JP2013501031A5 - - Google Patents
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- Publication number
- JP2013501031A5 JP2013501031A5 JP2012523342A JP2012523342A JP2013501031A5 JP 2013501031 A5 JP2013501031 A5 JP 2013501031A5 JP 2012523342 A JP2012523342 A JP 2012523342A JP 2012523342 A JP2012523342 A JP 2012523342A JP 2013501031 A5 JP2013501031 A5 JP 2013501031A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- oxo
- phenoxy
- pyridazin
- trifluoromethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0955504A FR2948939B1 (fr) | 2009-08-05 | 2009-08-05 | Derives de 2h pyridazin-3-ones, leur preparation et leur application en therapeutique humaine |
| FR0955504 | 2009-08-05 | ||
| PCT/EP2010/061426 WO2011015629A1 (en) | 2009-08-05 | 2010-08-05 | Derivatives of 2h pyridazin- 3 -ones, their preparation and their use as scd-1 inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013501031A JP2013501031A (ja) | 2013-01-10 |
| JP2013501031A5 true JP2013501031A5 (cg-RX-API-DMAC7.html) | 2013-09-12 |
| JP5901520B2 JP5901520B2 (ja) | 2016-04-13 |
Family
ID=41582079
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012523342A Expired - Fee Related JP5901520B2 (ja) | 2009-08-05 | 2010-08-05 | ２ｈピリダジン−３−オン誘導体、その製造、およびそれらのｓｃｄ−１インヒビターとしての使用 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8946225B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP2462121B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP5901520B2 (cg-RX-API-DMAC7.html) |
| AR (1) | AR077715A1 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2536841T3 (cg-RX-API-DMAC7.html) |
| FR (1) | FR2948939B1 (cg-RX-API-DMAC7.html) |
| HU (1) | HUE025513T2 (cg-RX-API-DMAC7.html) |
| PL (1) | PL2462121T3 (cg-RX-API-DMAC7.html) |
| TW (1) | TW201109313A (cg-RX-API-DMAC7.html) |
| WO (1) | WO2011015629A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR086113A1 (es) | 2011-04-30 | 2013-11-20 | Abbott Lab | Isoxazolinas como agentes terapeuticos |
| CA2850836A1 (en) * | 2011-10-15 | 2013-04-18 | Genentech, Inc. | Methods of using scd1 antagonists |
| US9238658B2 (en) | 2011-12-06 | 2016-01-19 | Janssen Pharmaceutica Nv | Substituted piperidinyl-carboxamide derivatives useful as SCD 1 inhibitors |
| WO2013085957A1 (en) * | 2011-12-06 | 2013-06-13 | Janssen Pharmaceutica Nv | Substituted piperidinyl-pyridazinyl derivatives useful as scd 1 inhibitors |
| CN114805540A (zh) | 2015-09-18 | 2022-07-29 | 国立大学法人宫崎大学 | 长效肾上腺髓质素衍生物 |
| CN117777121A (zh) | 2016-10-24 | 2024-03-29 | 詹森药业有限公司 | 化合物及其用途 |
| MA47212A (fr) | 2017-01-06 | 2019-11-13 | Yumanity Therapeutics Inc | Méthodes de traitement de troubles neurologiques |
| EP3700934A4 (en) | 2017-10-24 | 2021-10-27 | Yumanity Therapeutics, Inc. | COMPOUNDS AND USES OF THESE COMPOUNDS |
| CN112312913B (zh) | 2018-03-23 | 2024-03-08 | 詹森药业有限公司 | 化合物和其用途 |
| SG11202108079RA (en) | 2019-01-24 | 2021-08-30 | Yumanity Therapeutics Inc | Compounds and uses thereof |
| EA202192047A1 (ru) * | 2019-11-13 | 2021-12-08 | Юманити Терапьютикс, Инк. | Соединения и их применение |
| CN117164524A (zh) * | 2022-09-06 | 2023-12-05 | 杭州师范大学 | 具有parp7/hdac双靶点抑制活性的哒嗪酮衍生物及其制备方法和应用 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7759348B2 (en) | 2003-07-30 | 2010-07-20 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives and their use as therapeutic agents |
| WO2005011653A2 (en) * | 2003-07-30 | 2005-02-10 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives and their use as therapeutic agents |
| BRPI0507518A8 (pt) * | 2004-02-09 | 2015-12-01 | Nissan Chemical Ind Ltd | Inibidor de hiperplasia vascular da íntima |
| WO2007071023A1 (en) * | 2005-12-20 | 2007-06-28 | Merck Frosst Canada Ltd. | Heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
| JP4984701B2 (ja) * | 2006-07-18 | 2012-07-25 | 富士ゼロックス株式会社 | Ｌｅｄプリントヘッドの製造方法 |
| JP4695565B2 (ja) * | 2006-08-21 | 2011-06-08 | 株式会社リコー | 画像形成装置 |
| EP2065369A4 (en) * | 2006-08-23 | 2011-12-28 | Astellas Pharma Inc | UREA CONNECTION OR SALT THEREOF |
| US20090325956A1 (en) * | 2006-10-13 | 2009-12-31 | Takahiko Taniguchi | Aromatic amine derivative and use thereof |
| DE602008003586D1 (de) | 2007-08-08 | 2010-12-30 | Graceway Pharmaceuticals Llc | Phenoxypyrrolidinderivat, seine verwendung sowie zusammensetzungen daraus |
-
2009
- 2009-08-05 FR FR0955504A patent/FR2948939B1/fr not_active Expired - Fee Related
-
2010
- 2010-07-28 TW TW099124897A patent/TW201109313A/zh unknown
- 2010-08-05 ES ES10742811.2T patent/ES2536841T3/es active Active
- 2010-08-05 PL PL10742811T patent/PL2462121T3/pl unknown
- 2010-08-05 US US13/388,884 patent/US8946225B2/en active Active
- 2010-08-05 EP EP10742811.2A patent/EP2462121B1/en active Active
- 2010-08-05 JP JP2012523342A patent/JP5901520B2/ja not_active Expired - Fee Related
- 2010-08-05 WO PCT/EP2010/061426 patent/WO2011015629A1/en not_active Ceased
- 2010-08-05 HU HUE10742811A patent/HUE025513T2/hu unknown
- 2010-08-05 AR ARP100102874A patent/AR077715A1/es unknown
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