JP2013506679A - リゾホスファチジン酸受容体アンタゴニストとしての多環式化合物 - Google Patents

リゾホスファチジン酸受容体アンタゴニストとしての多環式化合物 Download PDF

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JP2013506679A
JP2013506679A JP2012532286A JP2012532286A JP2013506679A JP 2013506679 A JP2013506679 A JP 2013506679A JP 2012532286 A JP2012532286 A JP 2012532286A JP 2012532286 A JP2012532286 A JP 2012532286A JP 2013506679 A JP2013506679 A JP 2013506679A
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methyl
compound
biphenyl
isoxazol
phenyl
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ライアン・クラーク
ブライアン・アンドリュー・スターンズ
ルーシー・ザオ
トーマス・ジョン・シーダース
デボラ・ボルコッツ
ジニー・エム・アルーダ
デイビッド・ネイサン・ザラタン
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アミラ ファーマシューティカルス，インコーポレーテッド
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  • Urology & Nephrology (AREA)
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  • Diabetes (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Transplantation (AREA)
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  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
  • Dermatology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2012532286A 2009-10-01 2010-09-29 リゾホスファチジン酸受容体アンタゴニストとしての多環式化合物 Pending JP2013506679A (ja)

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Application Number Priority Date Filing Date Title
US24787709P 2009-10-01 2009-10-01
US61/247,877 2009-10-01
PCT/US2010/050786 WO2011041461A2 (en) 2009-10-01 2010-09-29 Polycyclic compounds as lysophosphatidic acid receptor antagonists

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JP2012532287A Ceased JP2013506680A (ja) 2009-10-01 2010-09-29 リゾホスファチジン酸受容体アンタゴニストとしての多環式化合物

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US (3) US8778983B2 (enExample)
EP (2) EP2483251B1 (enExample)
JP (2) JP2013506679A (enExample)
KR (1) KR20120097490A (enExample)
CN (2) CN102770415B (enExample)
AR (1) AR078495A1 (enExample)
AU (1) AU2010300594A1 (enExample)
BR (1) BR112012007102A2 (enExample)
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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2021506878A (ja) * 2017-12-19 2021-02-22 ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ Ｌｐａアンタゴニストとしてのシクロヘキシル酸イソキサゾールアジン
JP2021506863A (ja) * 2017-12-19 2021-02-22 ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ Ｌｐａアンタゴニストとしてのシクロヘキシル酸イソキサゾールアゾール

Families Citing this family (73)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010068775A2 (en) 2008-12-11 2010-06-17 Amira Pharmaceuticals, Inc. Alkyne antagonists of lysophosphatidic acid receptors
GB2466121B (en) 2008-12-15 2010-12-08 Amira Pharmaceuticals Inc Antagonists of lysophosphatidic acid receptors
GB2470833B (en) * 2009-06-03 2011-06-01 Amira Pharmaceuticals Inc Polycyclic antagonists of lysophosphatidic acid receptors
CN102574822A (zh) 2009-08-04 2012-07-11 阿米拉制药公司 作为溶血磷脂酸受体拮抗剂的化合物
GB2474748B (en) 2009-10-01 2011-10-12 Amira Pharmaceuticals Inc Polycyclic compounds as lysophosphatidic acid receptor antagonists
GB2474120B (en) * 2009-10-01 2011-12-21 Amira Pharmaceuticals Inc Compounds as Lysophosphatidic acid receptor antagonists
MX342405B (es) 2010-06-03 2016-09-28 Pharmacyclics Inc El uso de inhibidores de la tirosina quinasa de bruton (btk).
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