JP2013505252A - 三環式タンパク質キナーゼ調節剤 - Google Patents
三環式タンパク質キナーゼ調節剤 Download PDFInfo
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Classifications
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Enzymes And Modification Thereof (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
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| US24310409P | 2009-09-16 | 2009-09-16 | |
| US61/243,104 | 2009-09-16 | ||
| PCT/US2010/049113 WO2011035019A1 (en) | 2009-09-16 | 2010-09-16 | Novel tricyclic protein kinase modulators |
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| JP2013505252A true JP2013505252A (ja) | 2013-02-14 |
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| JP2012529900A Pending JP2013505252A (ja) | 2009-09-16 | 2010-09-16 | 三環式タンパク質キナーゼ調節剤 |
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| EP (1) | EP2477493A1 (enExample) |
| JP (1) | JP2013505252A (enExample) |
| KR (1) | KR20120104180A (enExample) |
| CN (1) | CN102647904A (enExample) |
| AU (1) | AU2010295619A1 (enExample) |
| BR (1) | BR112012005970A2 (enExample) |
| CA (1) | CA2774266A1 (enExample) |
| IL (1) | IL218631A0 (enExample) |
| IN (1) | IN2012DN03217A (enExample) |
| MX (1) | MX2012003322A (enExample) |
| SG (1) | SG179163A1 (enExample) |
| WO (1) | WO2011035019A1 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2017018060A1 (ja) * | 2015-07-27 | 2017-02-02 | 味の素株式会社 | システイン誘導体及びシステインスルホキシド誘導体の製造方法 |
| JP2023520883A (ja) * | 2020-03-30 | 2023-05-22 | センホア・バイオサイエンシーズ・インコーポレイテッド | Ｒｎａウイルス感染症、特にｃｏｖｉｄ－１９を処置するための抗ウイルス化合物および方法 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9342304B2 (en) | 2008-08-15 | 2016-05-17 | Apple Inc. | Processing vectors using wrapping increment and decrement instructions in the macroscalar architecture |
| US9335997B2 (en) | 2008-08-15 | 2016-05-10 | Apple Inc. | Processing vectors using a wrapping rotate previous instruction in the macroscalar architecture |
| US8583904B2 (en) | 2008-08-15 | 2013-11-12 | Apple Inc. | Processing vectors using wrapping negation instructions in the macroscalar architecture |
| US9335980B2 (en) | 2008-08-15 | 2016-05-10 | Apple Inc. | Processing vectors using wrapping propagate instructions in the macroscalar architecture |
| CA2856424A1 (en) * | 2011-11-29 | 2013-06-06 | Baylor College Of Medicine | A method to enhance cognition |
| US9389860B2 (en) | 2012-04-02 | 2016-07-12 | Apple Inc. | Prediction optimizations for Macroscalar vector partitioning loops |
| JP6280546B2 (ja) | 2012-06-26 | 2018-02-14 | デル マー ファーマシューティカルズ | ジアンヒドロガラクチトール、ジアセチルジアンヒドロガラクチトール、ジブロモズルシトール、又はこれらの類似体若しくは誘導体を用いた、遺伝子多型又はａｈｉ１の調節不全若しくは変異を有する患者におけるチロシンキナーゼインヒビター抵抗性悪性腫瘍を処置するための方法 |
| ES2649156T3 (es) | 2013-01-14 | 2018-01-10 | Incyte Holdings Corporation | Compuestos bicíclicos de carboxamida aromática útiles como inhibidores de quinasas Pim |
| PE20191245A1 (es) | 2013-01-15 | 2019-09-18 | Incyte Holdings Corp | Compuestos de tiazolcarboxamidas y piridinacarboxamida utiles como inhibidores de quinasa pim |
| US9817663B2 (en) | 2013-03-19 | 2017-11-14 | Apple Inc. | Enhanced Macroscalar predicate operations |
| US9348589B2 (en) | 2013-03-19 | 2016-05-24 | Apple Inc. | Enhanced predicate registers having predicates corresponding to element widths |
| KR20160061911A (ko) | 2013-04-08 | 2016-06-01 | 데니스 엠. 브라운 | 최적하 투여된 화학 화합물의 치료 효과 |
| EA201690458A1 (ru) | 2013-08-23 | 2016-07-29 | Инсайт Корпорейшн | Фуро- и тиенопиридинкарбоксамиды, используемые в качестве ингибиторов pim-киназы |
| US9822124B2 (en) | 2014-07-14 | 2017-11-21 | Incyte Corporation | Bicyclic heteroaromatic carboxamide compounds useful as Pim kinase inhibitors |
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- 2010-09-16 SG SG2012018453A patent/SG179163A1/en unknown
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017018060A1 (ja) * | 2015-07-27 | 2017-02-02 | 味の素株式会社 | システイン誘導体及びシステインスルホキシド誘導体の製造方法 |
| JPWO2017018060A1 (ja) * | 2015-07-27 | 2018-05-24 | 味の素株式会社 | システイン誘導体及びシステインスルホキシド誘導体の製造方法 |
| JP2023520883A (ja) * | 2020-03-30 | 2023-05-22 | センホア・バイオサイエンシーズ・インコーポレイテッド | Ｒｎａウイルス感染症、特にｃｏｖｉｄ－１９を処置するための抗ウイルス化合物および方法 |
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| MX2012003322A (es) | 2012-07-23 |
| WO2011035019A1 (en) | 2011-03-24 |
| EP2477493A1 (en) | 2012-07-25 |
| CN102647904A (zh) | 2012-08-22 |
| SG179163A1 (en) | 2012-05-30 |
| CA2774266A1 (en) | 2011-03-24 |
| BR112012005970A2 (pt) | 2015-09-08 |
| IN2012DN03217A (enExample) | 2015-10-23 |
| IL218631A0 (en) | 2012-05-31 |
| AU2010295619A1 (en) | 2012-05-10 |
| US20110071136A1 (en) | 2011-03-24 |
| KR20120104180A (ko) | 2012-09-20 |
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