JP2013510159A5 - - Google Patents
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- Publication number
- JP2013510159A5 JP2013510159A5 JP2012537955A JP2012537955A JP2013510159A5 JP 2013510159 A5 JP2013510159 A5 JP 2013510159A5 JP 2012537955 A JP2012537955 A JP 2012537955A JP 2012537955 A JP2012537955 A JP 2012537955A JP 2013510159 A5 JP2013510159 A5 JP 2013510159A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- difluoro
- formula
- fluoropyridine
- pyridin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN2663CH2009 | 2009-11-03 | ||
| IN2663/CHE/2009 | 2009-11-03 | ||
| PCT/US2010/055176 WO2011056806A1 (en) | 2009-11-03 | 2010-11-02 | Process for the preparation of pyrazinone thrombin inhibitor and its intermediates |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013510159A JP2013510159A (ja) | 2013-03-21 |
| JP2013510159A5 true JP2013510159A5 (https=) | 2013-12-19 |
Family
ID=43926105
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012537955A Pending JP2013510159A (ja) | 2009-11-03 | 2010-11-02 | ピラジノントロンビン阻害剤およびその中間体の製造方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8541580B2 (https=) |
| EP (1) | EP2496087A4 (https=) |
| JP (1) | JP2013510159A (https=) |
| KR (1) | KR20120106727A (https=) |
| CN (1) | CN102711481A (https=) |
| AU (1) | AU2010315338A1 (https=) |
| CA (1) | CA2778922A1 (https=) |
| MX (1) | MX2012005165A (https=) |
| RU (1) | RU2012118499A (https=) |
| WO (1) | WO2011056806A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20140090663A (ko) | 2011-11-07 | 2014-07-17 | 디아크론 파마슈티칼스, 인코포레이티드 | 직접 트롬빈 억제제의 연장 방출성 제형 |
| MX392191B (es) | 2015-10-26 | 2025-03-21 | Bayer Cropscience Ag | Derivados de heterociclos biciclicos condensados como agentes de control de plagas. |
| JP7535532B2 (ja) | 2019-02-26 | 2024-08-16 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としての縮合二環式複素環式誘導体 |
| EP3931193A1 (en) | 2019-02-26 | 2022-01-05 | Bayer Aktiengesellschaft | Fused bicyclic heterocycle derivatives as pesticides |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6147078A (en) * | 1998-05-19 | 2000-11-14 | Merck & Co., Inc. | Pyrazinone thrombin inhibitors |
| UA58636C2 (uk) * | 1999-06-04 | 2003-08-15 | Мерк Енд Ко., Інк. | Піразинонові інгібітори тромбіну, фармацевтична композиція, спосіб інгібування утворення тромбів у крові, спосіб лікування станів, пов'язаних із тромбоутворенням |
| EP1341784A2 (en) * | 2000-12-06 | 2003-09-10 | Merck & Co., Inc. | Process for making a thrombin inhibitor |
| EP1422221A1 (en) * | 2002-11-20 | 2004-05-26 | Bayer CropScience SA | Novel process for the preparation of 2-aminomethylpyridine derivative |
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2010
- 2010-11-02 CA CA2778922A patent/CA2778922A1/en not_active Abandoned
- 2010-11-02 AU AU2010315338A patent/AU2010315338A1/en not_active Abandoned
- 2010-11-02 EP EP10828989.3A patent/EP2496087A4/en not_active Withdrawn
- 2010-11-02 CN CN2010800499062A patent/CN102711481A/zh active Pending
- 2010-11-02 MX MX2012005165A patent/MX2012005165A/es active IP Right Grant
- 2010-11-02 JP JP2012537955A patent/JP2013510159A/ja active Pending
- 2010-11-02 US US12/938,297 patent/US8541580B2/en not_active Expired - Fee Related
- 2010-11-02 WO PCT/US2010/055176 patent/WO2011056806A1/en not_active Ceased
- 2010-11-02 RU RU2012118499/04A patent/RU2012118499A/ru not_active Application Discontinuation
- 2010-11-02 KR KR1020127010789A patent/KR20120106727A/ko not_active Ceased