JP2011510013A5 - - Google Patents
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- Publication number
- JP2011510013A5 JP2011510013A5 JP2010543227A JP2010543227A JP2011510013A5 JP 2011510013 A5 JP2011510013 A5 JP 2011510013A5 JP 2010543227 A JP2010543227 A JP 2010543227A JP 2010543227 A JP2010543227 A JP 2010543227A JP 2011510013 A5 JP2011510013 A5 JP 2011510013A5
- Authority
- JP
- Japan
- Prior art keywords
- independently
- compound
- alpha
- following structure
- use according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- RNTRQUCAVQIHDO-UHFFFAOYSA-N Fc1cccc(C(Cc2ccncc2)/N=C2\SCCN2)c1 Chemical compound Fc1cccc(C(Cc2ccncc2)/N=C2\SCCN2)c1 RNTRQUCAVQIHDO-UHFFFAOYSA-N 0.000 description 2
- 0 C(*c1ccccc1)c1ccncc1 Chemical compound C(*c1ccccc1)c1ccncc1 0.000 description 1
- JOLDLDJZLZMJIK-UHFFFAOYSA-N C(C(c1ccccc1)/N=C1\SCCN1)c1ccncc1 Chemical compound C(C(c1ccccc1)/N=C1\SCCN1)c1ccncc1 JOLDLDJZLZMJIK-UHFFFAOYSA-N 0.000 description 1
- KPLMTYILBIVJMN-UHFFFAOYSA-N C(C(c1ccccc1)/N=C1\SCCN1)c1nccnc1 Chemical compound C(C(c1ccccc1)/N=C1\SCCN1)c1nccnc1 KPLMTYILBIVJMN-UHFFFAOYSA-N 0.000 description 1
- JOLDLDJZLZMJIK-OAHLLOKOSA-N C([C@H](c1ccccc1)/N=C1\SCCN1)c1ccncc1 Chemical compound C([C@H](c1ccccc1)/N=C1\SCCN1)c1ccncc1 JOLDLDJZLZMJIK-OAHLLOKOSA-N 0.000 description 1
- LGOFDFRKSKNQTC-UHFFFAOYSA-N CC(CC1(C)C(Cc2ncccc2)/N=C2\SCCN2)C=CC1Cl Chemical compound CC(CC1(C)C(Cc2ncccc2)/N=C2\SCCN2)C=CC1Cl LGOFDFRKSKNQTC-UHFFFAOYSA-N 0.000 description 1
- JJAKPNMFQFKELV-UHFFFAOYSA-N COc1c(C(Cc2ccccn2)/N=C2\SCCN2)cccc1 Chemical compound COc1c(C(Cc2ccccn2)/N=C2\SCCN2)cccc1 JJAKPNMFQFKELV-UHFFFAOYSA-N 0.000 description 1
- XQHDTRQXMTUGAE-UHFFFAOYSA-N COc1c(C(Cc2cccnc2)/N=C2\SCCN2)cccc1 Chemical compound COc1c(C(Cc2cccnc2)/N=C2\SCCN2)cccc1 XQHDTRQXMTUGAE-UHFFFAOYSA-N 0.000 description 1
- YPCGRDLGSQQSIX-UHFFFAOYSA-N COc1ccccc1C(Cc1ccncc1)/N=C1\SCCN1 Chemical compound COc1ccccc1C(Cc1ccncc1)/N=C1\SCCN1 YPCGRDLGSQQSIX-UHFFFAOYSA-N 0.000 description 1
- ZKBSZRHCWYVJJM-UHFFFAOYSA-N Cc(cc1C(Cc2ccncc2)/N=C2\SCCN2)ccc1Cl Chemical compound Cc(cc1C(Cc2ccncc2)/N=C2\SCCN2)ccc1Cl ZKBSZRHCWYVJJM-UHFFFAOYSA-N 0.000 description 1
- FOBQLJDFOPROIT-UHFFFAOYSA-N Cc1c(C)c(C(Cc2cccnc2)/N=C2\SCCN2)ccc1 Chemical compound Cc1c(C)c(C(Cc2cccnc2)/N=C2\SCCN2)ccc1 FOBQLJDFOPROIT-UHFFFAOYSA-N 0.000 description 1
- ZNIFGCJXFIJIJX-UHFFFAOYSA-N Cc1cccc(C(Cc2ccncc2)/N=C2\SCCN2)c1C Chemical compound Cc1cccc(C(Cc2ccncc2)/N=C2\SCCN2)c1C ZNIFGCJXFIJIJX-UHFFFAOYSA-N 0.000 description 1
- WCJUGOFLLFFBQV-UHFFFAOYSA-N FC(c1ccc(C(Cc2nccnc2)/N=C2\SCCN2)cc1)(F)F Chemical compound FC(c1ccc(C(Cc2nccnc2)/N=C2\SCCN2)cc1)(F)F WCJUGOFLLFFBQV-UHFFFAOYSA-N 0.000 description 1
- FGSWUBATMWRUKR-UHFFFAOYSA-N [N-2]=C1SCCN1 Chemical compound [N-2]=C1SCCN1 FGSWUBATMWRUKR-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2214208P | 2008-01-18 | 2008-01-18 | |
| US12/353,406 US8809379B2 (en) | 2008-01-18 | 2009-01-14 | Selective subtype alpha 2 adrenergic agents and methods for use thereof |
| PCT/US2009/031077 WO2009091874A1 (en) | 2008-01-18 | 2009-01-15 | Selective subtype alpha 2 adrenergic agents and methods for use thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2011510013A JP2011510013A (ja) | 2011-03-31 |
| JP2011510013A5 true JP2011510013A5 (https=) | 2012-03-01 |
Family
ID=40383664
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010543227A Withdrawn JP2011510013A (ja) | 2008-01-18 | 2009-01-15 | 選択的サブタイプアルファ２アドレナリンアゴニスト及びその使用方法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US8809379B2 (https=) |
| EP (1) | EP2249834B1 (https=) |
| JP (1) | JP2011510013A (https=) |
| AU (1) | AU2009206137B2 (https=) |
| BR (1) | BRPI0906928A8 (https=) |
| CA (1) | CA2712269A1 (https=) |
| WO (1) | WO2009091874A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2242753B1 (en) * | 2008-01-18 | 2015-04-08 | Allergan, Inc. | Oxazolidine and thiazolidine selective subtype alpha 2 adrenergic agents and methods for use thereof |
| HUE038366T2 (hu) * | 2010-08-16 | 2018-10-29 | Allergan Inc | Módszer szabályozó T-sejtek alfa-2B adrenerg receptor agonistákkal való aktiválásához |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5212176A (en) | 1990-06-29 | 1993-05-18 | Abbott Laboratories | R(+)-terazosin |
| KR100639473B1 (ko) * | 2005-06-16 | 2006-10-27 | 주식회사 삼화양행 | 압전체의 온도 변화에 따른 주파수 특성을 비선형적으로구하는 방법 |
| CN101346374A (zh) | 2005-12-22 | 2009-01-14 | 巴斯夫欧洲公司 | 农业组合物 |
| US7709507B2 (en) | 2006-05-17 | 2010-05-04 | Allergan, Inc. | Therapeutic fluoroethyl ureas |
| WO2008123821A1 (en) | 2007-03-01 | 2008-10-16 | Albireo Ab | 4, 5-dihydro-lh-imidazol-2-amine derivatives for use in the treatment of respiratory, cardiovascular, neurological or gastrointestinal disorders |
| WO2008115141A1 (en) | 2007-03-19 | 2008-09-25 | Albireo Ab | 4, 5-dihydro-1,3-thiazol-2-amine derivatives and their use in the treatment of respiratory, cardiovascular, neurological or gastrointestinal disorders |
| EP2242753B1 (en) * | 2008-01-18 | 2015-04-08 | Allergan, Inc. | Oxazolidine and thiazolidine selective subtype alpha 2 adrenergic agents and methods for use thereof |
| JP5480819B2 (ja) * | 2008-01-18 | 2014-04-23 | アラーガン インコーポレイテッド | 選択的サブタイプアルファ２アドレナリンアゴニスト及びその使用方法 |
-
2009
- 2009-01-14 US US12/353,406 patent/US8809379B2/en not_active Expired - Fee Related
- 2009-01-15 WO PCT/US2009/031077 patent/WO2009091874A1/en not_active Ceased
- 2009-01-15 JP JP2010543227A patent/JP2011510013A/ja not_active Withdrawn
- 2009-01-15 AU AU2009206137A patent/AU2009206137B2/en not_active Ceased
- 2009-01-15 EP EP20090702616 patent/EP2249834B1/en not_active Not-in-force
- 2009-01-15 BR BRPI0906928A patent/BRPI0906928A8/pt not_active IP Right Cessation
- 2009-01-15 CA CA2712269A patent/CA2712269A1/en not_active Abandoned
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