AU2009206137B2 - Selective subtype alpha 2 adrenergic agents and methods for use thereof - Google Patents

Selective subtype alpha 2 adrenergic agents and methods for use thereof Download PDF

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Publication number
AU2009206137B2
AU2009206137B2 AU2009206137A AU2009206137A AU2009206137B2 AU 2009206137 B2 AU2009206137 B2 AU 2009206137B2 AU 2009206137 A AU2009206137 A AU 2009206137A AU 2009206137 A AU2009206137 A AU 2009206137A AU 2009206137 B2 AU2009206137 B2 AU 2009206137B2
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compound
alpha
independently
pain
lower alkyl
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AU2009206137A1 (en
Inventor
Smita S. Bhat
Ken Chow
Wenkui K. Fang
Todd M. Heidelbaugh
Ling Li
Phong X. Nguyen
Santosh C. Sinha
Janet A. Takeuchi
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Allergan Inc
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Allergan Inc
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
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  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
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AU2009206137A 2008-01-18 2009-01-15 Selective subtype alpha 2 adrenergic agents and methods for use thereof Ceased AU2009206137B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US2214208P 2008-01-18 2008-01-18
US61/022,142 2008-01-18
US12/353,406 2009-01-14
US12/353,406 US8809379B2 (en) 2008-01-18 2009-01-14 Selective subtype alpha 2 adrenergic agents and methods for use thereof
PCT/US2009/031077 WO2009091874A1 (en) 2008-01-18 2009-01-15 Selective subtype alpha 2 adrenergic agents and methods for use thereof

Publications (2)

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AU2009206137A1 AU2009206137A1 (en) 2009-07-23
AU2009206137B2 true AU2009206137B2 (en) 2014-03-27

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AU2009206137A Ceased AU2009206137B2 (en) 2008-01-18 2009-01-15 Selective subtype alpha 2 adrenergic agents and methods for use thereof

Country Status (7)

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US (1) US8809379B2 (https=)
EP (1) EP2249834B1 (https=)
JP (1) JP2011510013A (https=)
AU (1) AU2009206137B2 (https=)
BR (1) BRPI0906928A8 (https=)
CA (1) CA2712269A1 (https=)
WO (1) WO2009091874A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2242753B1 (en) * 2008-01-18 2015-04-08 Allergan, Inc. Oxazolidine and thiazolidine selective subtype alpha 2 adrenergic agents and methods for use thereof
HUE038366T2 (hu) * 2010-08-16 2018-10-29 Allergan Inc Módszer szabályozó T-sejtek alfa-2B adrenerg receptor agonistákkal való aktiválásához

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007013702A1 (en) * 2005-06-16 2007-02-01 Samhwa Yang Heng Co., Ltd. A method for calculating frequency characteristics of piezoelectric material non-linearly according to temperature rising

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5212176A (en) 1990-06-29 1993-05-18 Abbott Laboratories R(+)-terazosin
CN101346374A (zh) 2005-12-22 2009-01-14 巴斯夫欧洲公司 农业组合物
US7709507B2 (en) 2006-05-17 2010-05-04 Allergan, Inc. Therapeutic fluoroethyl ureas
WO2008123821A1 (en) 2007-03-01 2008-10-16 Albireo Ab 4, 5-dihydro-lh-imidazol-2-amine derivatives for use in the treatment of respiratory, cardiovascular, neurological or gastrointestinal disorders
WO2008115141A1 (en) 2007-03-19 2008-09-25 Albireo Ab 4, 5-dihydro-1,3-thiazol-2-amine derivatives and their use in the treatment of respiratory, cardiovascular, neurological or gastrointestinal disorders
EP2242753B1 (en) * 2008-01-18 2015-04-08 Allergan, Inc. Oxazolidine and thiazolidine selective subtype alpha 2 adrenergic agents and methods for use thereof
JP5480819B2 (ja) * 2008-01-18 2014-04-23 アラーガン インコーポレイテッド 選択的サブタイプアルファ2アドレナリンアゴニスト及びその使用方法

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007013702A1 (en) * 2005-06-16 2007-02-01 Samhwa Yang Heng Co., Ltd. A method for calculating frequency characteristics of piezoelectric material non-linearly according to temperature rising

Also Published As

Publication number Publication date
CA2712269A1 (en) 2009-07-23
AU2009206137A1 (en) 2009-07-23
BRPI0906928A8 (pt) 2018-12-11
US8809379B2 (en) 2014-08-19
US20090197898A1 (en) 2009-08-06
EP2249834A1 (en) 2010-11-17
WO2009091874A1 (en) 2009-07-23
BRPI0906928A2 (pt) 2017-06-13
EP2249834B1 (en) 2015-05-13
JP2011510013A (ja) 2011-03-31

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