JP2013530942A5 - - Google Patents

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Publication number
JP2013530942A5
JP2013530942A5 JP2013510192A JP2013510192A JP2013530942A5 JP 2013530942 A5 JP2013530942 A5 JP 2013530942A5 JP 2013510192 A JP2013510192 A JP 2013510192A JP 2013510192 A JP2013510192 A JP 2013510192A JP 2013530942 A5 JP2013530942 A5 JP 2013530942A5
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JP
Japan
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formula
compound
alkyl
methyl
analog
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Pending
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JP2013510192A
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English (en)
Japanese (ja)
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JP2013530942A (ja
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Priority claimed from PCT/US2011/035654 external-priority patent/WO2011140527A2/en
Publication of JP2013530942A publication Critical patent/JP2013530942A/ja
Publication of JP2013530942A5 publication Critical patent/JP2013530942A5/ja
Pending legal-status Critical Current

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JP2013510192A 2010-05-07 2011-05-06 移行型小胞体ａｔｐアーゼの阻害のための方法および組成物 Pending JP2013530942A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US33266710P 2010-05-07 2010-05-07
US61/332,667 2010-05-07
PCT/US2011/035654 WO2011140527A2 (en) 2010-05-07 2011-05-06 Methods and compositions for inhibition of the transitional endoplasmic reticulum atpase

Publications (2)

Publication Number Publication Date
JP2013530942A JP2013530942A (ja) 2013-08-01
JP2013530942A5 true JP2013530942A5 (https=) 2014-06-26

Family

ID=44904519

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013510192A Pending JP2013530942A (ja) 2010-05-07 2011-05-06 移行型小胞体ａｔｐアーゼの阻害のための方法および組成物

Country Status (8)

Country Link
US (1) US8865708B2 (https=)
EP (1) EP2566480A4 (https=)
JP (1) JP2013530942A (https=)
KR (1) KR20130128308A (https=)
CN (1) CN103068393A (https=)
AU (1) AU2011249859B2 (https=)
CA (1) CA2798698A1 (https=)
WO (1) WO2011140527A2 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2013530942A (ja) 2010-05-07 2013-08-01 カリフォルニア・インスティチュート・オブ・テクノロジー 移行型小胞体ａｔｐアーゼの阻害のための方法および組成物
US8906918B1 (en) * 2012-03-23 2014-12-09 University Of South Florida (A Florida Non-Profit Corporation) Compositions, methods of use, and methods of treatment
JP6109937B2 (ja) 2012-07-20 2017-04-05 クリーブ バイオサイエンシズ インコーポレイテッド ｐ９７複合体の阻害剤としての融合ピリミジン
EP2938610A2 (en) * 2012-12-28 2015-11-04 The U.S.A. as represented by the Secretary, Department of Health and Human Services Inhibitors of the usp1/uaf1 deubiquitinase complex and uses thereof
BR112015033042B1 (pt) 2013-07-16 2020-10-13 Basf Se composto de azina, processos para a preparação de composto de azina, composição agroquímica, processo para a preparação de composições agroquímicas, método para controlar vegetação e uso do composto de azina
DE102013110714A1 (de) * 2013-09-27 2015-04-02 Eberhard Karls Universität Tübingen Medizinische Fakultät Prophylaxe und Behandlung einer nicht auf einer Proteinfaltungsstörung beruhenden neurodegenerativen Erkrankung
WO2015057945A1 (en) * 2013-10-18 2015-04-23 Indiana University Research And Technology Corporation Hepatitis b viral assembly effectors
EP3080101A1 (en) 2013-12-10 2016-10-19 Cleave Biosciences, Inc. Monocyclic pyrimidine/pyridine compounds as inhibitors of p97 complex
JP6387111B2 (ja) * 2014-01-20 2018-09-05 クリーブ バイオサイエンシズ インコーポレイテッド ｐ９７複合体の阻害剤としての縮合ピリミジン
BR112016023178B1 (pt) 2014-04-11 2021-08-24 Basf Se Composto de diaminotriazina, composição agroquímica, método para o controle de vegetação indesejada e uso de um composto
JP6538077B2 (ja) * 2014-04-23 2019-07-03 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 除草剤としてのジアミノトリアジン化合物
EP3134391A1 (en) * 2014-04-23 2017-03-01 Basf Se Diaminotriazine compounds and their use as herbicides
CA2982811A1 (en) 2015-04-17 2016-10-20 Indiana University Research And Technology Corporation Hepatitis b viral assembly effectors
CN106518849B (zh) * 2016-10-27 2019-08-16 上海人类基因组研究中心 喹唑啉类化合物及其制备方法和用途
MX2021010323A (es) * 2019-03-01 2021-12-10 Revolution Medicines Inc Compuestos bicíclicos de heterociclilo y usos de este.
JPWO2024101336A1 (https=) * 2022-11-07 2024-05-16

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT64755A (en) * 1991-02-20 1994-02-28 Pfizer Process for the production of 2,4-diamino-quinazoline derivatives and of medical preparatives containing them
WO2003055866A1 (en) 2001-12-21 2003-07-10 Bayer Pharmaceuticals Corporation Quinazoline and quinoline derivative compounds as inhibitors of prolylpeptidase, inducers of apoptosis and cancer treatment agents
WO2004030672A1 (en) * 2002-10-02 2004-04-15 Merck Patent Gmbh Use of 4 amino-quinazolines as anti cancer agents
US20060025406A1 (en) * 2004-07-06 2006-02-02 Angion Biomedica Corporation Modulators of hepatocyte growth factor/c- Met activity
WO2006105056A2 (en) * 2005-03-28 2006-10-05 Fmc Corporation Insecticidal 2,4-diaminoquinazolines and related derivatives
WO2007041282A2 (en) * 2005-09-29 2007-04-12 The Johns Hopkins University Methods and compositions for treatment of cystic fibrosis
WO2008157500A1 (en) 2007-06-17 2008-12-24 Kalypsys, Inc. Aminoquinazoline cannabinoid receptor modulators for treatment of disease
CN101784276A (zh) * 2007-06-27 2010-07-21 传染性疾病研究院 化合物在用于制备抗结核药剂中的用途
US8637560B2 (en) 2007-07-18 2014-01-28 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Imidazolidinone compounds, methods to inhibit deubiquitination and methods of treatment
US9089572B2 (en) 2008-01-17 2015-07-28 California Institute Of Technology Inhibitors of p97
WO2010003908A1 (en) 2008-07-08 2010-01-14 Jakobsson, Andreas Screening assay for compounds targeting the p97 aaa-atpase complex in the ubiquitin proteasome system.
JP2013530942A (ja) 2010-05-07 2013-08-01 カリフォルニア・インスティチュート・オブ・テクノロジー 移行型小胞体ａｔｐアーゼの阻害のための方法および組成物

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