JP2013501031A5 - - Google Patents
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- Publication number
- JP2013501031A5 JP2013501031A5 JP2012523342A JP2012523342A JP2013501031A5 JP 2013501031 A5 JP2013501031 A5 JP 2013501031A5 JP 2012523342 A JP2012523342 A JP 2012523342A JP 2012523342 A JP2012523342 A JP 2012523342A JP 2013501031 A5 JP2013501031 A5 JP 2013501031A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- oxo
- phenoxy
- pyridazin
- trifluoromethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0955504A FR2948939B1 (fr) | 2009-08-05 | 2009-08-05 | Derives de 2h pyridazin-3-ones, leur preparation et leur application en therapeutique humaine |
| FR0955504 | 2009-08-05 | ||
| PCT/EP2010/061426 WO2011015629A1 (en) | 2009-08-05 | 2010-08-05 | Derivatives of 2h pyridazin- 3 -ones, their preparation and their use as scd-1 inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013501031A JP2013501031A (ja) | 2013-01-10 |
| JP2013501031A5 true JP2013501031A5 (enExample) | 2013-09-12 |
| JP5901520B2 JP5901520B2 (ja) | 2016-04-13 |
Family
ID=41582079
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012523342A Expired - Fee Related JP5901520B2 (ja) | 2009-08-05 | 2010-08-05 | ２ｈピリダジン−３−オン誘導体、その製造、およびそれらのｓｃｄ−１インヒビターとしての使用 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8946225B2 (enExample) |
| EP (1) | EP2462121B1 (enExample) |
| JP (1) | JP5901520B2 (enExample) |
| AR (1) | AR077715A1 (enExample) |
| ES (1) | ES2536841T3 (enExample) |
| FR (1) | FR2948939B1 (enExample) |
| HU (1) | HUE025513T2 (enExample) |
| PL (1) | PL2462121T3 (enExample) |
| TW (1) | TW201109313A (enExample) |
| WO (1) | WO2011015629A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR086113A1 (es) | 2011-04-30 | 2013-11-20 | Abbott Lab | Isoxazolinas como agentes terapeuticos |
| JP6254087B2 (ja) * | 2011-10-15 | 2017-12-27 | ジェネンテック， インコーポレイテッド | 癌を治療するためのｓｃｄ１アンタゴニスト |
| US9238658B2 (en) | 2011-12-06 | 2016-01-19 | Janssen Pharmaceutica Nv | Substituted piperidinyl-carboxamide derivatives useful as SCD 1 inhibitors |
| WO2013085957A1 (en) * | 2011-12-06 | 2013-06-13 | Janssen Pharmaceutica Nv | Substituted piperidinyl-pyridazinyl derivatives useful as scd 1 inhibitors |
| SG10202008963QA (en) | 2015-09-18 | 2020-10-29 | Univ Miyazaki | Long-acting adrenomedullin derivative |
| CN110099898B (zh) | 2016-10-24 | 2023-07-25 | 优曼尼蒂治疗公司 | 化合物及其用途 |
| KR20190108118A (ko) | 2017-01-06 | 2019-09-23 | 유마니티 테라퓨틱스, 인크. | 신경계 장애의 치료를 위한 방법 |
| EP3700934A4 (en) | 2017-10-24 | 2021-10-27 | Yumanity Therapeutics, Inc. | COMPOUNDS AND USES OF THESE COMPOUNDS |
| BR112020019191A2 (pt) | 2018-03-23 | 2021-01-05 | Yumanity Therapeutics, Inc. | Compostos e seus usos |
| EP3914593A4 (en) * | 2019-01-24 | 2022-11-02 | Yumanity Therapeutics, Inc. | CONNECTIONS AND USES THEREOF |
| EA202192047A1 (ru) | 2019-11-13 | 2021-12-08 | Юманити Терапьютикс, Инк. | Соединения и их применение |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20060037410A (ko) * | 2003-07-30 | 2006-05-03 | 제논 파마슈티칼스 인크. | 피리다진 유도체 및 그의 치료제로서의 용도 |
| US7759348B2 (en) | 2003-07-30 | 2010-07-20 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives and their use as therapeutic agents |
| RU2339381C2 (ru) * | 2004-02-09 | 2008-11-27 | Ниссан Кемикал Индастриз, Лтд. | Ингибитор гиперплазии интимы сосудов |
| AU2006326815A1 (en) * | 2005-12-20 | 2007-06-28 | Merck Frosst Canada Ltd. | Heteroaromatic compounds as inhibitors of stearoyl-coenzyme A delta-9 desaturase |
| JP4984701B2 (ja) * | 2006-07-18 | 2012-07-25 | 富士ゼロックス株式会社 | Ｌｅｄプリントヘッドの製造方法 |
| JP4695565B2 (ja) * | 2006-08-21 | 2011-06-08 | 株式会社リコー | 画像形成装置 |
| EP2065369A4 (en) * | 2006-08-23 | 2011-12-28 | Astellas Pharma Inc | UREA CONNECTION OR SALT THEREOF |
| WO2008044767A1 (en) * | 2006-10-13 | 2008-04-17 | Takeda Pharmaceutical Company Limited | Aromatic amine derivative and use thereof |
| EP2173711B1 (en) | 2007-08-08 | 2010-11-17 | Graceway Pharmaceuticals, LLC | Phenoxy-pyrrolidine derivative and its use and compositions |
-
2009
- 2009-08-05 FR FR0955504A patent/FR2948939B1/fr not_active Expired - Fee Related
-
2010
- 2010-07-28 TW TW099124897A patent/TW201109313A/zh unknown
- 2010-08-05 PL PL10742811T patent/PL2462121T3/pl unknown
- 2010-08-05 WO PCT/EP2010/061426 patent/WO2011015629A1/en not_active Ceased
- 2010-08-05 ES ES10742811.2T patent/ES2536841T3/es active Active
- 2010-08-05 EP EP10742811.2A patent/EP2462121B1/en active Active
- 2010-08-05 US US13/388,884 patent/US8946225B2/en active Active
- 2010-08-05 JP JP2012523342A patent/JP5901520B2/ja not_active Expired - Fee Related
- 2010-08-05 HU HUE10742811A patent/HUE025513T2/hu unknown
- 2010-08-05 AR ARP100102874A patent/AR077715A1/es unknown
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