JP2014513141A5 - - Google Patents

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Publication number
JP2014513141A5
JP2014513141A5 JP2014509519A JP2014509519A JP2014513141A5 JP 2014513141 A5 JP2014513141 A5 JP 2014513141A5 JP 2014509519 A JP2014509519 A JP 2014509519A JP 2014509519 A JP2014509519 A JP 2014509519A JP 2014513141 A5 JP2014513141 A5 JP 2014513141A5
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JP
Japan
Prior art keywords
composition
hydrogen
subject
compound
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2014509519A
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English (en)
Japanese (ja)
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JP2014513141A (ja
JP6122420B2 (ja
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Priority claimed from PCT/US2012/036841 external-priority patent/WO2012154695A2/en
Publication of JP2014513141A publication Critical patent/JP2014513141A/ja
Publication of JP2014513141A5 publication Critical patent/JP2014513141A5/ja
Application granted granted Critical
Publication of JP6122420B2 publication Critical patent/JP6122420B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2014509519A 2011-05-06 2012-05-07 多発性嚢胞疾患の治療 Active JP6122420B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161483630P 2011-05-06 2011-05-06
US61/483,630 2011-05-06
PCT/US2012/036841 WO2012154695A2 (en) 2011-05-06 2012-05-07 Treatment of polycystic disease

Publications (3)

Publication Number Publication Date
JP2014513141A JP2014513141A (ja) 2014-05-29
JP2014513141A5 true JP2014513141A5 (https=) 2015-09-10
JP6122420B2 JP6122420B2 (ja) 2017-04-26

Family

ID=47139933

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014509519A Active JP6122420B2 (ja) 2011-05-06 2012-05-07 多発性嚢胞疾患の治療

Country Status (6)

Country Link
US (1) US20140066462A1 (https=)
EP (1) EP2704723A4 (https=)
JP (1) JP6122420B2 (https=)
CN (1) CN103796655A (https=)
CA (1) CA2835197A1 (https=)
WO (1) WO2012154695A2 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1831225A2 (en) 2004-11-19 2007-09-12 The Regents of the University of California Anti-inflammatory pyrazolopyrimidines
US20110224223A1 (en) 2008-07-08 2011-09-15 The Regents Of The University Of California, A California Corporation MTOR Modulators and Uses Thereof
CN113620978A (zh) 2014-09-11 2021-11-09 加利福尼亚大学董事会 mTORC1抑制剂
US10118890B2 (en) 2014-10-10 2018-11-06 The Research Foundation For The State University Of New York Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration
AU2016342027B2 (en) * 2015-10-23 2021-05-13 Navitor Pharmaceuticals, Inc. Modulators of Sestrin-GATOR2 interaction and uses thereof
US10623555B2 (en) 2016-09-27 2020-04-14 Hartford Fire Insurance Company Controlling a graphical user interface for workflow
FR3075794A1 (fr) 2017-12-21 2019-06-28 Galderma Research & Development Nouveaux composes inhibiteurs de mtor
FR3075795A1 (fr) * 2017-12-21 2019-06-28 Galderma Research & Development Nouveaux composes inhibiteurs de mtor
MX2020011565A (es) 2018-05-01 2021-01-29 Revolution Medicines Inc Analogos de rapamicina ligados a c40, c28 y c-32 como inhibidores de mtor.
IL312291A (en) 2018-05-01 2024-06-01 Revolution Medicines Inc C-26-linked rapamycin analogs as MTOR inhibitors
CA3256390A1 (en) 2022-05-25 2023-11-30 Revolution Medicines, Inc. CANCER TREATMENT METHODS USING AN MTOR INHIBITOR

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0523659D0 (en) * 2005-11-21 2005-12-28 Novartis Ag Organic compounds
BRPI0915231A2 (pt) * 2008-07-08 2018-06-12 Intellikine Inc compostos inibidores de quinase e métodos de uso
US8476431B2 (en) * 2008-11-03 2013-07-02 Itellikine LLC Benzoxazole kinase inhibitors and methods of use
NZ598220A (en) * 2009-08-17 2014-02-28 Intellikine Llc Heterocyclic compounds and uses thereof
JP6047149B2 (ja) * 2011-05-04 2016-12-21 インテリカイン, エルエルシー 併用の医薬組成物およびその使用

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