JP2010510286A - 非ステロイド非イオン化親水性薬物の送達系 - Google Patents
非ステロイド非イオン化親水性薬物の送達系 Download PDFInfo
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- JP2010510286A JP2010510286A JP2009537627A JP2009537627A JP2010510286A JP 2010510286 A JP2010510286 A JP 2010510286A JP 2009537627 A JP2009537627 A JP 2009537627A JP 2009537627 A JP2009537627 A JP 2009537627A JP 2010510286 A JP2010510286 A JP 2010510286A
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- drug
- vinyl acetate
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Images
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
- A61K9/0036—Devices retained in the vagina or cervix for a prolonged period, e.g. intravaginal rings, medicated tampons, medicated diaphragms
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Urology & Nephrology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Gynecology & Obstetrics (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06124598 | 2006-11-22 | ||
| PCT/EP2007/062626 WO2008062008A1 (en) | 2006-11-22 | 2007-11-21 | Delivery system for a non-steroidal non-ionized hydrophilic drug |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010510286A true JP2010510286A (ja) | 2010-04-02 |
| JP2010510286A5 JP2010510286A5 (enExample) | 2011-01-13 |
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| JP2009537627A Withdrawn JP2010510286A (ja) | 2006-11-22 | 2007-11-21 | 非ステロイド非イオン化親水性薬物の送達系 |
| JP2009537628A Withdrawn JP2010510287A (ja) | 2006-11-22 | 2007-11-21 | リスペリドン用送達システム |
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| JP2009537628A Withdrawn JP2010510287A (ja) | 2006-11-22 | 2007-11-21 | リスペリドン用送達システム |
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|---|---|
| US (2) | US20100104619A1 (enExample) |
| EP (2) | EP2094348A1 (enExample) |
| JP (2) | JP2010510286A (enExample) |
| CA (2) | CA2670157A1 (enExample) |
| MX (2) | MX2009005444A (enExample) |
| WO (2) | WO2008062009A1 (enExample) |
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| GB0222522D0 (en) | 2002-09-27 | 2002-11-06 | Controlled Therapeutics Sct | Water-swellable polymers |
| US7858110B2 (en) * | 2003-08-11 | 2010-12-28 | Endo Pharmaceuticals Solutions, Inc. | Long term drug delivery devices with polyurethane based polymers and their manufacture |
| CA2437639C (en) * | 2003-08-11 | 2016-07-05 | Valera Pharmaceuticals, Inc. | Long term drug delivery devices with polyurethane based polymers and their manufacture |
| GB0417401D0 (en) | 2004-08-05 | 2004-09-08 | Controlled Therapeutics Sct | Stabilised prostaglandin composition |
| GB0613333D0 (en) | 2006-07-05 | 2006-08-16 | Controlled Therapeutics Sct | Hydrophilic polyurethane compositions |
| GB0613638D0 (en) * | 2006-07-08 | 2006-08-16 | Controlled Therapeutics Sct | Polyurethane elastomers |
| MX2009000053A (es) * | 2006-07-12 | 2009-02-23 | Controlled Therapeutics Sct | Polimero para el suministro de medicamentos con sal clorhidrato de clindamicina. |
| GB0620685D0 (en) | 2006-10-18 | 2006-11-29 | Controlled Therapeutics Sct | Bioresorbable polymers |
| US20100104619A1 (en) * | 2006-11-22 | 2010-04-29 | N.V. Organon | Delivery system for a non-steroidal non-ionized hydrophilic drug |
| WO2009129459A1 (en) * | 2008-04-18 | 2009-10-22 | Combinent Biomedical Systems, Inc. | Devices that include ethylene-vinyl acetate copolymers and methods of making and using same |
| KR101707791B1 (ko) * | 2008-09-30 | 2017-02-17 | 엔도 파마슈티컬즈, 솔루션스 아이엔씨. | 리스페리돈 전달용 이식형 장치 |
| CA2792484C (en) * | 2009-03-12 | 2017-10-31 | Delpor, Inc. | Implantable device for long-term delivery of drugs |
| WO2011116132A1 (en) | 2010-03-16 | 2011-09-22 | Titan Pharmaceuticals, Inc. | Heterogeneous implantable devices for drug delivery |
| US20170319833A1 (en) * | 2010-03-28 | 2017-11-09 | Evestra, Inc. | Intravaginal drug delivery device |
| US8580294B2 (en) | 2010-10-19 | 2013-11-12 | International Partnership For Microbicides | Platinum-catalyzed intravaginal rings |
| DE102013011399A1 (de) | 2012-07-31 | 2014-02-06 | Amw Gmbh | Implantat mit Risperidon |
| US10137031B2 (en) | 2013-11-14 | 2018-11-27 | International Partnership For Microbicides, Inc. | Combination therapy intravaginal rings |
| US10406336B2 (en) * | 2016-08-03 | 2019-09-10 | Neil S. Davey | Adjustable rate drug delivery implantable device |
| CA3087238A1 (en) | 2018-05-24 | 2019-11-28 | Celanese EVA Performance Polymers Corporation | Implantable device for sustained release of a macromolecular drug compound |
| EP3803866A4 (en) | 2018-05-24 | 2022-03-16 | Nureva Inc. | METHOD, APPARATUS, AND COMPUTER READABLE MATERIALS FOR MANAGING SEMI-CONSTANT (PERSISTENT) SOUND SOURCES IN MICROPHONE CATCH/HOME AREAS |
| CN111989068B (zh) * | 2018-05-24 | 2024-10-25 | 塞拉尼斯伊娃高性能聚合物公司 | 用于持续释放大分子药物化合物的可植入器件 |
| EP4329734A4 (en) | 2021-04-26 | 2025-04-02 | Celanese EVA Performance Polymers LLC | Implantable device for the delayed release of a macromolecular drug compound |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4016251A (en) * | 1972-08-17 | 1977-04-05 | Alza Corporation | Vaginal drug dispensing device |
| US4469671A (en) * | 1983-02-22 | 1984-09-04 | Eli Lilly And Company | Contraceptive device |
| GB9326255D0 (en) * | 1993-12-23 | 1994-02-23 | Roussel Lab Ltd | Medical device for the prevention and treatment of cancer |
| DK0836473T3 (da) * | 1995-07-04 | 2002-02-11 | Akzo Nobel Nv | Ringformede indretninger |
| US20040044080A1 (en) * | 1997-10-28 | 2004-03-04 | Place Virgil A. | Treatment of dyspareunia with topically administered nitroglycerin formulations |
| IL157771A0 (en) * | 2001-03-27 | 2004-03-28 | Galen Chemicals Ltd | Intravaginal drug delivery devices for the administration of an antimicrobial agent |
| US6887270B2 (en) * | 2002-02-08 | 2005-05-03 | Boston Scientific Scimed, Inc. | Implantable or insertable medical device resistant to microbial growth and biofilm formation |
| CA2496798A1 (en) * | 2002-08-30 | 2004-03-11 | Alza Corporation | Embossable and writable multilaminate backing construction |
| KR101242486B1 (ko) * | 2004-01-12 | 2013-03-13 | 더 트러스티스 오브 더 유니버시티 오브 펜실베니아 | 장기 전달을 위한 제형 및 그의 이용 방법 |
| JP2007530500A (ja) * | 2004-03-24 | 2007-11-01 | ナームローゼ・フエンノートチヤツプ・オルガノン | ポリエチレン酢酸ビニル共重合体に基づく薬物送達システム |
| EP1824460B1 (en) * | 2004-11-10 | 2014-12-24 | Tolmar Therapeutics, Inc. | A stabilized polymeric delivery system |
| US20100104619A1 (en) * | 2006-11-22 | 2010-04-29 | N.V. Organon | Delivery system for a non-steroidal non-ionized hydrophilic drug |
| AU2007324467A1 (en) * | 2006-11-22 | 2008-05-29 | N.V. Organon | Vaginal delivery system for mirtazapine |
-
2007
- 2007-11-21 US US12/515,897 patent/US20100104619A1/en not_active Abandoned
- 2007-11-21 WO PCT/EP2007/062628 patent/WO2008062009A1/en not_active Ceased
- 2007-11-21 US US12/515,882 patent/US20100203104A1/en not_active Abandoned
- 2007-11-21 JP JP2009537627A patent/JP2010510286A/ja not_active Withdrawn
- 2007-11-21 EP EP07822772A patent/EP2094348A1/en not_active Withdrawn
- 2007-11-21 WO PCT/EP2007/062626 patent/WO2008062008A1/en not_active Ceased
- 2007-11-21 JP JP2009537628A patent/JP2010510287A/ja not_active Withdrawn
- 2007-11-21 EP EP07822774A patent/EP2094270A1/en not_active Withdrawn
- 2007-11-21 CA CA002670157A patent/CA2670157A1/en not_active Abandoned
- 2007-11-21 CA CA002670454A patent/CA2670454A1/en not_active Abandoned
- 2007-11-21 MX MX2009005444A patent/MX2009005444A/es not_active Application Discontinuation
- 2007-11-21 MX MX2009005445A patent/MX2009005445A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MX2009005445A (es) | 2009-06-02 |
| WO2008062009A1 (en) | 2008-05-29 |
| MX2009005444A (es) | 2009-06-02 |
| EP2094348A1 (en) | 2009-09-02 |
| JP2010510287A (ja) | 2010-04-02 |
| CA2670454A1 (en) | 2008-05-29 |
| US20100104619A1 (en) | 2010-04-29 |
| EP2094270A1 (en) | 2009-09-02 |
| CA2670157A1 (en) | 2008-05-29 |
| WO2008062008A1 (en) | 2008-05-29 |
| US20100203104A1 (en) | 2010-08-12 |
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