CN101910171A - 可用作糖皮质激素受体AP-1和/或者NF-κB活性调节剂的非甾类化合物及其用途 - Google Patents

可用作糖皮质激素受体AP-1和/或者NF-κB活性调节剂的非甾类化合物及其用途 Download PDF

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Publication number
CN101910171A
CN101910171A CN2008801237144A CN200880123714A CN101910171A CN 101910171 A CN101910171 A CN 101910171A CN 2008801237144 A CN2008801237144 A CN 2008801237144A CN 200880123714 A CN200880123714 A CN 200880123714A CN 101910171 A CN101910171 A CN 101910171A
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alkyl
substituted
hydrogen
inhibitor
aryl
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T·G·M·达
肖海云
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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CN2008801237144A 2007-11-01 2008-10-30 可用作糖皮质激素受体AP-1和/或者NF-κB活性调节剂的非甾类化合物及其用途 Pending CN101910171A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US98451507P 2007-11-01 2007-11-01
US60/984,515 2007-11-01
PCT/US2008/081702 WO2009058944A2 (en) 2007-11-01 2008-10-30 Nonsteroidal compounds useful as modulators of glucocorticoid receptor ap-1 and /or nf- kappa b activity and use thereof

Publications (1)

Publication Number Publication Date
CN101910171A true CN101910171A (zh) 2010-12-08

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CN2008801237144A Pending CN101910171A (zh) 2007-11-01 2008-10-30 可用作糖皮质激素受体AP-1和/或者NF-κB活性调节剂的非甾类化合物及其用途

Country Status (6)

Country Link
US (1) US8309730B2 (enExample)
EP (1) EP2209780B1 (enExample)
JP (1) JP2011503081A (enExample)
CN (1) CN101910171A (enExample)
ES (1) ES2448839T3 (enExample)
WO (1) WO2009058944A2 (enExample)

Cited By (1)

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CN109761976A (zh) * 2013-11-25 2019-05-17 科赛普特治疗公司 八氢稠合的氮杂萘烷糖皮质激素受体调节剂

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CN109761976A (zh) * 2013-11-25 2019-05-17 科赛普特治疗公司 八氢稠合的氮杂萘烷糖皮质激素受体调节剂
CN109761976B (zh) * 2013-11-25 2021-11-23 科赛普特治疗公司 八氢稠合的氮杂萘烷糖皮质激素受体调节剂

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US20110263494A1 (en) 2011-10-27
US8309730B2 (en) 2012-11-13
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