JP2013501722A5 - - Google Patents

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Publication number
JP2013501722A5
JP2013501722A5 JP2012523949A JP2012523949A JP2013501722A5 JP 2013501722 A5 JP2013501722 A5 JP 2013501722A5 JP 2012523949 A JP2012523949 A JP 2012523949A JP 2012523949 A JP2012523949 A JP 2012523949A JP 2013501722 A5 JP2013501722 A5 JP 2013501722A5
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
compound
subject
formulated
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012523949A
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English (en)
Japanese (ja)
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JP2013501722A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2010/044570 external-priority patent/WO2011017534A2/en
Publication of JP2013501722A publication Critical patent/JP2013501722A/ja
Publication of JP2013501722A5 publication Critical patent/JP2013501722A5/ja
Pending legal-status Critical Current

Links

JP2012523949A 2009-08-07 2010-08-05 前立腺癌の処置 Pending JP2013501722A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US23225709P 2009-08-07 2009-08-07
US61/232,257 2009-08-07
US26126509P 2009-11-13 2009-11-13
US61/261,265 2009-11-13
PCT/US2010/044570 WO2011017534A2 (en) 2009-08-07 2010-08-05 Treatment of prostate cancer

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015221564A Division JP2016074687A (ja) 2009-08-07 2015-11-11 前立腺癌の処置

Publications (2)

Publication Number Publication Date
JP2013501722A JP2013501722A (ja) 2013-01-17
JP2013501722A5 true JP2013501722A5 (OSRAM) 2013-09-19

Family

ID=43535282

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2012523949A Pending JP2013501722A (ja) 2009-08-07 2010-08-05 前立腺癌の処置
JP2015221564A Pending JP2016074687A (ja) 2009-08-07 2015-11-11 前立腺癌の処置

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2015221564A Pending JP2016074687A (ja) 2009-08-07 2015-11-11 前立腺癌の処置

Country Status (8)

Country Link
US (5) US8791094B2 (OSRAM)
EP (1) EP2461814A4 (OSRAM)
JP (2) JP2013501722A (OSRAM)
KR (1) KR20120056267A (OSRAM)
AU (1) AU2010279398A1 (OSRAM)
BR (1) BR112012002797A2 (OSRAM)
CA (1) CA2770092A1 (OSRAM)
WO (1) WO2011017534A2 (OSRAM)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20100048524A1 (en) 2008-03-14 2010-02-25 Angela Brodie Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens;Synthesis In Vitro Biological Activities, Pharmacokinetics and Antitumor Activity
US8785423B2 (en) * 2008-04-14 2014-07-22 University Of Maryland, Baltimore Compositions and methods of inducing endoplasmic reticulum stress response for the treatment of cell proliferative diseases
CN102686600A (zh) 2009-02-05 2012-09-19 托凯药业股份有限公司 甾体cyp17抑制剂/抗雄激素物质的新型药物前体
WO2010149755A1 (en) 2009-06-26 2010-12-29 Novartis Ag 1, 3-disubstituted imidazolidin-2-one derivatives as inhibitors of cyp 17
AU2010279398A1 (en) 2009-08-07 2012-03-08 Tokai Pharmaceuticals, Inc. Treatment of prostate cancer
AU2012249421B9 (en) 2011-04-28 2015-10-22 Novartis Ag 17alpha-hydroxylase/C17,20-lyase inhibitors
CN103813794A (zh) * 2011-07-18 2014-05-21 拓凯制药公司 用于治疗前列腺癌的新型组合物及方法
US20130203615A1 (en) * 2011-08-05 2013-08-08 Gen-Probe Incorporated Antiandrogen therapy monitoring methods and compositions
WO2013071177A1 (en) * 2011-11-10 2013-05-16 Tokai Pharmaceuticals, Inc. Methods and compositions for inhibition of androgen receptor activity
CA2904170A1 (en) * 2013-03-14 2014-09-25 University Of Maryland, Baltimore Androgen receptor down-regulating agents and uses thereof
JP2016528252A (ja) 2013-08-12 2016-09-15 トーカイ ファーマシューティカルズ, インコーポレイテッド アンドロゲン標的治療を使用する新生物障害の処置のためのバイオマーカー
WO2015170336A1 (en) 2014-05-09 2015-11-12 Council Of Scientific & Industrial Research 16α-HETEROARYL PREGNENOLONE ACETATE AND A PROCESS FOR PREPARATION THEREOF
CN105732759A (zh) * 2015-01-29 2016-07-06 苏州晶云药物科技有限公司 (3β)-17-(1H-苯并咪唑-1-基)雄甾-5,16-二烯-3-醇的盐及其制备方法
CH714035B1 (it) * 2016-06-01 2021-02-15 Ind Chimica Srl Processo per la preparazione di 3Beta-idrossi-17-(1H-benzimidazol-1-il)androsta-5,16-diene.
ITUA20164043A1 (it) * 2016-06-01 2017-12-01 Ind Chimica Srl Processo per la preparazione di 3β-idrossi-17-(1H-benzimidazol-1-il)androsta-5,16-diene
CA3103679A1 (en) * 2018-06-14 2019-12-19 Astrazeneca Uk Limited Methods for treating and preventing symptoms of asthma with a corticosteroid pharmaceutical composition
CA3138176A1 (en) * 2019-04-27 2020-11-05 Health Research, Inc. Coumarin-modified androgens for the treatment of prostate cancer

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH621803A5 (OSRAM) * 1974-08-08 1981-02-27 Siphar Sa
US5604213A (en) * 1992-03-31 1997-02-18 British Technology Group Limited 17-substituted steroids useful in cancer treatment
CA2161531A1 (en) * 1993-04-30 1994-11-10 Donald C. Malins Dna profiles as an indicator of cellular redox potential and cancer risk
US5994335A (en) * 1997-10-17 1999-11-30 The University Of Maryland, Baltimore 17-azolyl steroids useful as androgen synthesis inhibitors
US20030054053A1 (en) * 2001-09-20 2003-03-20 Charles Young Methods and compositions for inhibiting the proliferation of prostate cancer cells
ATE513555T1 (de) 2003-07-29 2011-07-15 Dompe Spa Pharmazeutische kombination aus g-csf und plgf für blutstammzellen
JP4585201B2 (ja) * 2004-01-23 2010-11-24 丸善製薬株式会社 アンドロゲン受容体結合阻害剤、養毛剤、皮脂分泌抑制剤及び前立腺肥大抑制剤
NZ561571A (en) * 2005-03-02 2009-09-25 Univ Maryland Novel C-17-heteroaryl steroidal CYP17 inhibitors/antiandrogens: synthesis, in vitro biological activities, pharmacokinetics and antitumor activity
WO2008154382A1 (en) * 2007-06-06 2008-12-18 University Of Maryland, Baltimore Hdac inhibitors and hormone targeted drugs for the treatment of cancer
US20100048524A1 (en) * 2008-03-14 2010-02-25 Angela Brodie Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens;Synthesis In Vitro Biological Activities, Pharmacokinetics and Antitumor Activity
AU2010279398A1 (en) 2009-08-07 2012-03-08 Tokai Pharmaceuticals, Inc. Treatment of prostate cancer

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