LT3113772T (lt) | 2014-03-07 | 2020-12-28 | Biocryst Pharmaceuticals, Inc. | Trifluormetilo pakeistieji pirazolai kaip žmogaus plazmos kalikreino inhibitoriai |
| CN107108593B (zh) * | 2014-11-24 | 2020-03-24 | 美迪福伦Dbt有限公司 | 作为类香草素受体配体ii的基于取代的恶唑和噻唑的羧酰胺和脲衍生物 |
| CN114920697A (zh) * | 2022-05-16 | 2022-08-19 | 河南应用技术职业学院 | 杂环基取代的茚满丙酰胺类化合物及其应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2758289A1 (en) | 2009-05-07 | 2010-11-11 | Gruenenthal Gmbh | Substituted aromatic carboxamide and urea derivatives as vanilloid receptor ligands |
| JP5745505B2 (ja) | 2009-05-07 | 2015-07-08 | グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング | バニロイド受容体リガンドとしての置換フェニル尿素および置換フェニルアミド |
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2012
- 2012-11-08 EP EP12783220.2A patent/EP2776401A1/en not_active Withdrawn
- 2012-11-08 CA CA2854424A patent/CA2854424A1/en not_active Abandoned
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- 2012-11-08 AU AU2012334068A patent/AU2012334068A1/en not_active Abandoned
- 2012-11-08 JP JP2014540456A patent/JP2014532744A/ja not_active Withdrawn
- 2012-11-08 MX MX2014005233A patent/MX2014005233A/es not_active Application Discontinuation
- 2012-11-08 BR BR112014011108A patent/BR112014011108A2/pt not_active IP Right Cessation
- 2012-11-08 TW TW101141483A patent/TW201326135A/zh unknown
- 2012-11-08 WO PCT/EP2012/072143 patent/WO2013068464A1/en not_active Ceased
- 2012-11-08 KR KR1020147015421A patent/KR20140091041A/ko not_active Withdrawn
- 2012-11-08 HK HK15102581.4A patent/HK1202117A1/xx unknown
- 2012-11-08 CN CN201280055221.8A patent/CN104066720A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| HK1202117A1 (en) | 2015-09-18 |
| CN104066720A (zh) | 2014-09-24 |
| BR112014011108A2 (pt) | 2017-05-16 |
| AR088799A1 (es) | 2014-07-10 |
| MX2014005233A (es) | 2014-08-22 |
| CA2854424A1 (en) | 2013-05-16 |
| IN2014KN00865A (OSRAM) | 2015-10-02 |
| EP2776401A1 (en) | 2014-09-17 |
| AU2012334068A1 (en) | 2014-05-22 |
| TW201326135A (zh) | 2013-07-01 |
| KR20140091041A (ko) | 2014-07-18 |
| WO2013068464A1 (en) | 2013-05-16 |
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