JP2009537517A - ニコチン性アセチルコリン受容体リガンド１０１ - Google Patents
ニコチン性アセチルコリン受容体リガンド１０１ Download PDFInfo
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- JP2009537517A JP2009537517A JP2009510923A JP2009510923A JP2009537517A JP 2009537517 A JP2009537517 A JP 2009537517A JP 2009510923 A JP2009510923 A JP 2009510923A JP 2009510923 A JP2009510923 A JP 2009510923A JP 2009537517 A JP2009537517 A JP 2009537517A
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- furo
- azabicyclo
- spiro
- octane
- disease
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Classifications
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- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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Landscapes
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- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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| US74747606P | 2006-05-17 | 2006-05-17 | |
| US82497506P | 2006-09-08 | 2006-09-08 | |
| PCT/SE2007/000485 WO2007133155A1 (en) | 2006-05-17 | 2007-05-16 | Nicotinic acetylcholine receptor ligands 101 |
Publications (2)
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| JP2009537517A true JP2009537517A (ja) | 2009-10-29 |
| JP2009537517A5 JP2009537517A5 (https=) | 2010-04-02 |
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| CA (1) | CA2652610A1 (https=) |
| CL (1) | CL2007001405A1 (https=) |
| EC (1) | ECSP088971A (https=) |
| ES (1) | ES2392997T3 (https=) |
| IL (1) | IL195019A0 (https=) |
| MX (1) | MX2008014436A (https=) |
| NO (1) | NO20084915L (https=) |
| RU (1) | RU2441007C2 (https=) |
| SA (1) | SA07280244B1 (https=) |
| TW (1) | TW200813067A (https=) |
| UY (1) | UY30349A1 (https=) |
| WO (1) | WO2007133155A1 (https=) |
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| PE20060437A1 (es) | 2004-06-18 | 2006-06-08 | Novartis Ag | COMPUESTOS AZA-BICICLONONANOS COMO LIGANDOS COLINERGICOS DE nAChR |
| GB0415746D0 (en) | 2004-07-14 | 2004-08-18 | Novartis Ag | Organic compounds |
| GB0521508D0 (en) | 2005-10-21 | 2005-11-30 | Novartis Ag | Organic compounds |
| GB0525673D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| GB0525672D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| WO2009066107A1 (en) * | 2007-11-21 | 2009-05-28 | Astrazeneca Ab | Use of a nicotinic receptor agonist |
| JO3250B1 (ar) | 2009-09-22 | 2018-09-16 | Novartis Ag | إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7 |
| KR20140003580A (ko) | 2011-01-27 | 2014-01-09 | 노파르티스 아게 | 니코틴성 아세틸콜린 수용체 알파 7 활성화제의 용도 |
| WO2012127393A1 (en) | 2011-03-18 | 2012-09-27 | Novartis Ag | COMBINATIONS OF ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVATORS AND mGluR5 ANTAGONISTS FOR USE IN DOPAMINE INDUCED DYSKINESIA IN PARKINSON'S DISEASE |
| JP6162705B2 (ja) | 2011-10-20 | 2017-07-12 | ノバルティス アーゲー | アルファ７ニコチン性アセチルコリン受容体活性化剤による処置に対する応答性を予測するバイオマーカー |
| KR102043309B1 (ko) | 2012-12-11 | 2019-11-11 | 노파르티스 아게 | 알파 7 니코틴성 아세틸콜린 수용체 활성화제 치료에 대한 반응성의 예측 바이오마커 |
| CN105263492B (zh) | 2013-01-15 | 2018-04-10 | 诺华有限公司 | α7烟碱型乙酰胆碱受体激动剂在治疗发作性睡病中的应用 |
| BR112015016992A8 (pt) | 2013-01-15 | 2018-01-23 | Novartis Ag | uso de agonistas do receptor alfa 7 nicotínico de acetilcolina |
| EP2945633B1 (en) | 2013-01-15 | 2021-06-30 | Novartis AG | Use of alpha 7 nicotinic acetylcholine receptor agonists |
| US11209254B2 (en) * | 2016-03-09 | 2021-12-28 | Msato, Llc | Pellet shaped marking round for air rifles and pistols |
| HU231333B1 (hu) * | 2018-07-13 | 2023-01-28 | Richter Gedeon Nyrt | Spirokromán származékok |
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| JP2005527588A (ja) * | 2002-04-18 | 2005-09-15 | アストラゼネカ・アクチエボラーグ | チエニル化合物 |
| JP2005533012A (ja) * | 2002-04-18 | 2005-11-04 | アストラゼネカ・アクチエボラーグ | フリル化合物 |
| JP2005534624A (ja) * | 2002-04-18 | 2005-11-17 | アストラゼネカ・アクチエボラーグ | 複素環化合物 |
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| WO2005030778A1 (en) * | 2003-09-25 | 2005-04-07 | Astrazeneca Ab | Ligands |
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- 2007-05-14 AR ARP070102066A patent/AR060914A1/es not_active Application Discontinuation
- 2007-05-14 SA SA07280244A patent/SA07280244B1/ar unknown
- 2007-05-15 UY UY30349A patent/UY30349A1/es not_active Application Discontinuation
- 2007-05-16 KR KR1020087027857A patent/KR20090007753A/ko not_active Abandoned
- 2007-05-16 CA CA002652610A patent/CA2652610A1/en not_active Abandoned
- 2007-05-16 EP EP07748149A patent/EP2019831B1/en active Active
- 2007-05-16 JP JP2009510923A patent/JP2009537517A/ja active Pending
- 2007-05-16 MX MX2008014436A patent/MX2008014436A/es not_active Application Discontinuation
- 2007-05-16 BR BRPI0711941-0A patent/BRPI0711941A2/pt not_active IP Right Cessation
- 2007-05-16 AU AU2007250560A patent/AU2007250560B2/en not_active Ceased
- 2007-05-16 RU RU2008143450/04A patent/RU2441007C2/ru not_active IP Right Cessation
- 2007-05-16 CL CL2007001405A patent/CL2007001405A1/es unknown
- 2007-05-16 ES ES07748149T patent/ES2392997T3/es active Active
- 2007-05-16 WO PCT/SE2007/000485 patent/WO2007133155A1/en not_active Ceased
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2008
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- 2008-11-21 NO NO20084915A patent/NO20084915L/no not_active Application Discontinuation
- 2008-12-12 EC EC2008008971A patent/ECSP088971A/es unknown
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2010
- 2010-11-05 US US12/940,449 patent/US20110136804A1/en not_active Abandoned
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005527588A (ja) * | 2002-04-18 | 2005-09-15 | アストラゼネカ・アクチエボラーグ | チエニル化合物 |
| JP2005533012A (ja) * | 2002-04-18 | 2005-11-04 | アストラゼネカ・アクチエボラーグ | フリル化合物 |
| JP2005534624A (ja) * | 2002-04-18 | 2005-11-17 | アストラゼネカ・アクチエボラーグ | 複素環化合物 |
Also Published As
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| ES2392997T3 (es) | 2012-12-17 |
| TW200813067A (en) | 2008-03-16 |
| RU2441007C2 (ru) | 2012-01-27 |
| US20080139600A1 (en) | 2008-06-12 |
| SA07280244B1 (ar) | 2011-06-22 |
| UY30349A1 (es) | 2008-01-02 |
| US7842803B2 (en) | 2010-11-30 |
| MX2008014436A (es) | 2008-11-27 |
| AR060914A1 (es) | 2008-07-23 |
| EP2019831B1 (en) | 2012-09-12 |
| ECSP088971A (es) | 2009-01-30 |
| WO2007133155A1 (en) | 2007-11-22 |
| US20110136804A1 (en) | 2011-06-09 |
| AU2007250560A1 (en) | 2007-11-22 |
| CL2007001405A1 (es) | 2008-01-25 |
| AU2007250560B2 (en) | 2011-06-23 |
| CA2652610A1 (en) | 2007-11-22 |
| EP2019831A4 (en) | 2010-06-09 |
| NO20084915L (no) | 2009-02-13 |
| KR20090007753A (ko) | 2009-01-20 |
| IL195019A0 (en) | 2009-08-03 |
| EP2019831A1 (en) | 2009-02-04 |
| RU2008143450A (ru) | 2010-06-27 |
| BRPI0711941A2 (pt) | 2011-12-13 |
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