JP2013542958A - アンサマイトシン誘導体を含む細胞傷害性剤 - Google Patents

アンサマイトシン誘導体を含む細胞傷害性剤 Download PDF

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JP2013542958A
JP2013542958A JP2013537819A JP2013537819A JP2013542958A JP 2013542958 A JP2013542958 A JP 2013542958A JP 2013537819 A JP2013537819 A JP 2013537819A JP 2013537819 A JP2013537819 A JP 2013537819A JP 2013542958 A JP2013542958 A JP 2013542958A
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チャリ，ラビ・ヴイ・ジェイ
ウィディソン，ウェイン・シー
ウィルヘルム，シャロン・ディー
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イミュノジェン・インコーポレーテッド
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JP2013537819A 2010-11-03 2011-11-03 アンサマイトシン誘導体を含む細胞傷害性剤 Pending JP2013542958A (ja)

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US40983110P 2010-11-03 2010-11-03
US61/409,831 2010-11-03
PCT/US2011/059131 WO2012061590A1 (en) 2010-11-03 2011-11-03 Cytotoxic agents comprising new ansamitocin derivatives

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JP2013542958A5 JP2013542958A5 (enExample) 2014-12-18

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US (2) US9090629B2 (enExample)
EP (1) EP2635301A4 (enExample)
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CN (2) CN103269712B (enExample)
AU (1) AU2011323316B2 (enExample)
BR (1) BR112013010853A2 (enExample)
CA (1) CA2816681A1 (enExample)
EA (1) EA201390642A1 (enExample)
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JP2018521123A (ja) * 2015-06-09 2018-08-02 エックスディーシーエクスプローラー （シャンハイ） カンパニー リミテッド 抗体薬物複合体、中間体、その製造方法、薬学的組成物及び応用
JP2019502746A (ja) * 2016-01-25 2019-01-31 レゲネロン ファーマシューティカルス，インコーポレーテッド メイタンシノイド誘導体、そのコンジュゲート、及び使用方法

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CN106267225B (zh) 2015-05-29 2020-03-06 上海新理念生物医药科技有限公司 三马来酰亚胺型连接子及其应用
CN106279352B (zh) 2015-05-29 2020-05-22 上海新理念生物医药科技有限公司 海兔毒素10的衍生物及其应用
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CN106729743B (zh) 2015-11-23 2021-09-21 四川科伦博泰生物医药股份有限公司 抗ErbB2抗体-药物偶联物及其组合物、制备方法和应用
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