JP2009541205A - P2x7調節因子としてのビシクロへテロアリール化合物およびその使用 - Google Patents

P2x7調節因子としてのビシクロへテロアリール化合物およびその使用 Download PDF

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JP2009541205A
JP2009541205A JP2009500513A JP2009500513A JP2009541205A JP 2009541205 A JP2009541205 A JP 2009541205A JP 2009500513 A JP2009500513 A JP 2009500513A JP 2009500513 A JP2009500513 A JP 2009500513A JP 2009541205 A JP2009541205 A JP 2009541205A
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substituted
unsubstituted
compound
alkyl
disease
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JP2009541205A5 (enExample
Inventor
マイケル ジー. ケリー,
ジョン キンケード,
ユンフェン ファン,
イェユー カオ,
カール カウブ,
スミスラ ゴウルガリ,
チャン ワン,
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レノビス, インコーポレイテッド
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Priority claimed from PCT/US2007/006676 external-priority patent/WO2007109154A2/en
Publication of JP2009541205A publication Critical patent/JP2009541205A/ja
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
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    • C07D217/24Oxygen atoms
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    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
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  • Diabetes (AREA)
  • Pulmonology (AREA)
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JP2009500513A 2006-03-16 2007-03-16 P2x7調節因子としてのビシクロへテロアリール化合物およびその使用 Withdrawn JP2009541205A (ja)

Applications Claiming Priority (14)

Application Number Priority Date Filing Date Title
US78312106P 2006-03-16 2006-03-16
US78297306P 2006-03-16 2006-03-16
US78292206P 2006-03-16 2006-03-16
US78277606P 2006-03-16 2006-03-16
US78359006P 2006-03-16 2006-03-16
US78292306P 2006-03-16 2006-03-16
US78278206P 2006-03-16 2006-03-16
US78277506P 2006-03-16 2006-03-16
US78374806P 2006-03-16 2006-03-16
US78330406P 2006-03-16 2006-03-16
US83141606P 2006-07-17 2006-07-17
US84699306P 2006-09-25 2006-09-25
US91812307P 2007-03-15 2007-03-15
PCT/US2007/006676 WO2007109154A2 (en) 2006-03-16 2007-03-16 Bicycloheteroaryl compounds as p2x7 modulators and uses thereof

Publications (2)

Publication Number Publication Date
JP2009541205A true JP2009541205A (ja) 2009-11-26
JP2009541205A5 JP2009541205A5 (enExample) 2011-03-31

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ID=39878008

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JP2009500513A Withdrawn JP2009541205A (ja) 2006-03-16 2007-03-16 P2x7調節因子としてのビシクロへテロアリール化合物およびその使用

Country Status (3)

Country Link
US (1) US20090298825A1 (enExample)
EP (1) EP1996585A4 (enExample)
JP (1) JP2009541205A (enExample)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0200920D0 (sv) * 2002-03-25 2002-03-25 Astrazeneca Ab Novel compounds
AU2003301443A1 (en) * 2002-10-18 2004-05-04 E.I. Du Pont De Nemours And Company Azolecarboxamide herbicides
GB0312609D0 (en) * 2003-06-02 2003-07-09 Astrazeneca Ab Novel compounds

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EP1996585A4 (en) 2010-03-10
EP1996585A2 (en) 2008-12-03
US20090298825A1 (en) 2009-12-03

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