JP2010523692A5 - - Google Patents

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Publication number
JP2010523692A5
JP2010523692A5 JP2010503169A JP2010503169A JP2010523692A5 JP 2010523692 A5 JP2010523692 A5 JP 2010523692A5 JP 2010503169 A JP2010503169 A JP 2010503169A JP 2010503169 A JP2010503169 A JP 2010503169A JP 2010523692 A5 JP2010523692 A5 JP 2010523692A5
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JP
Japan
Prior art keywords
compound
chloro
pharmaceutically acceptable
acceptable salt
adamantan
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2010503169A
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English (en)
Japanese (ja)
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JP2010523692A (ja
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Publication date
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Priority claimed from PCT/US2008/059700 external-priority patent/WO2008127924A1/en
Publication of JP2010523692A publication Critical patent/JP2010523692A/ja
Publication of JP2010523692A5 publication Critical patent/JP2010523692A5/ja
Ceased legal-status Critical Current

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JP2010503169A 2007-04-11 2008-04-09 新規合成物 Ceased JP2010523692A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07105938 2007-04-11
US92325107P 2007-04-13 2007-04-13
PCT/US2008/059700 WO2008127924A1 (en) 2007-04-11 2008-04-09 Novel compounds

Publications (2)

Publication Number Publication Date
JP2010523692A JP2010523692A (ja) 2010-07-15
JP2010523692A5 true JP2010523692A5 (US07846941-20101207-C00217.png) 2011-05-26

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ID=39864303

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010503169A Ceased JP2010523692A (ja) 2007-04-11 2008-04-09 新規合成物

Country Status (10)

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US (1) US20100137377A1 (US07846941-20101207-C00217.png)
EP (1) EP2152081B1 (US07846941-20101207-C00217.png)
JP (1) JP2010523692A (US07846941-20101207-C00217.png)
CN (1) CN101677562A (US07846941-20101207-C00217.png)
AR (1) AR066043A1 (US07846941-20101207-C00217.png)
CA (1) CA2683852A1 (US07846941-20101207-C00217.png)
CL (1) CL2008001049A1 (US07846941-20101207-C00217.png)
ES (1) ES2399912T3 (US07846941-20101207-C00217.png)
TW (1) TWI361067B (US07846941-20101207-C00217.png)
WO (1) WO2008127924A1 (US07846941-20101207-C00217.png)

Families Citing this family (29)

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US8138342B2 (en) * 2004-10-12 2012-03-20 High Point Pharmacueticals, LLC 11β-hydroxysteroid dehydrogenase type 1 active spiro compounds
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US20100168083A1 (en) * 2006-03-21 2010-07-01 Soren Ebdrup Adamantane derivatives for the treatment of the metabolic syndrome
AU2007236049A1 (en) 2006-04-07 2007-10-18 High Point Pharmaceuticals, Llc 11beta-hydroxysteroid dehydrogenase type 1 active compounds
EP2038255A2 (en) * 2006-06-16 2009-03-25 High Point Pharmaceuticals, LLC Pharmaceutical use of substituted piperidine carboxamides
US8048908B2 (en) * 2006-07-13 2011-11-01 High Point Pharmaceuticals, Llc 11β-hydroxysteroid dehydrogenase type 1 active compounds
EP1878721A1 (en) * 2006-07-13 2008-01-16 Novo Nordisk A/S 4-Piperidylbenzamides as 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors
EP2125704A1 (en) * 2007-02-23 2009-12-02 High Point Pharmaceuticals, LLC N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
US20110003852A1 (en) * 2007-02-23 2011-01-06 Soren Ebdrup N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
EA016951B1 (ru) 2007-02-23 2012-08-30 ХАЙ ПОЙНТ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи N-АДАМАНТИЛБЕНЗАМИДЫ В КАЧЕСТВЕ ИНГИБИТОРОВ 11-β-ГИДРОКСИСТЕРОИДДЕГИДРОГЕНАЗЫ
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JP2010520864A (ja) * 2007-03-09 2010-06-17 ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー ヒドロキシステロイドデヒドロゲナーゼインヒビターとしてのインドール−及びベンズイミダゾールアミド類
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JP2010526777A (ja) * 2007-04-24 2010-08-05 ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー 置換アミドの医薬用途
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WO2012015715A1 (en) 2010-07-27 2012-02-02 High Point Pharmaceuticals, Llc Substituted thiazol-2-ylamine derivatives, pharmaceutical compositions, and methods of use as 11-beta hsd1 modulators
EP2612848A4 (en) * 2010-09-03 2013-12-25 Dainippon Sumitomo Pharma Co CYCLIC AMIDE DERIVATIVE
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors

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EP1948190A2 (en) * 2005-11-01 2008-07-30 Transtech Pharma Pharmaceutical use of substituted amides
US20100168083A1 (en) * 2006-03-21 2010-07-01 Soren Ebdrup Adamantane derivatives for the treatment of the metabolic syndrome
AU2007236049A1 (en) * 2006-04-07 2007-10-18 High Point Pharmaceuticals, Llc 11beta-hydroxysteroid dehydrogenase type 1 active compounds
US20110003852A1 (en) * 2007-02-23 2011-01-06 Soren Ebdrup N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
EP2125704A1 (en) * 2007-02-23 2009-12-02 High Point Pharmaceuticals, LLC N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
EA016951B1 (ru) * 2007-02-23 2012-08-30 ХАЙ ПОЙНТ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи N-АДАМАНТИЛБЕНЗАМИДЫ В КАЧЕСТВЕ ИНГИБИТОРОВ 11-β-ГИДРОКСИСТЕРОИДДЕГИДРОГЕНАЗЫ
JP2010520864A (ja) * 2007-03-09 2010-06-17 ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー ヒドロキシステロイドデヒドロゲナーゼインヒビターとしてのインドール−及びベンズイミダゾールアミド類
US20100056600A1 (en) * 2007-03-28 2010-03-04 Soren Ebdrup 11beta-hsd1 active compounds
JP2010526777A (ja) * 2007-04-24 2010-08-05 ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー 置換アミドの医薬用途
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