JP2013500267A - ｍＧＬｕＲ４増強剤としての置換されたベンゾイミダゾールスルホンアミド類および置換されたインドールスルホンアミド類 - Google Patents

ｍＧＬｕＲ４増強剤としての置換されたベンゾイミダゾールスルホンアミド類および置換されたインドールスルホンアミド類 Download PDF

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JP2013500267A
JP2013500267A JP2012521845A JP2012521845A JP2013500267A JP 2013500267 A JP2013500267 A JP 2013500267A JP 2012521845 A JP2012521845 A JP 2012521845A JP 2012521845 A JP2012521845 A JP 2012521845A JP 2013500267 A JP2013500267 A JP 2013500267A
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optionally substituted
hydrogen
compound
mglur4
disorder
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JP2013500267A5 (https=
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ジェフリー コン，ピー．
ダブリュ． リンズリー，クレイグ
アール． ホプキンス，コーリー
デイヴィッド ウェイバー，チャールズ
エム． ニスウェンダー，コリーン
チュン，ユ−イン
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Vanderbilt University
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Vanderbilt University
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    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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JP2012521845A 2009-07-23 2010-07-23 ｍＧＬｕＲ４増強剤としての置換されたベンゾイミダゾールスルホンアミド類および置換されたインドールスルホンアミド類 Withdrawn JP2013500267A (ja)

Applications Claiming Priority (3)

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US22813709P 2009-07-23 2009-07-23
US61/228,137 2009-07-23
PCT/US2010/043110 WO2011011722A1 (en) 2009-07-23 2010-07-23 Substituted benzoimidazolesulfonamides and substituted indolesulfonamides as mglur4 potentiators

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JP2013500267A true JP2013500267A (ja) 2013-01-07
JP2013500267A5 JP2013500267A5 (https=) 2013-09-05

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US (1) US20120184556A1 (https=)
EP (1) EP2456310A4 (https=)
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AU (1) AU2010275477A1 (https=)
BR (1) BR112012001532A2 (https=)
CA (1) CA2768832A1 (https=)
SG (1) SG177740A1 (https=)
WO (1) WO2011011722A1 (https=)

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