JP2010508328A5 - - Google Patents

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Publication number
JP2010508328A5
JP2010508328A5 JP2009535078A JP2009535078A JP2010508328A5 JP 2010508328 A5 JP2010508328 A5 JP 2010508328A5 JP 2009535078 A JP2009535078 A JP 2009535078A JP 2009535078 A JP2009535078 A JP 2009535078A JP 2010508328 A5 JP2010508328 A5 JP 2010508328A5
Authority
JP
Japan
Prior art keywords
trifluoromethyl
phenyl
methyl
pyrazole
tetrahydropyrano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2009535078A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010508328A (ja
Filing date
Publication date
Priority claimed from GB0621967A external-priority patent/GB0621967D0/en
Priority claimed from GB0717262A external-priority patent/GB0717262D0/en
Application filed filed Critical
Priority claimed from PCT/EP2007/061794 external-priority patent/WO2008053031A1/en
Publication of JP2010508328A publication Critical patent/JP2010508328A/ja
Publication of JP2010508328A5 publication Critical patent/JP2010508328A5/ja
Withdrawn legal-status Critical Current

Links

JP2009535078A 2006-11-03 2007-11-01 Ampa受容体を強化する化合物および医薬におけるその使用 Withdrawn JP2010508328A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0621967A GB0621967D0 (en) 2006-11-03 2006-11-03 Compounds
GB0717262A GB0717262D0 (en) 2007-09-05 2007-09-05 Compounds
PCT/EP2007/061794 WO2008053031A1 (en) 2006-11-03 2007-11-01 Compounds which potentiate ampa receptor and uses thereof in medicine

Publications (2)

Publication Number Publication Date
JP2010508328A JP2010508328A (ja) 2010-03-18
JP2010508328A5 true JP2010508328A5 (https=) 2010-12-24

Family

ID=39099804

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009535078A Withdrawn JP2010508328A (ja) 2006-11-03 2007-11-01 Ampa受容体を強化する化合物および医薬におけるその使用

Country Status (6)

Country Link
US (1) US20100137276A1 (https=)
EP (1) EP2086643B1 (https=)
JP (1) JP2010508328A (https=)
AT (1) ATE502675T1 (https=)
DE (1) DE602007013450D1 (https=)
WO (1) WO2008053031A1 (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0711088D0 (en) * 2007-06-08 2007-07-18 Glaxo Group Ltd Compounds
GB0711089D0 (en) * 2007-06-08 2007-07-18 Glaxo Group Ltd Compounds
JP6134654B2 (ja) * 2012-02-08 2017-05-24 武田薬品工業株式会社 複素環化合物およびその用途
US10604484B2 (en) 2015-04-29 2020-03-31 Janssen Pharmaceutica Nv Indolone compounds and their use as AMPA receptor modulators
RS61688B1 (sr) 2015-04-29 2021-05-31 Janssen Pharmaceutica Nv Azabenzimidazoli i njihiova upotreba kao modulatori ampa receptora
WO2016176457A1 (en) * 2015-04-29 2016-11-03 Janssen Pharmaceutica Nv Imidazopyrazines and pyrazolopyrimidines and their use as ampa receptor modulators
AU2016255424B2 (en) 2015-04-29 2020-10-08 Janssen Pharmaceutica Nv Benzimidazolone and benzothiazolone compounds and their use as AMPA receptor modulators
GB201702221D0 (en) * 2017-02-10 2017-03-29 Univ Of Sussex Compounds
GB201803340D0 (en) 2018-03-01 2018-04-18 Univ Of Sussex Compounds
WO2025231416A1 (en) * 2024-05-03 2025-11-06 Rapport Therapeutics, Inc. Methods of use of ampa receptor modulators

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2159479B1 (es) 1999-10-25 2002-05-01 Menarini Lab Nuevos indazoles como inhibidores de la ciclooxigenasa-ii
KR20070050070A (ko) 2004-08-09 2007-05-14 글락소 그룹 리미티드 글루타메이트 수용체를 강화시키는 화합물 및 의약에서의그의 용도

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