JP2009520791A5 - - Google Patents

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Publication number
JP2009520791A5
JP2009520791A5 JP2008546614A JP2008546614A JP2009520791A5 JP 2009520791 A5 JP2009520791 A5 JP 2009520791A5 JP 2008546614 A JP2008546614 A JP 2008546614A JP 2008546614 A JP2008546614 A JP 2008546614A JP 2009520791 A5 JP2009520791 A5 JP 2009520791A5
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JP
Japan
Prior art keywords
hydrogen
compound
ring
methyl
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2008546614A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009520791A (ja
JP5205276B2 (ja
Filing date
Publication date
Priority claimed from GB0526169A external-priority patent/GB0526169D0/en
Priority claimed from GB0620884A external-priority patent/GB0620884D0/en
Application filed filed Critical
Priority claimed from PCT/GB2006/004854 external-priority patent/WO2007072017A2/en
Publication of JP2009520791A publication Critical patent/JP2009520791A/ja
Publication of JP2009520791A5 publication Critical patent/JP2009520791A5/ja
Application granted granted Critical
Publication of JP5205276B2 publication Critical patent/JP5205276B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2008546614A 2005-12-22 2006-12-21 酵素阻害剤 Active JP5205276B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0526169.8 2005-12-22
GB0526169A GB0526169D0 (en) 2005-12-22 2005-12-22 Enzyme inhibitors
GB0620884A GB0620884D0 (en) 2006-10-20 2006-10-20 Enzyme inhibitors
GB0620884.7 2006-10-20
PCT/GB2006/004854 WO2007072017A2 (en) 2005-12-22 2006-12-21 Enzyme inhibitors

Publications (3)

Publication Number Publication Date
JP2009520791A JP2009520791A (ja) 2009-05-28
JP2009520791A5 true JP2009520791A5 (https=) 2010-02-12
JP5205276B2 JP5205276B2 (ja) 2013-06-05

Family

ID=38091678

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008546614A Active JP5205276B2 (ja) 2005-12-22 2006-12-21 酵素阻害剤

Country Status (5)

Country Link
US (1) US8088761B2 (https=)
EP (1) EP1963315B1 (https=)
JP (1) JP5205276B2 (https=)
ES (1) ES2526813T3 (https=)
WO (1) WO2007072017A2 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008121064A1 (en) * 2007-03-30 2008-10-09 Astrazeneca Ab New imidazo[4,5-b]pyridine-6-halo-7-aryl/heteroaryl compounds 705
WO2009001021A1 (en) * 2007-06-26 2008-12-31 Chroma Therapeutics Ltd. Imidazopyridine derivatives useful as enzyme inhibitors for the treatment of cell proliferative and autoimmune diseases
US8987307B2 (en) 2011-03-03 2015-03-24 Hoffmann-La Roche Inc. 3-amino-pyridines as GPBAR1 agonists
ES2567552T3 (es) * 2012-01-30 2016-04-25 Cephalon, Inc. Imidazo [4,5-b] derivados de piridina como los moduladores ALK y JAK para el tratamiento de trastornos proliferativos
AR090789A1 (es) * 2012-04-23 2014-12-10 Genentech Inc Intermediarios y procesos para la preparacion de compuestos
GB201211021D0 (en) * 2012-06-21 2012-08-01 Cancer Rec Tech Ltd Pharmaceutically active compounds
GB201211019D0 (en) * 2012-06-21 2012-08-01 Cancer Rec Tech Ltd Inhibitor compounds
CA2890288A1 (en) * 2012-11-16 2014-05-22 Merck Patent Gmbh Novel heterocyclic derivatives as modulators of kinase activity
UY36390A (es) * 2014-11-05 2016-06-01 Flexus Biosciences Inc Compuestos moduladores de la enzima indolamina 2,3-dioxigenasa (ido), sus métodos de síntesis y composiciones farmacéuticas que los contienen
MX2017005462A (es) 2014-11-05 2017-07-28 Flexus Biosciences Inc Agentes inmunorreguladores.
EP3253754B1 (en) 2015-02-02 2021-03-31 Kancera AB 2-phenyl-3h-imidazo[4,5-b]pyridine derivates useful as inhibitors of mammalian tyrosine kinase ror1 activity
CN109563092B (zh) 2016-07-11 2021-09-14 坎塞拉有限公司 可用作哺乳动物酪氨酸激酶ror1活性的抑制剂的2-苯基咪唑并[4,5-b]吡啶-7-胺衍生物
US11660303B2 (en) 2016-07-11 2023-05-30 Kancera Ab 2-phenylimidazo[4,5-b]pyridin-7-amine derivates useful as inhibitors of mammalian tyrosine kinase ROR1 activity
CN112239465A (zh) 2019-07-16 2021-01-19 微境生物医药科技(上海)有限公司 极光激酶抑制剂及其用途
AR129965A1 (es) * 2022-07-20 2024-10-16 Sanofi Sa Compuestos de imidazopiridina, preparación de los mismos y usos terapéuticos de los mismos
WO2026020051A1 (en) * 2024-07-19 2026-01-22 Nurix Therapeutics, Inc. Bifunctional compounds for degrading aurora kinase via ubiquitin proteosome pathway

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ID24300A (id) * 1997-08-05 2000-07-13 Pfizer Prod Inc 4-AMINOPIROL(3,2-d)PIRIMIDIN SEBAGAI ANTAGONIS-ANTAGONIS RESEPTOR NEUROPEPTIDA Y
JP2004503553A (ja) * 2000-06-14 2004-02-05 ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー 6,5−縮合二環式複素環
SE0202462D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel use
US7534796B2 (en) 2005-02-18 2009-05-19 Wyeth Imidazo[4,5-b]pyridine antagonists of gonadotropin releasing hormone receptor

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