JP2010531313A5 - - Google Patents

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Publication number
JP2010531313A5
JP2010531313A5 JP2010513710A JP2010513710A JP2010531313A5 JP 2010531313 A5 JP2010531313 A5 JP 2010531313A5 JP 2010513710 A JP2010513710 A JP 2010513710A JP 2010513710 A JP2010513710 A JP 2010513710A JP 2010531313 A5 JP2010531313 A5 JP 2010531313A5
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JP
Japan
Prior art keywords
phenyl
unsubstituted
independently
benzimidazole
methyl
Prior art date
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Granted
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JP2010513710A
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English (en)
Japanese (ja)
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JP5492770B2 (ja
JP2010531313A (ja
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Priority claimed from PCT/EP2008/004639 external-priority patent/WO2009000413A1/en
Publication of JP2010531313A publication Critical patent/JP2010531313A/ja
Publication of JP2010531313A5 publication Critical patent/JP2010531313A5/ja
Application granted granted Critical
Publication of JP5492770B2 publication Critical patent/JP5492770B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2010513710A 2007-06-26 2008-06-11 ベンゾイミダゾール及びアザベンゾイミダゾールの位置選択的銅触媒合成 Expired - Fee Related JP5492770B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07290800 2007-06-26
EP07290800.7 2007-06-26
PCT/EP2008/004639 WO2009000413A1 (en) 2007-06-26 2008-06-11 A regioselective copper catalyzed synthesis of benzimidazoles and azabenzimidazoles

Publications (3)

Publication Number Publication Date
JP2010531313A JP2010531313A (ja) 2010-09-24
JP2010531313A5 true JP2010531313A5 (https=) 2011-07-07
JP5492770B2 JP5492770B2 (ja) 2014-05-14

Family

ID=38646504

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010513710A Expired - Fee Related JP5492770B2 (ja) 2007-06-26 2008-06-11 ベンゾイミダゾール及びアザベンゾイミダゾールの位置選択的銅触媒合成

Country Status (12)

Country Link
US (1) US8735586B2 (https=)
EP (1) EP2173721B1 (https=)
JP (1) JP5492770B2 (https=)
KR (1) KR20100023907A (https=)
CN (1) CN101687815A (https=)
AT (1) ATE539063T1 (https=)
AU (1) AU2008267444A1 (https=)
BR (1) BRPI0813271A2 (https=)
CA (1) CA2691857A1 (https=)
IL (1) IL202823A0 (https=)
MX (1) MX2009013753A (https=)
WO (1) WO2009000413A1 (https=)

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DK2519522T3 (en) 2009-12-30 2014-12-08 Arqule Inc SUBSTITUTED IDAZOPYRIDINYL AMINOPYRIDINE COMPOUNDS
JP5894161B2 (ja) 2010-08-25 2016-03-23 ネオファーム カンパニー， リミテッド 新規の複素環化合物及びこれを用いた炎症性疾患治療用組成物
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US8815854B2 (en) 2011-06-24 2014-08-26 Arqule, Inc. Substituted imidazopyridinyl compounds
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US9073878B2 (en) 2012-11-21 2015-07-07 Zenith Epigenetics Corp. Cyclic amines as bromodomain inhibitors
US9765039B2 (en) 2012-11-21 2017-09-19 Zenith Epigenetics Ltd. Biaryl derivatives as bromodomain inhibitors
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CN103130811B (zh) * 2013-03-11 2015-02-25 河南师范大学 一种5,6-二氢吡唑并[1,5-c]喹唑啉类化合物的合成方法
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CN103965136B (zh) * 2014-05-07 2016-09-07 苏州波菲特新材料科技有限公司 一种制备n-甲基噻唑啉-2-酮类化合物的方法
EP3227281A4 (en) 2014-12-01 2018-05-30 Zenith Epigenetics Ltd. Substituted pyridinones as bromodomain inhibitors
HK1246273B (en) 2014-12-01 2019-12-06 恒翼生物医药(上海)股份有限公司 Substituted pyridines as bromodomain inhibitors
EP3230277B1 (en) 2014-12-11 2019-09-18 Zenith Epigenetics Ltd. Substituted heterocycles as bromodomain inhibitors
HK1245247A1 (zh) 2014-12-17 2018-08-24 恒翼生物医药科技(上海)有限公司 溴结构域的抑制剂
US10189841B2 (en) 2015-11-20 2019-01-29 Forma Therapeutics, Inc. Purinones as ubiquitin-specific protease 1 inhibitors
CN106519250A (zh) * 2016-09-29 2017-03-22 辽宁石油化工大学 含氮小分子有机配体调节荧光发射性质的一维链状铜配位聚合物的制备方法
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