JP2011520929A - 結晶性の2−((2s,3r,4e,6e,10e,12s)−13−(4−フルオロフェノキシ)−2,3,12−トリヒドロキシトリデカ−4,6,10−トリエン−8−イニルオキシ)酢酸の無水及び水和物形態 - Google Patents

結晶性の2−((2s,3r,4e,6e,10e,12s)−13−(4−フルオロフェノキシ)−2,3,12−トリヒドロキシトリデカ−4,6,10−トリエン−8−イニルオキシ)酢酸の無水及び水和物形態 Download PDF

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JP2011520929A
JP2011520929A JP2011509858A JP2011509858A JP2011520929A JP 2011520929 A JP2011520929 A JP 2011520929A JP 2011509858 A JP2011509858 A JP 2011509858A JP 2011509858 A JP2011509858 A JP 2011509858A JP 2011520929 A JP2011520929 A JP 2011520929A
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disease
crystalline
inflammatory
acid
fluorophenoxy
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Japanese (ja)
Inventor
バルテル,クラウス
グロスバッハ,ダンヤ
ギルフォード,ウィリアム
ザンダー,ミヒャエル
ビンター,ガブリーレ
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Bayer Pharma AG
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Bayer Schering Pharma AG
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    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/58Unsaturated compounds containing ether groups, groups, groups, or groups
    • C07C59/64Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings
    • C07C59/66Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings
    • C07C59/68Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings the oxygen atom of the ether group being bound to a non-condensed six-membered aromatic ring
    • C07C59/70Ethers of hydroxy-acetic acid, e.g. substitutes on the ring
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JP2011509858A 2008-05-22 2008-05-22 結晶性の2−((2s,3r,4e,6e,10e,12s)−13−(4−フルオロフェノキシ)−2,3,12−トリヒドロキシトリデカ−4,6,10−トリエン−8−イニルオキシ)酢酸の無水及び水和物形態 Withdrawn JP2011520929A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/EP2008/004100 WO2009140984A1 (en) 2008-05-22 2008-05-22 Anhydrous and hydrate forms of crystalline 2- ( (2s, 3r, 4e, 6e, 1oe, 12s) -13- (4-fluorophenoxy) -2,3, 12- (trihydroxytrideca-4, 6, 10-trien-8-ynyl) oxy) acetic acid

Publications (1)

Publication Number Publication Date
JP2011520929A true JP2011520929A (ja) 2011-07-21

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JP2011509858A Withdrawn JP2011520929A (ja) 2008-05-22 2008-05-22 結晶性の2−((2s,3r,4e,6e,10e,12s)−13−(4−フルオロフェノキシ)−2,3,12−トリヒドロキシトリデカ−4,6,10−トリエン−8−イニルオキシ)酢酸の無水及び水和物形態

Country Status (6)

Country Link
EP (1) EP2288414A1 (ko)
JP (1) JP2011520929A (ko)
KR (1) KR20110010755A (ko)
CN (1) CN102036714A (ko)
CA (1) CA2723769A1 (ko)
WO (1) WO2009140984A1 (ko)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6831186B2 (en) * 2001-11-06 2004-12-14 Schering Aktiengesellschft Lipoxin A4 analogs
TW200816991A (en) * 2006-08-23 2008-04-16 Bayer Schering Pharma Ag Treatment and prevention of intestinal fibrosis

Also Published As

Publication number Publication date
KR20110010755A (ko) 2011-02-07
CN102036714A (zh) 2011-04-27
WO2009140984A1 (en) 2009-11-26
EP2288414A1 (en) 2011-03-02
CA2723769A1 (en) 2009-11-26

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