JP2011513501A - 局所使用のためのビタミンｋ類似体製剤 - Google Patents
局所使用のためのビタミンｋ類似体製剤 Download PDFInfo
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- JP2011513501A JP2011513501A JP2010550880A JP2010550880A JP2011513501A JP 2011513501 A JP2011513501 A JP 2011513501A JP 2010550880 A JP2010550880 A JP 2010550880A JP 2010550880 A JP2010550880 A JP 2010550880A JP 2011513501 A JP2011513501 A JP 2011513501A
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- pharmaceutical formulation
- menadione
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- vitamin
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- DXGLGDHPHMLXJC-UHFFFAOYSA-N oxybenzone Chemical compound OC1=CC(OC)=CC=C1C(=O)C1=CC=CC=C1 DXGLGDHPHMLXJC-UHFFFAOYSA-N 0.000 description 1
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- 125000002467 phosphate group Chemical group [H]OP(=O)(O[H])O[*] 0.000 description 1
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- LFSXCDWNBUNEEM-UHFFFAOYSA-N phthalazine Chemical compound C1=NN=CC2=CC=CC=C21 LFSXCDWNBUNEEM-UHFFFAOYSA-N 0.000 description 1
- MBWXNTAXLNYFJB-LKUDQCMESA-N phylloquinone Chemical compound C1=CC=C2C(=O)C(C/C=C(C)/CCCC(C)CCCC(C)CCCC(C)C)=C(C)C(=O)C2=C1 MBWXNTAXLNYFJB-LKUDQCMESA-N 0.000 description 1
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- DQKXQSGTHWVTAD-UHFFFAOYSA-N pramocaine Chemical compound C1=CC(OCCCC)=CC=C1OCCCN1CCOCC1 DQKXQSGTHWVTAD-UHFFFAOYSA-N 0.000 description 1
- 230000002028 premature Effects 0.000 description 1
- 238000002360 preparation method Methods 0.000 description 1
- 239000011253 protective coating Substances 0.000 description 1
- 208000029561 pustule Diseases 0.000 description 1
- BWESROVQGZSBRX-UHFFFAOYSA-N pyrido[3,2-d]pyrimidine Chemical compound C1=NC=NC2=CC=CN=C21 BWESROVQGZSBRX-UHFFFAOYSA-N 0.000 description 1
- JOZPEVMCAKXSEY-UHFFFAOYSA-N pyrimido[5,4-d]pyrimidine Chemical compound N1=CN=CC2=NC=NC=C21 JOZPEVMCAKXSEY-UHFFFAOYSA-N 0.000 description 1
- 238000011002 quantification Methods 0.000 description 1
- JWVCLYRUEFBMGU-UHFFFAOYSA-N quinazoline Chemical compound N1=CN=CC2=CC=CC=C21 JWVCLYRUEFBMGU-UHFFFAOYSA-N 0.000 description 1
- LISFMEBWQUVKPJ-UHFFFAOYSA-N quinolin-2-ol Chemical compound C1=CC=C2NC(=O)C=CC2=C1 LISFMEBWQUVKPJ-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/12—Ketones
- A61K31/122—Ketones having the oxygen directly attached to a ring, e.g. quinones, vitamin K1, anthralin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| US20493909P | 2009-01-13 | 2009-01-13 | |
| PCT/US2009/037041 WO2009114745A1 (en) | 2008-03-13 | 2009-03-13 | Formulations of vitamin k analogs for topical use |
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| JP2014218037A Division JP2015042658A (ja) | 2008-03-13 | 2014-10-27 | 局所使用のためのビタミンｋ類似体製剤 |
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| JP2014218037A Pending JP2015042658A (ja) | 2008-03-13 | 2014-10-27 | 局所使用のためのビタミンｋ類似体製剤 |
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| US (2) | US8815953B2 (enExample) |
| EP (1) | EP2265255A1 (enExample) |
| JP (2) | JP2011513501A (enExample) |
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| AU (1) | AU2009223158B2 (enExample) |
| CA (1) | CA2718262A1 (enExample) |
| WO (1) | WO2009114745A1 (enExample) |
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| US20100010100A1 (en) * | 2008-07-09 | 2010-01-14 | Hinman Andrew W | Dermatological compositions with anti-aging and skin even-toning properties |
| WO2010014361A1 (en) * | 2008-07-30 | 2010-02-04 | Edison Pharmaceuticals, Inc. | Naphthoquinone compositions with anti-aging, anti- inflammatory and skin even-toning properties |
| CA2773957C (en) * | 2009-09-14 | 2018-01-09 | Nestec S.A. | Nutritional compositions for modulating inflammation including exogenous vitamin k2 |
| ITPD20100090A1 (it) * | 2010-03-22 | 2011-09-23 | Sanitas Farmaceutici S R L | Formulazione topica per il trattamento di eruzioni cutanee, in particolare conseguenti a trattamenti con farmaci anti egfr |
| EP2601168A4 (en) * | 2010-08-06 | 2013-12-04 | Ampere Life Sciences Inc | TREATMENT OF MITOCHONDRIAL DISEASES BY VITAMIN K |
| BR112012027864A2 (pt) | 2011-02-14 | 2016-08-09 | J Oil Mills Inc | agente de elevação do teor de colágeno na pele |
| US9421297B2 (en) | 2014-04-02 | 2016-08-23 | Adhezion Biomedical, Llc | Sterilized compositions of cyanoacrylate monomers and naphthoquinone 2,3-oxides |
| WO2019072877A1 (en) | 2017-10-10 | 2019-04-18 | Capsugel Belgium Nv | GETTING MULTIPARTICULAR COMPOSITIONS |
| JP2021506958A (ja) | 2017-12-13 | 2021-02-22 | オンクォリティ ファーマシューティカルズ チャイナ エルティーディーＯｎｑｕａｌｉｔｙ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｃｈｉｎａ Ｌｔｄ． | Ｅｇｆｒ阻害に関連する疾患を予防又は治療する方法 |
| WO2019201195A1 (zh) | 2018-04-16 | 2019-10-24 | 上海岸阔医药科技有限公司 | 预防或治疗肿瘤疗法副作用的方法 |
| WO2020067663A1 (ko) * | 2018-09-28 | 2020-04-02 | 주식회사 엘지생활건강 | 피부 턴오버 촉진 및 멜라닌 배출 촉진용 조성물 |
| WO2020214855A1 (en) * | 2019-04-17 | 2020-10-22 | Azora Therapeutics, Inc. | Topical compositions and methods for treating inflammatory skin diseases |
| WO2023119230A1 (en) | 2021-12-22 | 2023-06-29 | L'oreal | Coagulation pathway and nicotinamide-adenine dinucleotide pathway modulating compositions and methods of their use |
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| US20050092969A1 (en) * | 2003-10-08 | 2005-05-05 | Kaneka Corporation | Method of stabilizing compound having quinone skeleton and stabilized composition |
| KR20060002239A (ko) * | 2004-07-01 | 2006-01-09 | 삼성전자주식회사 | 레이저 출력 제어장치 |
| WO2006029893A2 (en) | 2004-09-17 | 2006-03-23 | Oystershell Nv | Composition for inhibiting or preventing the formation of a biofilm |
| US20090010887A1 (en) | 2004-10-06 | 2009-01-08 | Ben-Sasson Shmuel A | Method and composition for enhancing anti-angiogenic therapy |
| WO2006107827A1 (en) | 2005-04-05 | 2006-10-12 | Creighton University | Skin bonding process |
| US20060275504A1 (en) * | 2005-06-07 | 2006-12-07 | Tty Biopharm Company Limited | Methods and compositions for augmenting cancer chemotherapeutic agents |
| US7252816B1 (en) * | 2006-03-29 | 2007-08-07 | Dow Pharmaceutical Sciences | Topical acne vulgairs medication with a sunscreen |
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2009
- 2009-03-12 US US12/381,467 patent/US8815953B2/en active Active
- 2009-03-13 CA CA2718262A patent/CA2718262A1/en not_active Abandoned
- 2009-03-13 AU AU2009223158A patent/AU2009223158B2/en not_active Ceased
- 2009-03-13 KR KR1020107022900A patent/KR20110004382A/ko not_active Ceased
- 2009-03-13 WO PCT/US2009/037041 patent/WO2009114745A1/en not_active Ceased
- 2009-03-13 JP JP2010550880A patent/JP2011513501A/ja active Pending
- 2009-03-13 EP EP09718881A patent/EP2265255A1/en not_active Withdrawn
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2014
- 2014-07-21 US US14/336,876 patent/US20140336268A1/en not_active Abandoned
- 2014-10-27 JP JP2014218037A patent/JP2015042658A/ja active Pending
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| JPH02292228A (ja) * | 1989-04-14 | 1990-12-03 | Minnesota Mining & Mfg Co <3M> | 固体ゲル外用薬剤送達システム |
| JP2003226639A (ja) * | 2002-01-31 | 2003-08-12 | Hisamitsu Pharmaceut Co Inc | 神経成長因子活性増強剤としてのビタミンｋ類を含む医薬組成物およびその使用 |
| US20030170187A1 (en) * | 2002-03-01 | 2003-09-11 | Alfred Marchal | Skin treatments containing nano-sized vitamin K |
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| US20070025950A1 (en) * | 2005-07-28 | 2007-02-01 | Elson Melvin L | Composition and method for treating cellulite |
Also Published As
| Publication number | Publication date |
|---|---|
| US20140336268A1 (en) | 2014-11-13 |
| AU2009223158A1 (en) | 2009-09-17 |
| US8815953B2 (en) | 2014-08-26 |
| WO2009114745A1 (en) | 2009-09-17 |
| CA2718262A1 (en) | 2009-09-17 |
| JP2015042658A (ja) | 2015-03-05 |
| KR20110004382A (ko) | 2011-01-13 |
| AU2009223158B2 (en) | 2014-08-28 |
| EP2265255A1 (en) | 2010-12-29 |
| US20090234022A1 (en) | 2009-09-17 |
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