JP2010515882A - 睡眠関連障害を含むgaba関連神経学的障害を処置するためのgタンパク質共役受容体およびその調節因子 - Google Patents

睡眠関連障害を含むgaba関連神経学的障害を処置するためのgタンパク質共役受容体およびその調節因子 Download PDF

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JP2010515882A
JP2010515882A JP2009544931A JP2009544931A JP2010515882A JP 2010515882 A JP2010515882 A JP 2010515882A JP 2009544931 A JP2009544931 A JP 2009544931A JP 2009544931 A JP2009544931 A JP 2009544931A JP 2010515882 A JP2010515882 A JP 2010515882A
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ディディエー バグノル,
アンドリュー ジェイ. グロッティック,
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アリーナ ファーマシューティカルズ, インコーポレイテッド
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JP2009544931A 2007-01-05 2008-01-04 睡眠関連障害を含むgaba関連神経学的障害を処置するためのgタンパク質共役受容体およびその調節因子 Withdrawn JP2010515882A (ja)

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US87879607P 2007-01-05 2007-01-05
PCT/US2008/000116 WO2008085888A1 (en) 2007-01-05 2008-01-04 G protein-coupled receptor and modulators thereof for the treatment of gaba-related neurological disorders including sleep-related disorders

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JP2010515882A true JP2010515882A (ja) 2010-05-13
JP2010515882A5 JP2010515882A5 (enExample) 2012-03-08

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US (1) US20110038850A1 (enExample)
EP (1) EP2117577A1 (enExample)
JP (1) JP2010515882A (enExample)
WO (1) WO2008085888A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2017511386A (ja) * 2014-04-15 2017-04-20 バランス セラピューティックス,インコーポレイテッド 過眠症を治療するための方法

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TN2016000542A1 (en) 2014-06-03 2018-04-04 Idorsia Pharmaceuticals Ltd Pyrazole compounds and their use as t-type calcium channel blockers
ES2693052T3 (es) 2014-09-15 2018-12-07 Idorsia Pharmaceuticals Ltd Compuestos de triazol como bloqueantes de los canales de calcio de tipo T
HRP20220463T1 (hr) 2016-12-16 2022-05-27 Idorsia Pharmaceuticals Ltd Farmaceutska kombinacija koja sadrži blokator kalcijevih kanala t-tipa
WO2018141961A1 (en) 2017-02-06 2018-08-09 Idorsia Pharmaceuticals Ltd A novel process for the synthesis of 1-aryl-1-trifluoromethylcyclopropanes
EP3684463B1 (en) 2017-09-19 2025-05-14 Neuroenhancement Lab, LLC Method and apparatus for neuroenhancement
US11717686B2 (en) 2017-12-04 2023-08-08 Neuroenhancement Lab, LLC Method and apparatus for neuroenhancement to facilitate learning and performance
US11318277B2 (en) 2017-12-31 2022-05-03 Neuroenhancement Lab, LLC Method and apparatus for neuroenhancement to enhance emotional response
US12280219B2 (en) 2017-12-31 2025-04-22 NeuroLight, Inc. Method and apparatus for neuroenhancement to enhance emotional response
US11364361B2 (en) 2018-04-20 2022-06-21 Neuroenhancement Lab, LLC System and method for inducing sleep by transplanting mental states
US11452839B2 (en) 2018-09-14 2022-09-27 Neuroenhancement Lab, LLC System and method of improving sleep

Family Cites Families (5)

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IL149569A0 (en) * 1999-11-17 2002-11-10 Arena Pharm Inc Endogenous and non-endogenous versions of human g protein-coupled receptors
WO2005011612A2 (en) * 2003-07-31 2005-02-10 The Research Foundation Of State University Of New York Alpha 4 beta 2 delta gaba-a receptors as a strategy for pms and alcoholism
WO2005060625A2 (en) * 2003-12-11 2005-07-07 The Trustees Of Columbia University In The City Of New York Grp receptor-related methods for treating and preventing fear-related disorders
GB0328796D0 (en) * 2003-12-12 2004-01-14 Biofocus Plc Compounds which interact with the G-protein coupled receptor family
US8354241B2 (en) * 2005-04-27 2013-01-15 Arena Pharmaceuticals, Inc. Methods for identifying a GLP-1 secretagogue

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2017511386A (ja) * 2014-04-15 2017-04-20 バランス セラピューティックス,インコーポレイテッド 過眠症を治療するための方法
JP2020105200A (ja) * 2014-04-15 2020-07-09 バランス セラピューティックス,インコーポレイテッド 過眠症を治療するための方法

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US20110038850A1 (en) 2011-02-17
WO2008085888A1 (en) 2008-07-17

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