JP2010501541A5 - - Google Patents

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Publication number
JP2010501541A5
JP2010501541A5 JP2009525123A JP2009525123A JP2010501541A5 JP 2010501541 A5 JP2010501541 A5 JP 2010501541A5 JP 2009525123 A JP2009525123 A JP 2009525123A JP 2009525123 A JP2009525123 A JP 2009525123A JP 2010501541 A5 JP2010501541 A5 JP 2010501541A5
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JP
Japan
Prior art keywords
formula
compound
substituted
phenyl
pyridin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2009525123A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010501541A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2007/002405 external-priority patent/WO2008023248A2/en
Publication of JP2010501541A publication Critical patent/JP2010501541A/ja
Publication of JP2010501541A5 publication Critical patent/JP2010501541A5/ja
Pending legal-status Critical Current

Links

JP2009525123A 2006-08-24 2007-08-22 抗菌活性を有する新規マクロライド及びケトライド Pending JP2010501541A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1336MU2006 2006-08-24
PCT/IB2007/002405 WO2008023248A2 (en) 2006-08-24 2007-08-22 Novel macrolides and ketolides having antimicrobial activity

Publications (2)

Publication Number Publication Date
JP2010501541A JP2010501541A (ja) 2010-01-21
JP2010501541A5 true JP2010501541A5 (cg-RX-API-DMAC10.html) 2010-10-14

Family

ID=39107171

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009525123A Pending JP2010501541A (ja) 2006-08-24 2007-08-22 抗菌活性を有する新規マクロライド及びケトライド

Country Status (7)

Country Link
US (1) US8097594B2 (cg-RX-API-DMAC10.html)
EP (1) EP2056844A4 (cg-RX-API-DMAC10.html)
JP (1) JP2010501541A (cg-RX-API-DMAC10.html)
KR (1) KR20090042971A (cg-RX-API-DMAC10.html)
CN (1) CN101541331A (cg-RX-API-DMAC10.html)
CA (1) CA2661538A1 (cg-RX-API-DMAC10.html)
WO (1) WO2008023248A2 (cg-RX-API-DMAC10.html)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8222243B2 (en) 2007-08-27 2012-07-17 Dart Neuroscience (Cayman) Ltd Therapeutic isoxazole compounds
WO2009081970A1 (ja) * 2007-12-26 2009-07-02 Eisai R & D Management Co., Ltd. ヘテロ環置換ピリジン誘導体の製造方法
EP2435460B1 (en) * 2009-05-27 2015-01-07 Wockhardt Limited Ketolide compounds having antimicrobial activity
RU2601550C2 (ru) 2010-12-09 2016-11-10 Вокхардт Лимитед Кетолидные соединения
CN103619849B (zh) * 2011-03-01 2016-05-25 沃克哈特有限公司 酮内酯中间体的制备方法
EP2688900B1 (en) * 2011-03-22 2016-09-28 Wockhardt Limited Process for preparation of ketolide compounds
WO2012129564A2 (en) 2011-03-24 2012-09-27 H. Lee Moffitt Cancer Center And Research Institute, Inc. Proteasome chymotrypsin-like inhibition using pi-1833 analogs
CN102260225B (zh) * 2011-06-02 2013-08-21 蒋杰 用于抑制肿瘤转移和肿瘤血管生长的苯基哌嗪类衍生物
JP2017531663A (ja) * 2014-10-08 2017-10-26 プレジデント アンド フェローズ オブ ハーバード カレッジ 14員ケトライドならびにそれらの調製および使用の方法
KR20190129863A (ko) * 2017-03-16 2019-11-20 욱크하르트 리미티드 케톨라이드 화합물의 제조 방법
ES2948122A1 (es) * 2022-02-10 2023-08-31 Fundacion Instituto De Investig Sanitaria Aragon Compuestos para el tratamiento y/o prevención de una infección o enfermedad causada por Helicobacter o Campylobacter

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2473525A1 (fr) 1980-01-11 1981-07-17 Roussel Uclaf Nouvelles oximes derivees de l'erythromycine, leur procede de preparation et leur application comme medicaments
US4331803A (en) 1980-06-04 1982-05-25 Taisho Pharmaceutical Co., Ltd. Novel erythromycin compounds
YU43006B (en) 1981-03-06 1989-02-28 Pliva Pharm & Chem Works Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
FR2719587B1 (fr) 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
DE69733439T2 (de) 1996-09-04 2006-05-04 Abbott Laboratories, Abbott Park 6-o-Substituierte Ketoliden mit antibakteriellen Wirkung
MXPA03001607A (es) 2000-08-22 2003-06-04 Basilea Pharmaceutica Ag Nuevos macrolidos con actividad antibacteriana.
JP2004531471A (ja) * 2000-12-21 2004-10-14 グラクソ グループ リミテッド マクロライド抗生物質
GB0031312D0 (en) 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
MXPA04000565A (es) 2001-07-19 2005-06-17 Cv Therapeutics Inc Compuestos de piperazina sustituidos y su uso como inhibidores de oxidacion de acidos grasos.
GB0127349D0 (en) 2001-11-14 2002-01-02 Glaxo Group Ltd Macrolides
US6995143B2 (en) 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
US6727229B2 (en) 2002-08-19 2004-04-27 Enanta Pharmaceuticals, Inc. 11,12-substituted lactone ketolide derivatives having antibacterial activity
HRP20090302T1 (hr) * 2005-02-09 2009-07-31 Basilea Pharmaceutica Ag Novi makrolidi

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