JP2011503081A - グルココルチコイド受容体、ＡＰ−１および／またはＮＦ−κＢ活性の調節剤として有用な非ステロイド性化合物、並びにその使用 - Google Patents

グルココルチコイド受容体、ＡＰ−１および／またはＮＦ−κＢ活性の調節剤として有用な非ステロイド性化合物、並びにその使用 Download PDF

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JP2011503081A
JP2011503081A JP2010533163A JP2010533163A JP2011503081A JP 2011503081 A JP2011503081 A JP 2011503081A JP 2010533163 A JP2010533163 A JP 2010533163A JP 2010533163 A JP2010533163 A JP 2010533163A JP 2011503081 A JP2011503081 A JP 2011503081A
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alkyl
disease
hydrogen
inhibitor
substituted
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JP2011503081A5 (enExample
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ティ・ジー・ムラリ・ダー
ハイ−ユン・シャオ
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Bristol Myers Squibb Co
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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JP2010533163A 2007-11-01 2008-10-30 グルココルチコイド受容体、ＡＰ−１および／またはＮＦ−κＢ活性の調節剤として有用な非ステロイド性化合物、並びにその使用 Withdrawn JP2011503081A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US98451507P 2007-11-01 2007-11-01
PCT/US2008/081702 WO2009058944A2 (en) 2007-11-01 2008-10-30 Nonsteroidal compounds useful as modulators of glucocorticoid receptor ap-1 and /or nf- kappa b activity and use thereof

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JP2011503081A true JP2011503081A (ja) 2011-01-27
JP2011503081A5 JP2011503081A5 (enExample) 2011-04-07

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JP2010533163A Withdrawn JP2011503081A (ja) 2007-11-01 2008-10-30 グルココルチコイド受容体、ＡＰ−１および／またはＮＦ−κＢ活性の調節剤として有用な非ステロイド性化合物、並びにその使用

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US (1) US8309730B2 (enExample)
EP (1) EP2209780B1 (enExample)
JP (1) JP2011503081A (enExample)
CN (1) CN101910171A (enExample)
ES (1) ES2448839T3 (enExample)
WO (1) WO2009058944A2 (enExample)

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EP2209780B1 (en) 2014-01-01
ES2448839T3 (es) 2014-03-17
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CN101910171A (zh) 2010-12-08
US20110263494A1 (en) 2011-10-27

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