JP2009537600A - 新規１，４−ジアザ−ビシクロ［３．２．２］ノナン誘導体及びそれらの医学的使用 - Google Patents
新規１，４−ジアザ−ビシクロ［３．２．２］ノナン誘導体及びそれらの医学的使用 Download PDFInfo
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- JP2009537600A JP2009537600A JP2009511494A JP2009511494A JP2009537600A JP 2009537600 A JP2009537600 A JP 2009537600A JP 2009511494 A JP2009511494 A JP 2009511494A JP 2009511494 A JP2009511494 A JP 2009511494A JP 2009537600 A JP2009537600 A JP 2009537600A
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- alkyl
- diaza
- bicyclo
- pain
- disease
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Reproductive Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Endocrinology (AREA)
- Gynecology & Obstetrics (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pulmonology (AREA)
- Pregnancy & Childbirth (AREA)
- Psychology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Addiction (AREA)
- Vascular Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Child & Adolescent Psychology (AREA)
- Obesity (AREA)
- Dermatology (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US80252906P | 2006-05-23 | 2006-05-23 | |
| DKPA200600707 | 2006-05-23 | ||
| PCT/EP2007/054871 WO2007135122A1 (en) | 2006-05-23 | 2007-05-21 | Novel 1,4-diaza-bicyclo[3.2.2]nonane derivatives and their medical use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009537600A true JP2009537600A (ja) | 2009-10-29 |
| JP2009537600A5 JP2009537600A5 (enExample) | 2010-06-24 |
Family
ID=38353613
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009511494A Abandoned JP2009537600A (ja) | 2006-05-23 | 2007-05-21 | 新規１，４−ジアザ−ビシクロ［３．２．２］ノナン誘導体及びそれらの医学的使用 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20090186880A1 (enExample) |
| EP (1) | EP2027122B1 (enExample) |
| JP (1) | JP2009537600A (enExample) |
| AT (1) | ATE460416T1 (enExample) |
| DE (1) | DE602007005255D1 (enExample) |
| WO (1) | WO2007135122A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2011504909A (ja) * | 2007-11-30 | 2011-02-17 | ノイロサーチ アクティーゼルスカブ | 新規なカルボン酸４−フェニルアゾ−フェニルエステル誘導体及びモノアミン神経伝達物質再取り込み阻害薬としてのそれらの使用 |
| WO2009109517A1 (en) * | 2008-03-05 | 2009-09-11 | Neurosearch A/S | Novel 3,8-diaza-bicyclo[3.2.1]octane- and 3,9-diaza-bicyclo[3.3.1]-nonane-3-carboxylic acid ester derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| TWI558398B (zh) | 2009-09-22 | 2016-11-21 | 諾華公司 | 菸鹼乙醯膽鹼受體α７活化劑之用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60216830T2 (de) | 2001-02-06 | 2007-06-14 | Pfizer Products Inc., Groton | Pharmazeutische Zusammensetzungen zur Behandlung von Störungen des ZNS oder anderen Erkrankungen |
| JP2005510523A (ja) * | 2001-11-09 | 2005-04-21 | ファルマシア アンド アップジョン カンパニー リミティド ライアビリティー カンパニー | アザ二環式フェニル縮合複素環式化合物、及びα７ＮＡＣＨＲリガンドとしての当該化合物の使用 |
| RU2386633C2 (ru) * | 2004-05-07 | 2010-04-20 | Мемори Фармасьютиклз Корпорейшн | 1h-индазолы, бензотиазолы, 1, 2-бензоизоксазолы, 1, 2-бензоизотиазолы и хромоны и их получение и применения |
-
2007
- 2007-05-21 WO PCT/EP2007/054871 patent/WO2007135122A1/en not_active Ceased
- 2007-05-21 EP EP07729315A patent/EP2027122B1/en not_active Not-in-force
- 2007-05-21 AT AT07729315T patent/ATE460416T1/de not_active IP Right Cessation
- 2007-05-21 JP JP2009511494A patent/JP2009537600A/ja not_active Abandoned
- 2007-05-21 US US12/299,594 patent/US20090186880A1/en not_active Abandoned
- 2007-05-21 DE DE602007005255T patent/DE602007005255D1/de active Active
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007135122A1 (en) | 2007-11-29 |
| EP2027122A1 (en) | 2009-02-25 |
| ATE460416T1 (de) | 2010-03-15 |
| EP2027122B1 (en) | 2010-03-10 |
| US20090186880A1 (en) | 2009-07-23 |
| DE602007005255D1 (de) | 2010-04-22 |
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